CA1051420A - ESTERS OF .alpha.-SUBSTITUTED AMIDINOPENICILLANIC ACIDS - Google Patents

ESTERS OF .alpha.-SUBSTITUTED AMIDINOPENICILLANIC ACIDS

Info

Publication number
CA1051420A
CA1051420A CA165,831A CA165831A CA1051420A CA 1051420 A CA1051420 A CA 1051420A CA 165831 A CA165831 A CA 165831A CA 1051420 A CA1051420 A CA 1051420A
Authority
CA
Canada
Prior art keywords
formula
compound
process according
penicillanate
ethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA165,831A
Other languages
English (en)
French (fr)
Other versions
CA165831S (en
Inventor
Peter Bamberg
Bertil A. Ekstrom
Berndt O.H. Sjoberg
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Astra Lakemedel AB
Original Assignee
Astra Lakemedel AB
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Lakemedel AB filed Critical Astra Lakemedel AB
Application granted granted Critical
Publication of CA1051420A publication Critical patent/CA1051420A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA165,831A 1972-03-13 1973-03-12 ESTERS OF .alpha.-SUBSTITUTED AMIDINOPENICILLANIC ACIDS Expired CA1051420A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB1168972A GB1427139A (en) 1972-03-13 1972-03-13 Penicillins

Publications (1)

Publication Number Publication Date
CA1051420A true CA1051420A (en) 1979-03-27

Family

ID=9990894

Family Applications (1)

Application Number Title Priority Date Filing Date
CA165,831A Expired CA1051420A (en) 1972-03-13 1973-03-12 ESTERS OF .alpha.-SUBSTITUTED AMIDINOPENICILLANIC ACIDS

Country Status (10)

Country Link
JP (3) JPS5526147B2 (de)
AT (1) AT331391B (de)
CA (1) CA1051420A (de)
CH (2) CH582708A5 (de)
DE (1) DE2311131C3 (de)
DK (1) DK145699C (de)
FR (1) FR2181811B1 (de)
GB (1) GB1427139A (de)
NL (1) NL176943C (de)
SE (2) SE416811B (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1427139A (en) * 1972-03-13 1976-03-10 Astra Laekemedel Ab Penicillins
SU566843A1 (ru) * 1975-01-06 1977-07-30 Ордена Трудового Красного Знамени Институт Органической Синтеза Ан Латвийской Сср Способ получени производных 6- -амидинопенициллановой кислоты
GB1529448A (en) * 1975-10-29 1978-10-18 Leo Pharm Prod Ltd 6-amidinopenicillanic acid derivatives
GB1579931A (en) * 1976-04-15 1980-11-26 Leo Pharm Prod Ltd Bis-penicillanoyl-oxy-alkanes
US4345071A (en) 1976-06-29 1982-08-17 Leo Pharmaceutical Products, Ltd. A/S Derivatives of penicillanic acid
GB1585165A (en) * 1976-06-29 1981-02-25 Leo Pharm Prod Ltd Derivatives of 6-amidino penicillanic acid
LU77362A1 (de) * 1977-05-17 1979-01-19
IL54859A (en) * 1977-06-21 1982-01-31 Rech Applications Therap Derivatives of amidinopenicillanic acid,their production and pharmaceutical compositions containing them
JPS57156495A (en) * 1981-03-23 1982-09-27 Kyoto Yakuhin Kogyo Kk Cephalosporin derivative and remedy for microbism used in oral administration
JPS5865474U (ja) * 1981-10-28 1983-05-04 松下電器産業株式会社 電動弁
IT1190897B (it) * 1982-06-29 1988-02-24 Opos Biochimica Srl Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
JPH0495170U (de) * 1990-12-27 1992-08-18

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1003479A (en) * 1963-05-30 1965-09-02 Wyeth John & Brother Ltd Acetoxymethyl benzylpenicillinate
DE1795423C3 (de) * 1967-09-29 1974-02-28 Loevens Kemiske Fabrik Produktionsaktieselskab, Ballerup (Daenemark) Pivaloyloxymethyl-alpha-aminobenzylpenicillinat
BE758782A (fr) * 1969-11-11 1971-05-10 Leo Pharm Prod Ltd Nouveaux derives d'acide 6-amidino penicillanique leur procede de preparation et leurs applications comme antibiotiques
JPS4828904A (de) * 1971-08-19 1973-04-17
GB1427139A (en) * 1972-03-13 1976-03-10 Astra Laekemedel Ab Penicillins

Also Published As

Publication number Publication date
DE2311131B2 (de) 1979-02-22
SE416811B (sv) 1981-02-09
SE7805910L (sv) 1978-05-24
NL176943B (nl) 1985-02-01
JPS53101394A (en) 1978-09-04
CH582707A5 (de) 1976-12-15
AU5321273A (en) 1974-09-12
CH582708A5 (de) 1976-12-15
JPS5526147B2 (de) 1980-07-11
DK145699B (da) 1983-01-31
DE2311131C3 (de) 1982-06-09
AT331391B (de) 1976-08-25
JPS55105688A (en) 1980-08-13
FR2181811B1 (de) 1976-07-02
DK145699C (da) 1983-07-25
FR2181811A1 (de) 1973-12-07
ATA213973A (de) 1975-11-15
JPS49287A (de) 1974-01-05
GB1427139A (en) 1976-03-10
NL7303434A (de) 1973-09-17
NL176943C (nl) 1985-07-01
DE2311131A1 (de) 1973-10-18

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