CA1094063A - Agents anti-allergenes a base de thieno ¬2,3-d| pyrimidine - Google Patents

Agents anti-allergenes a base de thieno ¬2,3-d| pyrimidine

Info

Publication number
CA1094063A
CA1094063A CA288,853A CA288853A CA1094063A CA 1094063 A CA1094063 A CA 1094063A CA 288853 A CA288853 A CA 288853A CA 1094063 A CA1094063 A CA 1094063A
Authority
CA
Canada
Prior art keywords
formula
procedure
compound
pyrimidine
ethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA288,853A
Other languages
English (en)
Inventor
Davis L. Temple, Jr.
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Squibb Co
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/826,591 external-priority patent/US4159377A/en
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Application granted granted Critical
Publication of CA1094063A publication Critical patent/CA1094063A/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
CA288,853A 1977-08-22 1977-10-17 Agents anti-allergenes a base de thieno ¬2,3-d| pyrimidine Expired CA1094063A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/826,591 US4159377A (en) 1975-09-10 1977-08-22 Selected thieno[2,3-d]pyrimidines
US826,591 1977-08-22

Publications (1)

Publication Number Publication Date
CA1094063A true CA1094063A (fr) 1981-01-20

Family

ID=25246995

Family Applications (1)

Application Number Title Priority Date Filing Date
CA288,853A Expired CA1094063A (fr) 1977-08-22 1977-10-17 Agents anti-allergenes a base de thieno ¬2,3-d| pyrimidine

Country Status (2)

Country Link
CA (1) CA1094063A (fr)
FR (3) FR2401163A1 (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4761474A (en) * 1986-02-25 1988-08-02 Merrell Dow Pharmaceuticals Inc. 3-(1H-tetrazol-5-yl)thieno[2,3-d]pyrimidin-4(3H)-ones
GB9426021D0 (en) * 1994-12-22 1995-02-22 Smithkline Beecham Plc Pharmaceuticals
AU1595997A (en) * 1996-01-26 1997-08-20 Smithkline Beecham Plc Thienoxazinone derivatives useful as antiviral agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2035767A1 (fr) * 1969-03-07 1970-12-24 Centre Etd Ind Pharma
FR2121341A1 (en) * 1971-01-04 1972-08-25 Ferlux 2-substd-3,1-benzoxazin-4-ones - antiinflammatories, analgesics sedatives and diuretics
GB1468012A (en) * 1973-08-09 1977-03-23 Beecham Group Ltd 2-amino-3-carboxy-thiophene derivatives
BE859818A (fr) * 1977-10-17 1978-04-17 Bristol Myers Co Thieno(2,3-d)pyrimidines antiallergiques

Also Published As

Publication number Publication date
FR2401152A1 (fr) 1979-03-23
FR2401164A1 (fr) 1979-03-23
FR2401163B1 (fr) 1982-04-02
FR2401152B1 (fr) 1982-04-02
FR2401163A1 (fr) 1979-03-23
FR2401164B1 (fr) 1982-04-02

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JP2514812B2 (ja) ３−（１Ｈ−テトラゾ−ル−５− イル） チエノ〔２，３−ｄ〕 ピリミジン−４（３Ｈ）−オン類

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