CA1010444A - Process for preparing 6-(a-(guanylureidoalkanylamino) aracylamino) penicillanic acids - Google Patents
Process for preparing 6-(a-(guanylureidoalkanylamino) aracylamino) penicillanic acidsInfo
- Publication number
- CA1010444A CA1010444A CA167,956A CA167956A CA1010444A CA 1010444 A CA1010444 A CA 1010444A CA 167956 A CA167956 A CA 167956A CA 1010444 A CA1010444 A CA 1010444A
- Authority
- CA
- Canada
- Prior art keywords
- guanylureidoalkanylamino
- aracylamino
- preparing
- penicillanic acids
- penicillanic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/04—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms
- C07C275/06—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an acyclic and saturated carbon skeleton
- C07C275/16—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an acyclic and saturated carbon skeleton being further substituted by carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
- C07C279/28—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to cyano groups, e.g. cyanoguanidines, dicyandiamides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C335/30—Isothioureas
- C07C335/34—Isothioureas having sulfur atoms of isothiourea groups bound to carbon atoms of rings other than six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C335/30—Isothioureas
- C07C335/38—Isothioureas containing any of the groups, X being a hetero atom, Y being any atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/30—Oxygen or sulfur atoms
- C07D233/42—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
- C07D233/46—Nitrogen atoms not forming part of a nitro radical with only hydrogen atoms attached to said nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Cephalosporin Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US00253856A US3838153A (en) | 1972-05-16 | 1972-05-16 | 6-(alpha-(guanylureidoalkanoylamino)aracylamino)penicillanic acids |
Publications (1)
Publication Number | Publication Date |
---|---|
CA1010444A true CA1010444A (en) | 1977-05-17 |
Family
ID=22961983
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA167,956A Expired CA1010444A (en) | 1972-05-16 | 1973-04-04 | Process for preparing 6-(a-(guanylureidoalkanylamino) aracylamino) penicillanic acids |
Country Status (23)
Country | Link |
---|---|
US (1) | US3838153A (fi) |
JP (1) | JPS5533712B2 (fi) |
AR (1) | AR195914A1 (fi) |
AT (1) | AT325767B (fi) |
AU (1) | AU475922B2 (fi) |
BE (1) | BE798170A (fi) |
CA (1) | CA1010444A (fi) |
CH (1) | CH573434A5 (fi) |
DE (1) | DE2318986A1 (fi) |
DK (1) | DK137046B (fi) |
ES (1) | ES413937A1 (fi) |
FI (1) | FI56534C (fi) |
FR (1) | FR2184609B1 (fi) |
GB (1) | GB1404469A (fi) |
IE (1) | IE37491B1 (fi) |
IL (1) | IL41937A (fi) |
NL (1) | NL7305355A (fi) |
PH (1) | PH10024A (fi) |
PL (1) | PL89245B1 (fi) |
SE (1) | SE415976B (fi) |
SU (1) | SU504491A3 (fi) |
YU (1) | YU36965B (fi) |
ZA (1) | ZA732343B (fi) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1462421A (en) * | 1973-12-14 | 1977-01-26 | Pfizer | 6-a-amidino-and -'midoylaminoalkanoylamino aracylamino-penicillanic acids and their preparation |
US3994965A (en) * | 1974-08-09 | 1976-11-30 | Pfizer Inc. | D-N-(guanylureidoacetyl)-α-aminophenyl acetic acid and D-N-(guanylureidoacetyl)-α-aminophenyl acetyl chloride |
JPS5562537U (fi) * | 1978-10-20 | 1980-04-28 | ||
DE3014353A1 (de) * | 1980-04-15 | 1982-01-21 | Bayer Ag, 5090 Leverkusen | Trisubstituierte cyanguanidine, verfahren zu ihrer herstellung sowie ihre verwendung als fungizide |
JPS56161152A (en) * | 1980-05-12 | 1981-12-11 | Tachikawa Spring Co | Manufacture of steel band with resin |
US7973156B2 (en) * | 1997-08-21 | 2011-07-05 | Quark Pharmaceuticals Inc. | Hypoxia-regulated genes |
IL134298A0 (en) | 1997-08-21 | 2001-04-30 | Quark Biotech Inc | Hypoxia-regulating genes |
US20030104973A1 (en) * | 1997-08-21 | 2003-06-05 | Quark Biotech, Inc. | Hypoxia-regulated genes |
-
1972
- 1972-05-16 US US00253856A patent/US3838153A/en not_active Expired - Lifetime
- 1972-09-11 GB GB4217972A patent/GB1404469A/en not_active Expired
-
1973
- 1973-03-30 SE SE7304567A patent/SE415976B/xx unknown
- 1973-04-03 IE IE521/73A patent/IE37491B1/xx unknown
- 1973-04-03 IL IL41937A patent/IL41937A/en unknown
- 1973-04-04 CA CA167,956A patent/CA1010444A/en not_active Expired
- 1973-04-04 ZA ZA732343A patent/ZA732343B/xx unknown
- 1973-04-09 AU AU54283/73A patent/AU475922B2/en not_active Expired
- 1973-04-11 YU YU0977/73A patent/YU36965B/xx unknown
- 1973-04-13 FR FR7313445A patent/FR2184609B1/fr not_active Expired
- 1973-04-13 FI FI1178/73A patent/FI56534C/fi active
- 1973-04-13 BE BE1004965A patent/BE798170A/xx unknown
- 1973-04-14 DE DE2318986A patent/DE2318986A1/de active Pending
- 1973-04-17 AT AT341573A patent/AT325767B/de not_active IP Right Cessation
- 1973-04-17 NL NL7305355A patent/NL7305355A/xx not_active Application Discontinuation
- 1973-04-18 AR AR247615A patent/AR195914A1/es active
- 1973-04-18 DK DK216373AA patent/DK137046B/da unknown
- 1973-04-19 ES ES413937A patent/ES413937A1/es not_active Expired
- 1973-04-19 SU SU1912246A patent/SU504491A3/ru active
- 1973-04-19 CH CH569673A patent/CH573434A5/xx not_active IP Right Cessation
- 1973-04-20 JP JP4424473A patent/JPS5533712B2/ja not_active Expired
- 1973-05-15 PL PL1973162558A patent/PL89245B1/pl unknown
-
1975
- 1975-04-11 PH PH14505*[A patent/PH10024A/en unknown
Also Published As
Publication number | Publication date |
---|---|
YU97773A (en) | 1982-06-18 |
AR195914A1 (es) | 1973-11-15 |
PH10024A (en) | 1976-07-13 |
IE37491L (en) | 1973-11-16 |
YU36965B (en) | 1984-08-31 |
FI56534C (fi) | 1980-02-11 |
SE415976B (sv) | 1980-11-17 |
DK137046C (fi) | 1978-06-12 |
BE798170A (fr) | 1973-10-15 |
PL89245B1 (fi) | 1976-11-30 |
IL41937A (en) | 1976-10-31 |
CH573434A5 (fi) | 1976-03-15 |
AU5428373A (en) | 1974-10-10 |
ES413937A1 (es) | 1976-06-01 |
FR2184609A1 (fi) | 1973-12-28 |
IL41937A0 (en) | 1973-06-29 |
NL7305355A (fi) | 1973-11-20 |
US3838153A (en) | 1974-09-24 |
GB1404469A (en) | 1975-08-28 |
SU504491A3 (ru) | 1976-02-25 |
ATA341573A (de) | 1975-01-15 |
IE37491B1 (en) | 1977-08-03 |
JPS4924991A (fi) | 1974-03-05 |
FR2184609B1 (fi) | 1976-10-22 |
AU475922B2 (en) | 1976-09-09 |
DK137046B (da) | 1978-01-09 |
FI56534B (fi) | 1979-10-31 |
ZA732343B (en) | 1974-01-30 |
AT325767B (de) | 1975-11-10 |
DE2318986A1 (de) | 1973-12-06 |
JPS5533712B2 (fi) | 1980-09-02 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
JPS53101394A (en) | Process for freparing novel penicillanic derivative | |
CA1010444A (en) | Process for preparing 6-(a-(guanylureidoalkanylamino) aracylamino) penicillanic acids | |
YU298573A (en) | Process for obtaining 6-aminopenicillanic acid | |
CA978999A (en) | Process for the production of ortho-dihydrocarbylphosphinobenzoic acids | |
CA1012974A (en) | Process for preparing sulfamylbenzoic acids | |
CA1023348A (en) | PROCESS FOR PREPARING 6-(.alpha.-AMIDINO-AND IMIDOYLAMINOALKANOYLAMINO) ARACYLAMINO) PENICILLANIC ACIDS | |
YU36966B (en) | Process for obtaining 6-(amidino-and imidoylaminoalkanoylamino0aracylamino penicillanic acids | |
CA1007635A (en) | Process for preparing penicillin sulfoxide | |
CA903224A (en) | Process for the production of pyridones | |
CA1034115A (en) | Process for producing desacetoxycephalosporin derivatives | |
CA967976A (en) | Process for producing trimethyl-p-benzoquinone | |
CA987326A (en) | Process for producing 2-acyl-5-nitrothiazoles | |
CA994805A (en) | Process for the production of formaldehyde | |
CA913621A (en) | Process for producing 6-aminopenicillanic acid | |
AU462293B2 (en) | 6-amino penicillanic acid derivatives | |
CA893694A (en) | Process for preparing 6-aminopenicillanic acid compounds | |
CA905412A (en) | Process for preparing 6-aminopenicillanic acid compounds | |
CA894235A (en) | Process for producing 1-acylindole derivatives | |
CA900476A (en) | Process for producing 1-aminoalkylbenzodiazepine derivatives | |
CA891499A (en) | Process for preparing 3-indolylacetic acids | |
CA892005A (en) | Process for producing orotidylic acid | |
AU425419B2 (en) | Process for producing 6 aminoacylamido penicillanic acids | |
AU462377B2 (en) | 6-amino penicillanic acid derivatives | |
CA892024A (en) | Method for producing penicillins | |
CA903947A (en) | Process for producing polyamides |