CA1050969A - CRYSTALLINE SESQUIHYDRATE OF 7-(D-AMINO-.alpha.-(P-HYDROXYPHENYL) ACETAMIDO)-3-(1,2,3,-TRIAZOL-5-YITHIOMETHYL)-3-CEPHEM-4-CARBOXYLIC ACID - Google Patents
CRYSTALLINE SESQUIHYDRATE OF 7-(D-AMINO-.alpha.-(P-HYDROXYPHENYL) ACETAMIDO)-3-(1,2,3,-TRIAZOL-5-YITHIOMETHYL)-3-CEPHEM-4-CARBOXYLIC ACIDInfo
- Publication number
- CA1050969A CA1050969A CA226,752A CA226752A CA1050969A CA 1050969 A CA1050969 A CA 1050969A CA 226752 A CA226752 A CA 226752A CA 1050969 A CA1050969 A CA 1050969A
- Authority
- CA
- Canada
- Prior art keywords
- cephem
- hydroxyphenyl
- triazol
- amino
- alpha
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/36—Methylene radicals, substituted by sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/473,039 US3985747A (en) | 1974-05-24 | 1974-05-24 | Crystalline sesquihydrate of 7-[D-α-amino-α-(p-hydroxyphenyl)acetamido]-3-(1,2,3-triazol-5-ylthiomethyl)-3-cephem-4-carboxylic acid |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA1050969A true CA1050969A (en) | 1979-03-20 |
Family
ID=23877939
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA226,752A Expired CA1050969A (en) | 1974-05-24 | 1975-05-12 | CRYSTALLINE SESQUIHYDRATE OF 7-(D-AMINO-.alpha.-(P-HYDROXYPHENYL) ACETAMIDO)-3-(1,2,3,-TRIAZOL-5-YITHIOMETHYL)-3-CEPHEM-4-CARBOXYLIC ACID |
Country Status (13)
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2400519A1 (fr) * | 1977-08-17 | 1979-03-16 | Roussel Uclaf | Forme cristalline du sel de sodium d'un derive oximine de l'acide 7-amino-thiazolyl acetamido cephalosporanique, son procede de preparation et son application comme medicament |
| IE49374B1 (en) * | 1979-02-01 | 1985-09-18 | Lilly Co Eli | Crystalline 3-hydroxycephalosporin solvates |
| US4600773A (en) * | 1983-12-01 | 1986-07-15 | Eli Lilly And Company | Crystalline cephalexin hydrochloride monohydrate |
| IT1186778B (it) * | 1985-10-15 | 1987-12-16 | Lark Spa | Cefatrizina glicerolo solvato cristallino e procedimento per la sua preparazione |
| JP3449658B2 (ja) * | 1994-12-21 | 2003-09-22 | 杏林製薬株式会社 | 安定性に優れた８−アルコキシキノロンカルボン酸水和物並びにその製造方法 |
| US7230097B2 (en) * | 2003-03-10 | 2007-06-12 | Lupin Ltd. | Process for preparation of 7-[α-Amino (4-hydroxyphenyl) acetamido]-3-substituted-3-cephem-4-carboxylic acid |
| DE102005009203A1 (de) * | 2005-02-25 | 2006-08-31 | Behr Gmbh & Co. Kg | Vorrichtung zur Beeinflussung eines Luftstroms |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1241844A (en) * | 1968-08-23 | 1971-08-04 | Beecham Group Ltd | Penicillins |
| US3641021A (en) * | 1969-04-18 | 1972-02-08 | Lilly Co Eli | 3 7-(ring-substituted) cephalosporin compounds |
| US3855213A (en) * | 1971-02-18 | 1974-12-17 | Smith Kline French Lab | 3-heterocyclic thiomethyl-cephalosporins |
| US3759904A (en) * | 1971-07-29 | 1973-09-18 | Bristol Myers Co | Ds and salts thereof 3 - (s-(1,2,3-triazole-5-yl)thiomethyl)-3 - cephem - 4-carboxylic aci7-(d-(alpha-amino-alpha-phenyl-, 2-thienyl- and 3-thienylacetamido))- |
-
1974
- 1974-05-24 US US05/473,039 patent/US3985747A/en not_active Expired - Lifetime
-
1975
- 1975-05-12 CA CA226,752A patent/CA1050969A/en not_active Expired
- 1975-05-16 ZA ZA00753174A patent/ZA753174B/xx unknown
- 1975-05-19 AU AU81283/75A patent/AU8128375A/en not_active Expired
- 1975-05-20 GB GB21508/75A patent/GB1487658A/en not_active Expired
- 1975-05-21 NL NL7505961A patent/NL7505961A/xx unknown
- 1975-05-21 DK DK223875A patent/DK223875A/da unknown
- 1975-05-21 SE SE7505807A patent/SE7505807L/xx unknown
- 1975-05-21 BE BE156571A patent/BE829329R/xx active
- 1975-05-22 FR FR7515944A patent/FR2271830A2/fr active Pending
- 1975-05-22 LU LU72558A patent/LU72558A1/xx unknown
- 1975-05-23 JP JP50061156A patent/JPS6011040B2/ja not_active Expired
- 1975-05-23 DE DE19752522998 patent/DE2522998A1/de active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| FR2271830A2 (US08088918-20120103-C00476.png) | 1975-12-19 |
| JPS511627A (US08088918-20120103-C00476.png) | 1976-01-08 |
| GB1487658A (en) | 1977-10-05 |
| ZA753174B (en) | 1976-04-28 |
| DE2522998A1 (de) | 1975-12-11 |
| SE7505807L (sv) | 1975-11-25 |
| JPS6011040B2 (ja) | 1985-03-22 |
| LU72558A1 (US08088918-20120103-C00476.png) | 1976-03-17 |
| DK223875A (da) | 1975-11-25 |
| US3985747A (en) | 1976-10-12 |
| BE829329R (fr) | 1975-11-21 |
| NL7505961A (nl) | 1975-11-26 |
| AU8128375A (en) | 1976-11-25 |
| USB473039I5 (US08088918-20120103-C00476.png) | 1976-02-10 |
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