BRPI0810330A2 - "PROCESS FOR PREPARING (R) -2-METHYL-PYROROLIDINE L-TARTARATE, PROCESS FOR PREPARING 6- {4- [3 - ((R) -2-METHYL-PYROLIDIN-1-IL) -PROPOXY] -Phenyl} - 2H-PYRIDAZIN-3-ONA, PROCESS FOR PREPARING (S) -2-METHYL PYROLIDINE D-TARTARATE " - Google Patents

"PROCESS FOR PREPARING (R) -2-METHYL-PYROROLIDINE L-TARTARATE, PROCESS FOR PREPARING 6- {4- [3 - ((R) -2-METHYL-PYROLIDIN-1-IL) -PROPOXY] -Phenyl} - 2H-PYRIDAZIN-3-ONA, PROCESS FOR PREPARING (S) -2-METHYL PYROLIDINE D-TARTARATE "

Info

Publication number
BRPI0810330A2
BRPI0810330A2 BRPI0810330-5A2A BRPI0810330A BRPI0810330A2 BR PI0810330 A2 BRPI0810330 A2 BR PI0810330A2 BR PI0810330 A BRPI0810330 A BR PI0810330A BR PI0810330 A2 BRPI0810330 A2 BR PI0810330A2
Authority
BR
Brazil
Prior art keywords
preparing
methyl
tartarate
pyrorolidine
pyrolidin
Prior art date
Application number
BRPI0810330-5A2A
Other languages
Portuguese (pt)
Inventor
Michael Christie
Joseph J Petraitis
Original Assignee
Cephalon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cephalon Inc filed Critical Cephalon Inc
Publication of BRPI0810330A2 publication Critical patent/BRPI0810330A2/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/06—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with radicals, containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cosmetics (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
  • Pyrrole Compounds (AREA)
BRPI0810330-5A2A 2007-05-03 2008-05-02 "PROCESS FOR PREPARING (R) -2-METHYL-PYROROLIDINE L-TARTARATE, PROCESS FOR PREPARING 6- {4- [3 - ((R) -2-METHYL-PYROLIDIN-1-IL) -PROPOXY] -Phenyl} - 2H-PYRIDAZIN-3-ONA, PROCESS FOR PREPARING (S) -2-METHYL PYROLIDINE D-TARTARATE " BRPI0810330A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US92735607P 2007-05-03 2007-05-03
PCT/US2008/005702 WO2008137087A1 (en) 2007-05-03 2008-05-02 Processes for preparing (r)-2-methylpyrrolidine and (s)-2-methylpyrrolidine and tartrate salts thereof

Publications (1)

Publication Number Publication Date
BRPI0810330A2 true BRPI0810330A2 (en) 2014-10-14

Family

ID=39688886

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0810330-5A2A BRPI0810330A2 (en) 2007-05-03 2008-05-02 "PROCESS FOR PREPARING (R) -2-METHYL-PYROROLIDINE L-TARTARATE, PROCESS FOR PREPARING 6- {4- [3 - ((R) -2-METHYL-PYROLIDIN-1-IL) -PROPOXY] -Phenyl} - 2H-PYRIDAZIN-3-ONA, PROCESS FOR PREPARING (S) -2-METHYL PYROLIDINE D-TARTARATE "

Country Status (14)

Country Link
EP (1) EP2152669A1 (en)
JP (1) JP5698887B2 (en)
KR (1) KR20100017565A (en)
CN (1) CN101679237A (en)
AU (1) AU2008248168B2 (en)
BR (1) BRPI0810330A2 (en)
CA (1) CA2686033A1 (en)
EA (1) EA019031B1 (en)
IL (1) IL201627A (en)
MX (1) MX2009011787A (en)
NZ (1) NZ580948A (en)
UA (1) UA99913C2 (en)
WO (1) WO2008137087A1 (en)
ZA (1) ZA200907643B (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2397283T3 (en) 2006-07-25 2013-03-06 Cephalon, Inc. Pyridizinone derivatives
US8383657B2 (en) 2007-12-21 2013-02-26 Abbott Laboratories Thiazolylidine urea and amide derivatives and methods of use thereof
EP2752406A1 (en) * 2008-01-30 2014-07-09 Cephalon, Inc. Substituted pyridazine derivatives which have histamine H3 antagonist activity
EP3237408B1 (en) * 2014-12-23 2018-10-31 Cephalon, Inc. Methods for preparing fused bicyclic 2, 4-diaminopyrimidine derivatives

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3329974A1 (en) 1983-08-19 1985-02-28 Bayer Ag, 5090 Leverkusen MANUFACTURE OF HYDRATED NITRILE RUBBER
DE3433392A1 (en) 1984-09-12 1986-03-20 Bayer Ag, 5090 Leverkusen HYDROGENATION OF UNSATURATED POLYMER WITH NITRILE GROUPS
FR2714849B1 (en) 1994-01-13 1996-04-05 Inst Francais Du Petrole Process for the preparation of a hydrogenation catalyst soluble in the organic liquid phase.
DE4403479A1 (en) 1994-02-04 1995-08-10 Basf Ag Process for the preparation of hydroxylammonium salts
WO2004024707A2 (en) * 2002-09-16 2004-03-25 Abbott Laboratories Process for preparing amine type substituted benzofurans
US7153889B2 (en) 2002-11-12 2006-12-26 Abbott Laboratories Bicyclic-substituted amines as histamine-3 receptor ligands
CN100543050C (en) 2004-03-08 2009-09-23 独立行政法人科学技术振兴机构 Polymer-supported metal cluster compositions
US7145005B2 (en) 2004-05-12 2006-12-05 Abbott Laboratories 2-(6-{2-[(2R)-2-Methyl-1-pyrrolidin-1-yl]-ethyl}-2-naphthalen-2-yl)-2H-pyridazin-3-one salts and their preparation
ES2299074T3 (en) 2004-06-02 2008-05-16 F. Hoffmann-La Roche Ag USEFUL NAFTALEN DERIVATIVES AS LEGANDS OF THE RECEIVER 3 OF HISTAMINE.
WO2006059778A1 (en) 2004-12-01 2006-06-08 Banyu Pharmaceutical Co., Ltd. Substituted pyridone derivative
JP2008524252A (en) 2004-12-17 2008-07-10 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Tetrahydroisoquinoline compounds for the treatment of CNS disorders
JP2008526895A (en) 2005-01-21 2008-07-24 シェーリング コーポレイション Imidazole and benzimidazole derivatives useful as histamine H3 antagonists
CA2602336A1 (en) 2005-03-31 2006-10-05 Ucb Pharma S.A. Compounds comprising an oxazole or thiazole moiety, processes for making them, and their uses
GB0514812D0 (en) 2005-07-19 2005-08-24 Glaxo Group Ltd Compounds
CA2627234A1 (en) 2005-10-27 2007-05-03 Ucb Pharma, S.A. Compounds comprising a lactam or a lactam derivative moiety, processes for making them, and their uses
WO2007094962A2 (en) 2006-02-09 2007-08-23 Athersys, Inc. Pyrazoles for the treatment of obesity and other cns disorders
WO2007099423A1 (en) 2006-03-02 2007-09-07 Pfizer Products Inc. 1-pyrrolidine indane derivatives as histamine-3 receptor antagonists
US20090163482A1 (en) 2006-03-13 2009-06-25 Mchardy Stanton Furst Tetralines antagonists of the h-3 receptor
WO2008005338A1 (en) 2006-06-29 2008-01-10 Arena Pharmaceuticals, Inc. Modulators of the histamine h3-receptor useful for the treatment of disorders related thereto
ES2397283T3 (en) * 2006-07-25 2013-03-06 Cephalon, Inc. Pyridizinone derivatives

Also Published As

Publication number Publication date
WO2008137087A1 (en) 2008-11-13
JP5698887B2 (en) 2015-04-08
IL201627A0 (en) 2010-05-31
CN101679237A (en) 2010-03-24
JP2010526142A (en) 2010-07-29
AU2008248168A1 (en) 2008-11-13
AU2008248168B2 (en) 2013-03-21
NZ580948A (en) 2011-04-29
EA019031B1 (en) 2013-12-30
ZA200907643B (en) 2014-03-26
EA200971019A1 (en) 2010-04-30
CA2686033A1 (en) 2008-11-13
UA99913C2 (en) 2012-10-25
IL201627A (en) 2014-06-30
KR20100017565A (en) 2010-02-16
EP2152669A1 (en) 2010-02-17
MX2009011787A (en) 2009-11-13

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 8A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2384 DE 13-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

B350 Update of information on the portal [chapter 15.35 patent gazette]