CA2223414A1 - Acides d'heteroaryle diol antagonistes des leucotrienes - Google Patents

Acides d'heteroaryle diol antagonistes des leucotrienes

Info

Publication number
CA2223414A1
CA2223414A1 CA002223414A CA2223414A CA2223414A1 CA 2223414 A1 CA2223414 A1 CA 2223414A1 CA 002223414 A CA002223414 A CA 002223414A CA 2223414 A CA2223414 A CA 2223414A CA 2223414 A1 CA2223414 A1 CA 2223414A1
Authority
CA
Canada
Prior art keywords
heteroaryl
leukotriene antagonists
diol
acids
diol acids
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
CA002223414A
Other languages
English (en)
Other versions
CA2223414C (fr
Inventor
Nathalie Chauret
Claude Dufresne
Yves Gareau
Marc Labelle
Deborah Nicoll-Griffith
Laird Trimble
Xin Xu
James Yergey
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Canada Inc
Original Assignee
Merck Frosst Canada Inc.
Merck Frosst Canada Incorporated
Merck Frosst Canada & Co./Merck Frosst Canada & Cie
Nathalie Chauret
Claude Dufresne
Yves Gareau
Marc Labelle
Deborah Nicoll-Griffith
Laird Trimble
Xin Xu
James Yergey
Merck Frosst Canada Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/475,139 external-priority patent/US5750539A/en
Application filed by Merck Frosst Canada Inc., Merck Frosst Canada Incorporated, Merck Frosst Canada & Co./Merck Frosst Canada & Cie, Nathalie Chauret, Claude Dufresne, Yves Gareau, Marc Labelle, Deborah Nicoll-Griffith, Laird Trimble, Xin Xu, James Yergey, Merck Frosst Canada Ltd. filed Critical Merck Frosst Canada Inc.
Publication of CA2223414A1 publication Critical patent/CA2223414A1/fr
Application granted granted Critical
Publication of CA2223414C publication Critical patent/CA2223414C/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/18—Halogen atoms or nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CA002223414A 1995-06-07 1996-06-03 Acides d'heteroaryle diol antagonistes des leucotrienes Expired - Fee Related CA2223414C (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US475,139 1995-06-07
US08/475,139 US5750539A (en) 1995-06-07 1995-06-07 Heteroaryl diol acids as leukotriene antagonists
PCT/US1996/008446 WO1996040638A1 (fr) 1995-06-07 1996-06-03 Acides d'heteroaryle diol antagonistes des leucotrienes

Publications (2)

Publication Number Publication Date
CA2223414A1 true CA2223414A1 (fr) 1996-12-19
CA2223414C CA2223414C (fr) 2007-08-14

Family

ID=38434464

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002223414A Expired - Fee Related CA2223414C (fr) 1995-06-07 1996-06-03 Acides d'heteroaryle diol antagonistes des leucotrienes

Country Status (1)

Country Link
CA (1) CA2223414C (fr)

Also Published As

Publication number Publication date
CA2223414C (fr) 2007-08-14

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Legal Events

Date Code Title Description
EEER Examination request
MKLA Lapsed