CA1117533A - Benzisothiazole-1,1-dioxides - Google Patents

Benzisothiazole-1,1-dioxides

Info

Publication number
CA1117533A
CA1117533A CA000317751A CA317751A CA1117533A CA 1117533 A CA1117533 A CA 1117533A CA 000317751 A CA000317751 A CA 000317751A CA 317751 A CA317751 A CA 317751A CA 1117533 A CA1117533 A CA 1117533A
Authority
CA
Canada
Prior art keywords
hydrogen
halogen
compound
lower alkyl
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000317751A
Other languages
English (en)
French (fr)
Inventor
Peter C. Wade
Berthold R. Vogt
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/875,022 external-priority patent/US4148798A/en
Priority claimed from US05/924,340 external-priority patent/US4147698A/en
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Application granted granted Critical
Publication of CA1117533A publication Critical patent/CA1117533A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D275/06—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA000317751A 1978-02-03 1978-12-12 Benzisothiazole-1,1-dioxides Expired CA1117533A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US05/875,022 US4148798A (en) 1978-02-03 1978-02-03 [(1,1-dioxo-1,2-benzisothiazol-3-yl)amino]alkanoic acids and esters thereof
US875,022 1978-02-03
US924,340 1978-07-13
US05/924,340 US4147698A (en) 1978-07-13 1978-07-13 3-(Heterocyclicalkylamino)benzisothiazole-1,1-dioxides

Publications (1)

Publication Number Publication Date
CA1117533A true CA1117533A (en) 1982-02-02

Family

ID=27128366

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000317751A Expired CA1117533A (en) 1978-02-03 1978-12-12 Benzisothiazole-1,1-dioxides

Country Status (6)

Country Link
JP (1) JPS54106464A (enrdf_load_stackoverflow)
CA (1) CA1117533A (enrdf_load_stackoverflow)
DE (1) DE2856528A1 (enrdf_load_stackoverflow)
FR (1) FR2416226A1 (enrdf_load_stackoverflow)
GB (1) GB2013654B (enrdf_load_stackoverflow)
IT (1) IT1160414B (enrdf_load_stackoverflow)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4748182A (en) * 1986-03-05 1988-05-31 Merrell Dow Pharmaceuticals Inc. Aromatic 2-aminoalkyl-1,2-benzoisothiazol-3(2H)one-1,1-dioxide derivatives and their use as anti-hypertensive and anxiolytic agents
ES2530523T3 (es) * 2010-04-02 2015-03-03 Sumitomo Seika Chemicals Método para producir 3-halo-1,2-benzoisotiazoles

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2751392A (en) * 1953-11-23 1956-06-19 Geschickter Fund Med Res Tertiary amine derivatives of nu-and omicron-saccharin
DE1670797A1 (de) * 1967-02-10 1971-03-25 Hoechst Ag Benzisothiazol-1,1-dioxyde und Verfahren zu ihrer Herstellung
US4104387A (en) * 1977-05-23 1978-08-01 E. R. Squibb & Sons, Inc. 3-(Arylcycloiminoalkyl)benzisothiazole 1,1-dioxides

Also Published As

Publication number Publication date
GB2013654B (en) 1982-07-14
FR2416226A1 (fr) 1979-08-31
GB2013654A (en) 1979-08-15
JPS54106464A (en) 1979-08-21
FR2416226B1 (enrdf_load_stackoverflow) 1981-08-14
DE2856528A1 (de) 1979-08-09
IT1160414B (it) 1987-03-11
IT7831384A0 (it) 1978-12-28

Similar Documents

Publication Publication Date Title
CA1274523A (en) Thiazolidine derivatives, their production and use
US3822258A (en) 4-hydroxy-3-(3-isoxazolylcarbamoyl)-2h-1,2-benzothiazine 1,1-dioxides and process for their production
FI86064C (fi) Foerfarande foer framstaellning av nya terapeutiskt anvaendbara aminotiazol- och aminooxazolderivat.
US3905984A (en) Pyridyl substituted thioalkyl-and oxyalkyl-thioureas and ureas
US4242507A (en) Sulfonic acid esters
CS207791B2 (en) Method of making the derivatives of the thiadiazole
EP0279598B1 (en) Arylpiperazinyl-alkylene-phenyl-heterocyclic compounds
IE41457B1 (en) Thienothiazine derivatives
SK278349B6 (en) 2-iminobenzothiazoline derivative, preparation method thereof and pharmaceutical agent containing this derivative
US4147698A (en) 3-(Heterocyclicalkylamino)benzisothiazole-1,1-dioxides
CA1117533A (en) Benzisothiazole-1,1-dioxides
US4104388A (en) 3-Substituted benzisothiazole, 1,1-dioxides
US5026717A (en) 2-imino-6-polyfluoroalkoxybenzothiazole derivatives, and pharmaceutical compositions containing them
EP0010398B1 (en) Isatin derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same
CA2140006A1 (en) Thiazoline derivatives
CA1048025A (en) 4-hydroxy-2h-naphtho (2,1-e)-1,2-thiazine-3-carboxamide-1,1-dioxides, processes for their preparation and pharmaceuticals containing them
CA1175842A (en) 2,3-di-substituted-5,6-dihydroimidazo ¬2,1-b| thiazole, its salts, production thereof and anti- inflammatory agent containing the same
DE69226931T2 (de) Guanidinothiazolederivate und ihre Anwendung als H2-Rezeptor-Antagonisten
US4104387A (en) 3-(Arylcycloiminoalkyl)benzisothiazole 1,1-dioxides
US3925369A (en) New tricyclic ureas processes for their production and pharmaceutical compositions
CA1038379A (en) Acylated 2-aminothiazole derivatives and a process for the preparation thereof
CA1244827A (en) Process for preparing 4,5,6,7-tetrahydro-thiazolo ¬5,4-c|-pyridine derivatives
US4246260A (en) Substituted omicron-phenylenediamine derivatives, process for their preparation and their use as medicaments
CA1201119A (en) Diaza-cyclic derivatives of guanidine
US4178451A (en) 3-(Substituted hydrazino)benzisothiazole-1,1-dioxides

Legal Events

Date Code Title Description
MKEX Expiry
MKEX Expiry

Effective date: 19990202