CA2079373A1 - (azaarylmethoxy)indoles as inhibitors of leukotriene biosynthesis - Google Patents

(azaarylmethoxy)indoles as inhibitors of leukotriene biosynthesis

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Publication number
CA2079373A1
CA2079373A1 CA002079373A CA2079373A CA2079373A1 CA 2079373 A1 CA2079373 A1 CA 2079373A1 CA 002079373 A CA002079373 A CA 002079373A CA 2079373 A CA2079373 A CA 2079373A CA 2079373 A1 CA2079373 A1 CA 2079373A1
Authority
CA
Canada
Prior art keywords
inhibitors
leukotriene biosynthesis
azaarylmethoxy
indoles
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
CA002079373A
Other languages
French (fr)
Other versions
CA2079373C (en
Inventor
Petpiboon Prasit
John H. Hutchinson
Michel Therien
John W. Gillard
Richard Frenette
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Canada Inc
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2079373A1 publication Critical patent/CA2079373A1/en
Application granted granted Critical
Publication of CA2079373C publication Critical patent/CA2079373C/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Abstract

Compounds having the formula I:
(see formula I) are inhibitors of leukotriene biosynthesis. These compounds are useful as anti-asthmatic, anti-allergic, anti-inflammatory, and cytoprotective agents. They are also useful in treating diarrhea, hypertension, angina, platelet aggregation, cerebral spasm, premature labor, spontaneous abortion, dysmenorrhea, and migraine.
CA002079373A 1991-09-30 1992-09-29 (azaarylmethoxy)indoles as inhibitors of leukotriene biosynthesis Expired - Fee Related CA2079373C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US76814091A 1991-09-30 1991-09-30
US768,140 1991-09-30

Publications (2)

Publication Number Publication Date
CA2079373A1 true CA2079373A1 (en) 1993-03-31
CA2079373C CA2079373C (en) 2003-08-05

Family

ID=25081657

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002079373A Expired - Fee Related CA2079373C (en) 1991-09-30 1992-09-29 (azaarylmethoxy)indoles as inhibitors of leukotriene biosynthesis

Country Status (2)

Country Link
AU (1) AU3153993A (en)
CA (1) CA2079373C (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN112898256A (en) * 2021-01-29 2021-06-04 遵义医科大学 Preparation method of 1, 2-dihydrocyclopenta [ b ] chromene-3, 9-diketone compound

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN112898256A (en) * 2021-01-29 2021-06-04 遵义医科大学 Preparation method of 1, 2-dihydrocyclopenta [ b ] chromene-3, 9-diketone compound
CN112898256B (en) * 2021-01-29 2023-01-31 遵义医科大学 Preparation method of 1, 2-dihydrocyclopenta [ b ] chromene-3, 9-diketone compound

Also Published As

Publication number Publication date
CA2079373C (en) 2003-08-05
AU3153993A (en) 1994-07-04

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