CA1083152A - Agents therapeutiques a base de phenyl-tetrazolyl- pyrimidin-4-one - Google Patents

Agents therapeutiques a base de phenyl-tetrazolyl- pyrimidin-4-one

Info

Publication number
CA1083152A
CA1083152A CA271,406A CA271406A CA1083152A CA 1083152 A CA1083152 A CA 1083152A CA 271406 A CA271406 A CA 271406A CA 1083152 A CA1083152 A CA 1083152A
Authority
CA
Canada
Prior art keywords
integer
alkyl
mixture
oxo
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA271,406A
Other languages
English (en)
Inventor
Peter F. Juby
Richard A. Partyka
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Squibb Co
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/748,851 external-priority patent/US4082751A/en
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Application granted granted Critical
Publication of CA1083152A publication Critical patent/CA1083152A/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C07D239/36—One oxygen atom as doubly bound oxygen atom or as unsubstituted hydroxy radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA271,406A 1976-02-13 1977-02-09 Agents therapeutiques a base de phenyl-tetrazolyl- pyrimidin-4-one Expired CA1083152A (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US65778776A 1976-02-13 1976-02-13
US657,787 1976-02-13
US748,851 1976-12-08
US05/748,851 US4082751A (en) 1976-02-13 1976-12-08 Therapeutic agents

Publications (1)

Publication Number Publication Date
CA1083152A true CA1083152A (fr) 1980-08-05

Family

ID=27097492

Family Applications (1)

Application Number Title Priority Date Filing Date
CA271,406A Expired CA1083152A (fr) 1976-02-13 1977-02-09 Agents therapeutiques a base de phenyl-tetrazolyl- pyrimidin-4-one

Country Status (14)

Country Link
JP (1) JPS52118481A (fr)
AU (1) AU508970B2 (fr)
CA (1) CA1083152A (fr)
CH (1) CH635339A5 (fr)
DE (1) DE2705609A1 (fr)
DK (1) DK149044C (fr)
FI (1) FI62533C (fr)
FR (1) FR2340943A1 (fr)
GB (1) GB1541351A (fr)
IE (1) IE44603B1 (fr)
LU (1) LU76722A1 (fr)
NL (1) NL173055C (fr)
SE (1) SE433494B (fr)
YU (1) YU41567B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4419357A (en) * 1982-01-18 1983-12-06 The Dow Chemical Company 3-(1H-Tetrazol-5-yl)-4(3H)-quinazolinones
CN101747282A (zh) * 2008-12-10 2010-06-23 上海特化医药科技有限公司 一类含有嘧啶酮苯基的化合物、其药物组合物及其制备方法和用途

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3883653A (en) * 1972-10-24 1975-05-13 Pfizer Method of preventing asthmatic symptoms

Also Published As

Publication number Publication date
NL173055B (nl) 1983-07-01
NL7701483A (nl) 1977-08-16
LU76722A1 (fr) 1977-08-18
DK57377A (da) 1977-08-14
IE44603B1 (en) 1982-01-27
DK149044C (da) 1986-06-02
FR2340943B1 (fr) 1981-01-09
CH635339A5 (en) 1983-03-31
YU35477A (en) 1982-10-31
YU41567B (en) 1987-10-31
SE7701552L (sv) 1977-09-23
JPS52118481A (en) 1977-10-04
FI62533B (fi) 1982-09-30
DE2705609A1 (de) 1977-08-25
GB1541351A (en) 1979-02-28
FI62533C (fi) 1983-01-10
AU508970B2 (en) 1980-04-17
AU2189577A (en) 1978-08-10
JPS6139947B2 (fr) 1986-09-06
FI770427A (fr) 1977-08-14
FR2340943A1 (fr) 1977-09-09
SE433494B (sv) 1984-05-28
IE44603L (en) 1977-08-13
NL173055C (nl) 1983-12-01
DK149044B (da) 1985-12-30
DE2705609C2 (fr) 1988-12-15

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Legal Events

Date Code Title Description
MKEX Expiry