CA1244450A - N-(1-substituted-4,5-dihydro-1h-pyrazol-4-yl) benzamides - Google Patents

N-(1-substituted-4,5-dihydro-1h-pyrazol-4-yl) benzamides

Info

Publication number
CA1244450A
CA1244450A CA000478382A CA478382A CA1244450A CA 1244450 A CA1244450 A CA 1244450A CA 000478382 A CA000478382 A CA 000478382A CA 478382 A CA478382 A CA 478382A CA 1244450 A CA1244450 A CA 1244450A
Authority
CA
Canada
Prior art keywords
amino
compound
acid addition
addition salt
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000478382A
Other languages
English (en)
French (fr)
Inventor
Lennox B. Turnbull
Gunnar E. Jagdmann, Jr.
John A. Donohue
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth LLC
Original Assignee
AH Robins Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by AH Robins Co Inc filed Critical AH Robins Co Inc
Application granted granted Critical
Publication of CA1244450A publication Critical patent/CA1244450A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Otolaryngology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hospice & Palliative Care (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Inks, Pencil-Leads, Or Crayons (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
CA000478382A 1984-04-06 1985-04-04 N-(1-substituted-4,5-dihydro-1h-pyrazol-4-yl) benzamides Expired CA1244450A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/597,421 US4547518A (en) 1984-04-06 1984-04-06 Antiemetic N-(1-substituted-4,5-dihydro-1H-pyrazol-4-yl)benzamides
US597,421 1984-04-06

Publications (1)

Publication Number Publication Date
CA1244450A true CA1244450A (en) 1988-11-08

Family

ID=24391432

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000478382A Expired CA1244450A (en) 1984-04-06 1985-04-04 N-(1-substituted-4,5-dihydro-1h-pyrazol-4-yl) benzamides

Country Status (21)

Country Link
US (1) US4547518A (enEXAMPLES)
EP (1) EP0161074B1 (enEXAMPLES)
JP (1) JPS60228462A (enEXAMPLES)
KR (1) KR900001207B1 (enEXAMPLES)
AT (1) ATE36156T1 (enEXAMPLES)
AU (1) AU569153B2 (enEXAMPLES)
CA (1) CA1244450A (enEXAMPLES)
DE (1) DE3564109D1 (enEXAMPLES)
DK (1) DK154585A (enEXAMPLES)
ES (1) ES541719A0 (enEXAMPLES)
FI (1) FI851389L (enEXAMPLES)
HU (1) HU193329B (enEXAMPLES)
IL (1) IL74423A (enEXAMPLES)
IN (1) IN160249B (enEXAMPLES)
NO (1) NO163365C (enEXAMPLES)
NZ (1) NZ211698A (enEXAMPLES)
PH (1) PH22090A (enEXAMPLES)
PL (1) PL144918B1 (enEXAMPLES)
PT (1) PT80234B (enEXAMPLES)
YU (1) YU49985A (enEXAMPLES)
ZA (1) ZA851193B (enEXAMPLES)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE632034A (enEXAMPLES) * 1962-05-09
DE2428673A1 (de) * 1974-06-14 1976-01-02 Bayer Ag Carbonsaeureamide, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
US4207327A (en) * 1977-08-19 1980-06-10 A. H. Robins Company, Inc. N-(4-Pyrazolidinyl)benzamides and their amino precursors

Also Published As

Publication number Publication date
NO163365B (no) 1990-02-05
FI851389A7 (fi) 1985-10-07
ATE36156T1 (de) 1988-08-15
DK154585D0 (da) 1985-04-03
DE3564109D1 (en) 1988-09-08
ES8602683A1 (es) 1985-12-01
EP0161074B1 (en) 1988-08-03
JPS60228462A (ja) 1985-11-13
FI851389L (fi) 1985-10-07
DK154585A (da) 1985-10-07
NO163365C (no) 1990-05-16
HUT37601A (en) 1986-01-23
ES541719A0 (es) 1985-12-01
AU4090085A (en) 1985-10-10
US4547518A (en) 1985-10-15
NO851352L (no) 1985-10-07
IL74423A0 (en) 1985-05-31
PH22090A (en) 1988-05-20
AU569153B2 (en) 1988-01-21
KR900001207B1 (ko) 1990-02-28
HU193329B (en) 1987-09-28
YU49985A (en) 1988-02-29
IN160249B (enEXAMPLES) 1987-07-04
PL252808A1 (en) 1986-12-30
PL144918B1 (en) 1988-07-30
PT80234B (en) 1986-11-13
FI851389A0 (fi) 1985-04-04
PT80234A (en) 1985-05-01
ZA851193B (en) 1985-10-30
NZ211698A (en) 1988-01-08
KR850007592A (ko) 1985-12-07
IL74423A (en) 1988-12-30
EP0161074A1 (en) 1985-11-13

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Legal Events

Date Code Title Description
MKEX Expiry