BRPI0923279A2 - formas cristalinas do composto 2-[4-(7-etil-5h-pirrol[2,3-b]pirazin-6-il)-fenil]-propan-2-ol, seu uso e processo de obtenção - Google Patents
formas cristalinas do composto 2-[4-(7-etil-5h-pirrol[2,3-b]pirazin-6-il)-fenil]-propan-2-ol, seu uso e processo de obtençãoInfo
- Publication number
- BRPI0923279A2 BRPI0923279A2 BRPI0923279A BRPI0923279A BRPI0923279A2 BR PI0923279 A2 BRPI0923279 A2 BR PI0923279A2 BR PI0923279 A BRPI0923279 A BR PI0923279A BR PI0923279 A BRPI0923279 A BR PI0923279A BR PI0923279 A2 BRPI0923279 A2 BR PI0923279A2
- Authority
- BR
- Brazil
- Prior art keywords
- pyrazin
- pyrrol
- propan
- phenyl
- ethyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Cardiology (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Immunology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US11986608P | 2008-12-04 | 2008-12-04 | |
PCT/US2009/066489 WO2010065690A1 (en) | 2008-12-04 | 2009-12-03 | Crystalline forms |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0923279A2 true BRPI0923279A2 (pt) | 2016-01-26 |
Family
ID=42109934
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0923279A BRPI0923279A2 (pt) | 2008-12-04 | 2009-12-03 | formas cristalinas do composto 2-[4-(7-etil-5h-pirrol[2,3-b]pirazin-6-il)-fenil]-propan-2-ol, seu uso e processo de obtenção |
Country Status (15)
Country | Link |
---|---|
US (1) | US20110257190A1 (pt) |
EP (1) | EP2373655A1 (pt) |
JP (1) | JP2012511005A (pt) |
KR (1) | KR20110108334A (pt) |
CN (1) | CN102239169A (pt) |
AR (1) | AR074538A1 (pt) |
AU (1) | AU2009322409A1 (pt) |
BR (1) | BRPI0923279A2 (pt) |
CA (1) | CA2745262A1 (pt) |
IL (1) | IL213288A0 (pt) |
MX (1) | MX2011004793A (pt) |
RU (1) | RU2011127147A (pt) |
TW (1) | TW201033211A (pt) |
UY (1) | UY32293A (pt) |
WO (1) | WO2010065690A1 (pt) |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PT1221918E (pt) | 1999-10-21 | 2005-06-30 | Alcon Inc | Administracao de drogas sub-tenon |
US20050059639A1 (en) | 2003-09-11 | 2005-03-17 | Wei Edward T. | Ophthalmic compositions and method for treating eye discomfort and pain |
CL2007002617A1 (es) | 2006-09-11 | 2008-05-16 | Sanofi Aventis | Compuestos derivados de pirrolo[2,3-b]pirazin-6-ilo; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar inflamacion de las articulaciones, artritis reumatoide, tumores, linfoma de las celulas del manto. |
-
2009
- 2009-12-03 WO PCT/US2009/066489 patent/WO2010065690A1/en active Application Filing
- 2009-12-03 RU RU2011127147/04A patent/RU2011127147A/ru not_active Application Discontinuation
- 2009-12-03 EP EP09775419A patent/EP2373655A1/en not_active Withdrawn
- 2009-12-03 KR KR1020117014527A patent/KR20110108334A/ko not_active Application Discontinuation
- 2009-12-03 TW TW098141270A patent/TW201033211A/zh unknown
- 2009-12-03 MX MX2011004793A patent/MX2011004793A/es not_active Application Discontinuation
- 2009-12-03 AU AU2009322409A patent/AU2009322409A1/en not_active Abandoned
- 2009-12-03 BR BRPI0923279A patent/BRPI0923279A2/pt not_active Application Discontinuation
- 2009-12-03 CN CN2009801482672A patent/CN102239169A/zh active Pending
- 2009-12-03 CA CA2745262A patent/CA2745262A1/en not_active Abandoned
- 2009-12-03 JP JP2011539673A patent/JP2012511005A/ja not_active Withdrawn
- 2009-12-04 UY UY0001032293A patent/UY32293A/es not_active Application Discontinuation
- 2009-12-04 AR ARP090104692A patent/AR074538A1/es unknown
-
2011
- 2011-05-31 IL IL213288A patent/IL213288A0/en unknown
- 2011-06-02 US US13/151,853 patent/US20110257190A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
JP2012511005A (ja) | 2012-05-17 |
IL213288A0 (en) | 2011-07-31 |
AU2009322409A1 (en) | 2011-06-23 |
US20110257190A1 (en) | 2011-10-20 |
EP2373655A1 (en) | 2011-10-12 |
AR074538A1 (es) | 2011-01-26 |
RU2011127147A (ru) | 2013-01-10 |
KR20110108334A (ko) | 2011-10-05 |
CN102239169A (zh) | 2011-11-09 |
WO2010065690A1 (en) | 2010-06-10 |
CA2745262A1 (en) | 2010-06-10 |
TW201033211A (en) | 2010-09-16 |
MX2011004793A (es) | 2011-05-30 |
UY32293A (es) | 2010-07-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |