CA1055927A - Method for preparation of aminomethylaryl-methylpenicillin derivatives - Google Patents

Method for preparation of aminomethylaryl-methylpenicillin derivatives

Info

Publication number
CA1055927A
CA1055927A CA238,728A CA238728A CA1055927A CA 1055927 A CA1055927 A CA 1055927A CA 238728 A CA238728 A CA 238728A CA 1055927 A CA1055927 A CA 1055927A
Authority
CA
Canada
Prior art keywords
acid
ester
aminomethyl
penicillanic acid
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA238,728A
Other languages
English (en)
French (fr)
Other versions
CA238728S (en
Inventor
James W. Mcfarland
Colin Thomson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Ltd Great Britain
Original Assignee
Pfizer Ltd Great Britain
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd Great Britain filed Critical Pfizer Ltd Great Britain
Application granted granted Critical
Publication of CA1055927A publication Critical patent/CA1055927A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA238,728A 1974-11-12 1975-10-31 Method for preparation of aminomethylaryl-methylpenicillin derivatives Expired CA1055927A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/523,024 US3966710A (en) 1974-11-12 1974-11-12 Aminomethylarylmethylpenicillin derivatives

Publications (1)

Publication Number Publication Date
CA1055927A true CA1055927A (en) 1979-06-05

Family

ID=24083369

Family Applications (1)

Application Number Title Priority Date Filing Date
CA238,728A Expired CA1055927A (en) 1974-11-12 1975-10-31 Method for preparation of aminomethylaryl-methylpenicillin derivatives

Country Status (14)

Country Link
US (1) US3966710A (https=)
AR (1) AR210746A1 (https=)
AU (1) AU472498B2 (https=)
BE (1) BE835411A (https=)
CA (1) CA1055927A (https=)
DE (1) DE2550010C3 (https=)
DK (1) DK143405C (https=)
ES (1) ES442514A1 (https=)
FR (1) FR2290899A1 (https=)
GB (1) GB1470289A (https=)
IE (1) IE41862B1 (https=)
LU (1) LU73784A1 (https=)
NL (1) NL7513174A (https=)
SE (1) SE423815B (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4118563A (en) * 1977-11-25 1978-10-03 Bristol-Myers Company Production of 7-(2-aminomethylphenylacetamido-3-(1-carboxymethyltetrazol-5-ylthiomethyl)-3-cephem-4-carboxylic acid
US4197240A (en) * 1977-12-23 1980-04-08 Yeda Research And Development Co. Ltd. Penicillin derivatives
US4308259A (en) * 1979-03-01 1981-12-29 Beecham Group Limited Penicillin derivatives

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1057029A (en) * 1962-10-24 1967-02-01 Distillers Co Yeast Ltd New penicillins

Also Published As

Publication number Publication date
US3966710A (en) 1976-06-29
AU472498B2 (en) 1976-05-27
IE41862L (en) 1976-05-12
ES442514A1 (es) 1977-04-16
BE835411A (fr) 1976-05-10
SE423815B (sv) 1982-06-07
IE41862B1 (en) 1980-04-09
FR2290899B1 (https=) 1978-11-10
SE7512658L (sv) 1976-05-13
DK143405B (da) 1981-08-17
DE2550010B2 (de) 1979-01-04
NL7513174A (nl) 1976-05-14
LU73784A1 (https=) 1976-09-06
DK143405C (da) 1981-12-14
GB1470289A (en) 1977-04-14
FR2290899A1 (fr) 1976-06-11
DE2550010C3 (de) 1979-09-13
AR210746A1 (es) 1977-09-15
DE2550010A1 (de) 1976-05-13
DK507275A (da) 1976-05-13
AU8653475A (en) 1976-05-27

Similar Documents

Publication Publication Date Title
US4389408A (en) Novel ampicillin esters and production thereof
US4263302A (en) Quinolinecarboxylic acid substituted penicillins and pharmaceutical compositions containing the same
US5830889A (en) Antibacterial penem esters derivatives
CA1055927A (en) Method for preparation of aminomethylaryl-methylpenicillin derivatives
US3997527A (en) Aminomethylarylmethylpenicillin derivatives
US4009160A (en) Aminomethylarylmethylpenicillin derivatives
JPS5917117B2 (ja) 抗菌剤の製法
CA1197840A (en) Penicillin derivatives and process for preparation of the same
US3838153A (en) 6-(alpha-(guanylureidoalkanoylamino)aracylamino)penicillanic acids
US3759898A (en) Synthesis of alpha-(carbo(5-indanyloxy)) benzylpenicillin
US3899394A (en) Production of antibacterial agents
US3819601A (en) Alpha-carboxy-2-thienylmethylpenicillin and cephalosporin and esters and salts thereof
US4311842A (en) Cephalosporin compounds
US3835115A (en) Alpha-(substituted sulfonamido)arylmethylpenicillins
US3781277A (en) Dioxo-thiazolidinyl derivatives of 6-aminopenicillanic acid
DE2600842A1 (de) Neue penicillin-derivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
CA1104562A (en) Cephalosporins, processes for their preparation and their use as medicaments
AU613649B2 (en) Compositions and methods for promoting growth of animals
US3898240A (en) Alpha-amino-omega-aralkylimino penicillanic acids
FI56840C (fi) Foerfarande foer framstaellning av saosom antibakteriska aemnen anvaendbara 6-(2-fenyl-2-(amidino- och imidoylamino-alkanoylamino)acetamido)penicillansyror
JPS6043072B2 (ja) ペニシリンの製造方法
US4454128A (en) 6α-Methoxy-penicillins
US4091215A (en) 7-D-α-Amino-.alpha.-(p-acetoxyphenyl)acetamido-3-methyl-3-cephem-4-carboxylic acid
US3819600A (en) Alpha-carboxamido acyl derivatives of penicillin
US3728334A (en) 6-(1-carboxycycloalkylcarboxamido)penicillanic acid,derivatives and salts thereof