CA1117533A - Benzisothiazole-1,1-dioxides - Google Patents

Benzisothiazole-1,1-dioxides

Info

Publication number
CA1117533A
CA1117533A CA000317751A CA317751A CA1117533A CA 1117533 A CA1117533 A CA 1117533A CA 000317751 A CA000317751 A CA 000317751A CA 317751 A CA317751 A CA 317751A CA 1117533 A CA1117533 A CA 1117533A
Authority
CA
Canada
Prior art keywords
hydrogen
halogen
compound
lower alkyl
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000317751A
Other languages
English (en)
French (fr)
Inventor
Peter C. Wade
Berthold R. Vogt
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/875,022 external-priority patent/US4148798A/en
Priority claimed from US05/924,340 external-priority patent/US4147698A/en
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Application granted granted Critical
Publication of CA1117533A publication Critical patent/CA1117533A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D275/06—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA000317751A 1978-02-03 1978-12-12 Benzisothiazole-1,1-dioxides Expired CA1117533A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US875,022 1978-02-03
US05/875,022 US4148798A (en) 1978-02-03 1978-02-03 [(1,1-dioxo-1,2-benzisothiazol-3-yl)amino]alkanoic acids and esters thereof
US05/924,340 US4147698A (en) 1978-07-13 1978-07-13 3-(Heterocyclicalkylamino)benzisothiazole-1,1-dioxides
US924,340 1978-07-13

Publications (1)

Publication Number Publication Date
CA1117533A true CA1117533A (en) 1982-02-02

Family

ID=27128366

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000317751A Expired CA1117533A (en) 1978-02-03 1978-12-12 Benzisothiazole-1,1-dioxides

Country Status (6)

Country Link
JP (1) JPS54106464A (enrdf_load_stackoverflow)
CA (1) CA1117533A (enrdf_load_stackoverflow)
DE (1) DE2856528A1 (enrdf_load_stackoverflow)
FR (1) FR2416226A1 (enrdf_load_stackoverflow)
GB (1) GB2013654B (enrdf_load_stackoverflow)
IT (1) IT1160414B (enrdf_load_stackoverflow)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4748182A (en) * 1986-03-05 1988-05-31 Merrell Dow Pharmaceuticals Inc. Aromatic 2-aminoalkyl-1,2-benzoisothiazol-3(2H)one-1,1-dioxide derivatives and their use as anti-hypertensive and anxiolytic agents
JP6078338B2 (ja) * 2010-04-02 2017-02-08 住友精化株式会社 ３−ハロ−１，２−ベンゾイソチアゾール類の製造方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2751392A (en) * 1953-11-23 1956-06-19 Geschickter Fund Med Res Tertiary amine derivatives of nu-and omicron-saccharin
DE1670797A1 (de) * 1967-02-10 1971-03-25 Hoechst Ag Benzisothiazol-1,1-dioxyde und Verfahren zu ihrer Herstellung
US4104387A (en) * 1977-05-23 1978-08-01 E. R. Squibb & Sons, Inc. 3-(Arylcycloiminoalkyl)benzisothiazole 1,1-dioxides

Also Published As

Publication number Publication date
FR2416226A1 (fr) 1979-08-31
JPS54106464A (en) 1979-08-21
GB2013654B (en) 1982-07-14
GB2013654A (en) 1979-08-15
DE2856528A1 (de) 1979-08-09
FR2416226B1 (enrdf_load_stackoverflow) 1981-08-14
IT1160414B (it) 1987-03-11
IT7831384A0 (it) 1978-12-28

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Legal Events

Date Code Title Description
MKEX Expiry
MKEX Expiry

Effective date: 19990202