CA1091230A - Derives des acides 7-acylamino-8-oxo-3-oxa-1- azabicyclo-¬4.2.0|octane-2-carboxyliques - Google Patents
Derives des acides 7-acylamino-8-oxo-3-oxa-1- azabicyclo-¬4.2.0|octane-2-carboxyliquesInfo
- Publication number
- CA1091230A CA1091230A CA286,049A CA286049A CA1091230A CA 1091230 A CA1091230 A CA 1091230A CA 286049 A CA286049 A CA 286049A CA 1091230 A CA1091230 A CA 1091230A
- Authority
- CA
- Canada
- Prior art keywords
- oxo
- cis
- acid
- solution
- azido
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C07D205/085—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/721,251 US4089956A (en) | 1976-09-08 | 1976-09-08 | 7-Acylamino-8-oxo-3-oxa-1-azabicyclo[4.2.0]octane-2-carboxylic acid derivatives and bactericidal compositions and use thereof |
| US721,251 | 1985-04-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA1091230A true CA1091230A (fr) | 1980-12-09 |
Family
ID=24897172
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA286,049A Expired CA1091230A (fr) | 1976-09-08 | 1977-09-02 | Derives des acides 7-acylamino-8-oxo-3-oxa-1- azabicyclo-¬4.2.0|octane-2-carboxyliques |
Country Status (22)
| Country | Link |
|---|---|
| US (2) | US4089956A (fr) |
| JP (1) | JPS5334797A (fr) |
| AT (1) | AT354626B (fr) |
| AU (1) | AU508738B2 (fr) |
| BE (1) | BE858356A (fr) |
| CA (1) | CA1091230A (fr) |
| CH (1) | CH631987A5 (fr) |
| DE (1) | DE2740280A1 (fr) |
| DK (1) | DK394177A (fr) |
| ES (1) | ES462173A1 (fr) |
| FI (1) | FI772628A (fr) |
| FR (2) | FR2372165B1 (fr) |
| GB (2) | GB1592332A (fr) |
| IE (1) | IE46153B1 (fr) |
| IL (1) | IL52878A0 (fr) |
| LU (1) | LU78079A1 (fr) |
| NL (1) | NL7709788A (fr) |
| NO (1) | NO773081L (fr) |
| PH (1) | PH14942A (fr) |
| PT (1) | PT67004B (fr) |
| SE (1) | SE7710114L (fr) |
| ZA (1) | ZA774803B (fr) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4187375A (en) * | 1976-09-08 | 1980-02-05 | Smithkline Corporation | Process for preparing oxazine ring compounds |
| US4264597A (en) * | 1978-06-06 | 1981-04-28 | Masashi Hashimoto | Cephalosporin analogues and processes for the preparation thereof |
| JPS565457A (en) * | 1979-06-27 | 1981-01-20 | Dai Ichi Seiyaku Co Ltd | Thienamycin intermediate |
| US4400323A (en) * | 1979-07-23 | 1983-08-23 | Merck & Co., Inc. | 3-[1-Hydroxyethyl]-4-carboxymethyl-azetidin-2-one |
| NO802713L (no) * | 1979-09-13 | 1981-03-16 | Kyowa Hakko Kogyo Kk | Fremgangsmaate til fremstilling av racemiske eller optisk aktive cefalosporin-analoge karbacefemforbindelser eller farmaseutisk akseptable salter derav |
| US4663450A (en) * | 1979-10-25 | 1987-05-05 | Kyowa Hakko Kogyo Co., Ltd. | Optically active cephalosporin analogs |
| US4287123A (en) * | 1980-01-14 | 1981-09-01 | Merck & Co., Inc. | Synthesis of thienamycin via (3SR, 4RS)-3-((RS)-1-acyloxyethyl)-2-oxo-4-azetidineacetate |
| US4309346A (en) * | 1980-03-27 | 1982-01-05 | Merck & Co., Inc. | Process for the preparation of 1-carbapenems and intermediates via trithioorthoacetates |
| EP0067517B1 (fr) * | 1981-05-14 | 1986-02-26 | Beecham Group Plc | Procédé de préparation d'un énantiomère d'un dérivé béta-lactame |
| JPS5976056A (ja) * | 1982-10-21 | 1984-04-28 | Kanegafuchi Chem Ind Co Ltd | ３−アミノアゼチジン−２−オン及びその製造法 |
| JPS59231090A (ja) * | 1983-06-14 | 1984-12-25 | Shionogi & Co Ltd | フルオロメチルチオオキサセフアロスポリン |
| JPH0730190Y2 (ja) * | 1990-02-28 | 1995-07-12 | 利和 奥野 | コイリングマシン |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1914366A1 (de) * | 1969-03-21 | 1970-10-01 | Bayer Ag | Arzneimittel auf Basis neuer,heterocyclischer Verbindungen |
| US3769277A (en) * | 1970-01-23 | 1973-10-30 | Glaxo Lab Ltd | Preparation of delta3-4 carboxy cephalosporins having a 3-vinyl or substituted 3-vinyl group |
| DE2046823A1 (de) * | 1970-09-23 | 1972-03-30 | Farbwerke Hoechst AG vormals Meister Lucius & Brüning, 6000 Frankfurt | Neue Azetidinone-(2) und Verfahren zu deren Herstellung |
| US3728342A (en) * | 1970-12-03 | 1973-04-17 | Lilly Co Eli | 3-acyloxymethyl cephalosporins and method of preparation |
| US3795672A (en) * | 1971-06-09 | 1974-03-05 | Lilly Co Eli | Process for the preparation of delta2-cephem-4-carboxylic acid esters |
| NL178005C (nl) * | 1972-11-06 | 1986-01-02 | Merck & Co Inc | Werkwijze voor het bereiden van een farmaceutisch preparaat met antibacteriele werking, alsmede werkwijze ter bereiding van een cefalosporine-antibioticum. |
| NL7314706A (fr) * | 1972-11-06 | 1974-05-08 | ||
| GB1510794A (en) * | 1974-08-06 | 1978-05-17 | Univ Kingston | 1-oxacephems and intermediates therefor |
| US4012383A (en) * | 1975-01-02 | 1977-03-15 | Bristol-Myers Company | Δ2,3 -1,4-morpholine-2-carboxylic acids and derivatives thereof useful in preparation of antibacteria agents |
| US4011216A (en) * | 1975-04-11 | 1977-03-08 | Bristol-Myers Company | Δ2,3-0-2-Isocephem-4-carboxylic acid and derivatives thereof as antibacterial agents |
| US4013648A (en) * | 1975-07-23 | 1977-03-22 | Bristol-Myers Company | Δ2,3 -0-2-Isocephem-4-carboxylic acid and derivatives as antibacterial agents |
| US4017143A (en) * | 1975-12-16 | 1977-04-12 | Litton Systems, Inc. | Solderless electrical contact |
-
1976
- 1976-09-08 US US05/721,251 patent/US4089956A/en not_active Expired - Lifetime
-
1977
- 1977-08-08 US US05/822,774 patent/US4122262A/en not_active Expired - Lifetime
- 1977-08-09 ZA ZA00774803A patent/ZA774803B/xx unknown
- 1977-08-31 GB GB36301/77A patent/GB1592332A/en not_active Expired
- 1977-08-31 GB GB15584/80A patent/GB1592333A/en not_active Expired
- 1977-09-01 FR FR7726555A patent/FR2372165B1/fr not_active Expired
- 1977-09-01 AU AU28481/77A patent/AU508738B2/en not_active Expired
- 1977-09-01 PH PH20180A patent/PH14942A/en unknown
- 1977-09-02 IL IL52878A patent/IL52878A0/xx unknown
- 1977-09-02 BE BE180637A patent/BE858356A/fr not_active IP Right Cessation
- 1977-09-02 CA CA286,049A patent/CA1091230A/fr not_active Expired
- 1977-09-05 FI FI772628A patent/FI772628A/fi not_active Application Discontinuation
- 1977-09-05 DK DK394177A patent/DK394177A/da unknown
- 1977-09-06 NO NO773081A patent/NO773081L/no unknown
- 1977-09-06 LU LU78079A patent/LU78079A1/xx unknown
- 1977-09-06 AT AT639977A patent/AT354626B/de not_active IP Right Cessation
- 1977-09-06 NL NL7709788A patent/NL7709788A/xx not_active Application Discontinuation
- 1977-09-06 PT PT67004A patent/PT67004B/fr unknown
- 1977-09-06 JP JP10766577A patent/JPS5334797A/ja active Pending
- 1977-09-07 ES ES462173A patent/ES462173A1/es not_active Expired
- 1977-09-07 CH CH1097077A patent/CH631987A5/de not_active IP Right Cessation
- 1977-09-07 IE IE1856/77A patent/IE46153B1/en unknown
- 1977-09-07 DE DE19772740280 patent/DE2740280A1/de not_active Ceased
- 1977-09-08 SE SE7710114A patent/SE7710114L/xx not_active Application Discontinuation
-
1978
- 1978-01-27 FR FR7802279A patent/FR2375239A1/fr active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| DE2740280A1 (de) | 1978-03-09 |
| IE46153L (en) | 1978-03-08 |
| FI772628A (fi) | 1978-03-09 |
| AT354626B (de) | 1979-01-25 |
| SE7710114L (sv) | 1978-03-09 |
| US4089956A (en) | 1978-05-16 |
| PH14942A (en) | 1982-02-02 |
| AU2848177A (en) | 1979-03-08 |
| PT67004B (fr) | 1979-02-12 |
| FR2372165A1 (fr) | 1978-06-23 |
| FR2375239B1 (fr) | 1980-07-18 |
| ES462173A1 (es) | 1978-06-16 |
| GB1592332A (en) | 1981-07-08 |
| IE46153B1 (en) | 1983-03-09 |
| FR2375239A1 (fr) | 1978-07-21 |
| GB1592333A (en) | 1981-07-08 |
| NO773081L (no) | 1978-03-09 |
| JPS5334797A (en) | 1978-03-31 |
| PT67004A (fr) | 1977-10-01 |
| FR2372165B1 (fr) | 1980-07-18 |
| ZA774803B (en) | 1978-06-28 |
| NL7709788A (nl) | 1978-03-10 |
| DK394177A (da) | 1978-03-09 |
| CH631987A5 (de) | 1982-09-15 |
| BE858356A (fr) | 1978-03-02 |
| US4122262A (en) | 1978-10-24 |
| AU508738B2 (en) | 1980-04-03 |
| IL52878A0 (en) | 1977-11-30 |
| ATA639977A (de) | 1979-06-15 |
| LU78079A1 (fr) | 1978-01-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MKEX | Expiry |