CA1120030A - Somatostatin analogs and intermediates thereto - Google Patents

Somatostatin analogs and intermediates thereto

Info

Publication number
CA1120030A
CA1120030A CA000301485A CA301485A CA1120030A CA 1120030 A CA1120030 A CA 1120030A CA 000301485 A CA000301485 A CA 000301485A CA 301485 A CA301485 A CA 301485A CA 1120030 A CA1120030 A CA 1120030A
Authority
CA
Canada
Prior art keywords
phe
resin
acid
tetradecapeptide
lys
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000301485A
Other languages
English (en)
French (fr)
Inventor
James E. Shields
Tsung-Min Lin
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US04/874,173 external-priority patent/US4151394A/en
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Application granted granted Critical
Publication of CA1120030A publication Critical patent/CA1120030A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • C07K14/655Somatostatins
    • C07K14/6555Somatostatins at least 1 amino acid in D-form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Medicinal Chemistry (AREA)
  • Zoology (AREA)
  • Biochemistry (AREA)
  • Toxicology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
CA000301485A 1977-04-21 1978-04-19 Somatostatin analogs and intermediates thereto Expired CA1120030A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US78947377A 1977-04-21 1977-04-21
US789,473 1977-04-21
US04/874,173 US4151394A (en) 1978-02-01 1978-02-01 Guidance system for arc welder
US874,173 1978-02-01

Publications (1)

Publication Number Publication Date
CA1120030A true CA1120030A (en) 1982-03-16

Family

ID=27120917

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000301485A Expired CA1120030A (en) 1977-04-21 1978-04-19 Somatostatin analogs and intermediates thereto

Country Status (23)

Country Link
JP (1) JPS53132589A (xx)
AR (1) AR229798A1 (xx)
AT (1) AT360675B (xx)
AU (1) AU518731B2 (xx)
BG (2) BG28705A4 (xx)
CA (1) CA1120030A (xx)
CH (1) CH634040A5 (xx)
DD (1) DD136739A5 (xx)
DE (1) DE2816855A1 (xx)
DK (1) DK174178A (xx)
EG (1) EG14800A (xx)
ES (2) ES469004A1 (xx)
FI (1) FI64575C (xx)
FR (1) FR2387942A1 (xx)
GB (1) GB1596329A (xx)
GR (1) GR69789B (xx)
IE (1) IE46617B1 (xx)
IL (1) IL54532A (xx)
IT (1) IT1094471B (xx)
NL (1) NL7804219A (xx)
NZ (1) NZ187010A (xx)
PT (1) PT67912B (xx)
SE (1) SE7804398L (xx)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8423431D0 (en) * 1984-09-17 1984-10-24 Sandoz Ltd Organic compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2608336A1 (de) * 1975-03-11 1976-09-30 Sandoz Ag Neue organische verbindungen, ihre herstellung und verwendung
US4372884A (en) * 1975-08-06 1983-02-08 The Salk Institute For Biological Studies Pharmaceutically active peptides

Also Published As

Publication number Publication date
GB1596329A (en) 1981-08-26
CH634040A5 (en) 1983-01-14
AT360675B (de) 1981-01-26
SE7804398L (sv) 1978-10-22
IT1094471B (it) 1985-08-02
FI781183A (fi) 1978-10-22
DD136739A5 (de) 1979-07-25
FI64575C (fi) 1983-12-12
DE2816855A1 (de) 1978-11-02
ATA282978A (de) 1980-06-15
NL7804219A (nl) 1978-10-24
IE780766L (en) 1978-10-21
DK174178A (da) 1978-10-22
IL54532A (en) 1983-03-31
GR69789B (xx) 1982-07-07
PT67912B (en) 1979-11-14
IE46617B1 (en) 1983-08-10
ES476913A1 (es) 1979-09-16
BG28704A3 (en) 1980-06-16
AR229798A1 (es) 1983-11-30
AU3534178A (en) 1979-10-25
FR2387942A1 (fr) 1978-11-17
FR2387942B1 (xx) 1981-06-26
ES469004A1 (es) 1979-09-01
NZ187010A (en) 1980-08-26
IL54532A0 (en) 1978-07-31
JPS53132589A (en) 1978-11-18
BG28705A4 (en) 1980-06-16
FI64575B (fi) 1983-08-31
AU518731B2 (en) 1981-10-15
IT7822553A0 (it) 1978-04-20
PT67912A (en) 1978-05-01
EG14800A (en) 1985-06-30

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Legal Events

Date Code Title Description
MKEX Expiry