CA2191203A1 - Production modulaire systematique de molecules a base d'aminimide et d'oxazolone possedant au moins deux elements de diversite structurelle - Google Patents

Production modulaire systematique de molecules a base d'aminimide et d'oxazolone possedant au moins deux elements de diversite structurelle

Info

Publication number
CA2191203A1
CA2191203A1 CA002191203A CA2191203A CA2191203A1 CA 2191203 A1 CA2191203 A1 CA 2191203A1 CA 002191203 A CA002191203 A CA 002191203A CA 2191203 A CA2191203 A CA 2191203A CA 2191203 A1 CA2191203 A1 CA 2191203A1
Authority
CA
Canada
Prior art keywords
butyl
methyl
ethyl
molecules
propyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002191203A
Other languages
English (en)
Inventor
Joseph C. Hogan, Jr.
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Arqule Inc
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2191203A1 publication Critical patent/CA2191203A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/28—Nitrogen atoms
    • C07D295/32—Nitrogen atoms acylated with carboxylic or carbonic acids, or their nitrogen or sulfur analogues
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/36—One oxygen atom
    • C07D263/42—One oxygen atom attached in position 5

Abstract

Des molécules à base d'aminimide et d'oxazolone et des assemblages de celles-ci, possédant au moins deux éléments de diversité structurelle, sont obtenues par production modulaire systématique. Une bibliothèque combinatoire de molécules à base d'aminimide et d'oxazolone est créée par production modulaire systématique.
CA002191203A 1994-05-23 1995-05-18 Production modulaire systematique de molecules a base d'aminimide et d'oxazolone possedant au moins deux elements de diversite structurelle Abandoned CA2191203A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24826394A 1994-05-23 1994-05-23
US248,263 1994-05-23

Publications (1)

Publication Number Publication Date
CA2191203A1 true CA2191203A1 (fr) 1995-11-30

Family

ID=22938357

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002191203A Abandoned CA2191203A1 (fr) 1994-05-23 1995-05-18 Production modulaire systematique de molecules a base d'aminimide et d'oxazolone possedant au moins deux elements de diversite structurelle

Country Status (5)

Country Link
EP (1) EP0763015A1 (fr)
JP (1) JPH10500685A (fr)
AU (1) AU2553195A (fr)
CA (1) CA2191203A1 (fr)
WO (1) WO1995032184A1 (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6004823A (en) * 1997-05-07 1999-12-21 Smithkline Beecham Corporation Compounds
US5908960A (en) * 1997-05-07 1999-06-01 Smithkline Beecham Corporation Compounds
US6998249B1 (en) 1999-09-27 2006-02-14 Pharmacia & Upjohn Company Toxicity screening method
EP1406493A4 (fr) 2001-06-11 2006-06-14 Xenoport Inc Administration d'agents via le transporteur de peptides pept-2
US8187874B2 (en) 2003-10-27 2012-05-29 Vertex Pharmaceuticals Incorporated Drug discovery method
ATE535612T1 (de) 2006-03-06 2011-12-15 Ceetox Inc Toxizitätsscreeningverfahren

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2262660A1 (en) * 1974-02-28 1975-09-26 Ici Australia Ltd Tris-(hydroxy-alkyl)-amine-imide surfactants - prepd. by reacting hydrazines with alkylene oxides
US4078901A (en) * 1976-12-20 1978-03-14 Texaco Inc. Detergent fuel composition

Also Published As

Publication number Publication date
AU2553195A (en) 1995-12-18
JPH10500685A (ja) 1998-01-20
WO1995032184A1 (fr) 1995-11-30
EP0763015A1 (fr) 1997-03-19

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Legal Events

Date Code Title Description
FZDE Discontinued
FZDE Discontinued

Effective date: 20000518