BRPI0614810A2 - combinação de compostos orgánicos - Google Patents
combinação de compostos orgánicosInfo
- Publication number
- BRPI0614810A2 BRPI0614810A2 BRPI0614810-7A BRPI0614810A BRPI0614810A2 BR PI0614810 A2 BRPI0614810 A2 BR PI0614810A2 BR PI0614810 A BRPI0614810 A BR PI0614810A BR PI0614810 A2 BRPI0614810 A2 BR PI0614810A2
- Authority
- BR
- Brazil
- Prior art keywords
- combination
- organic compounds
- compound
- treating
- preventing
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
COMBINAçãO DE COMPOSTOS ORGáNICOS. A invenção proporciona uma combinação farmacêutica que compreende: a) um composto de pirimidilaminobenzamida; e b) um composto de inibidor de HDAC, e um método para tratar ou prevenir uma doença proliferativa usando tal combinação.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US70743605P | 2005-08-11 | 2005-08-11 | |
PCT/US2006/031563 WO2007022044A2 (en) | 2005-08-11 | 2006-08-10 | Combination of organic compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0614810A2 true BRPI0614810A2 (pt) | 2009-08-04 |
Family
ID=37735081
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0614810-7A BRPI0614810A2 (pt) | 2005-08-11 | 2006-08-10 | combinação de compostos orgánicos |
Country Status (11)
Country | Link |
---|---|
US (1) | US20080200489A1 (pt) |
EP (1) | EP1915154A2 (pt) |
JP (1) | JP2009504674A (pt) |
KR (1) | KR20080044277A (pt) |
CN (1) | CN101282728A (pt) |
AU (2) | AU2006279781A1 (pt) |
BR (1) | BRPI0614810A2 (pt) |
CA (1) | CA2617979A1 (pt) |
MX (1) | MX2008001971A (pt) |
RU (1) | RU2008108911A (pt) |
WO (1) | WO2007022044A2 (pt) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2060565A1 (en) * | 2007-11-16 | 2009-05-20 | 4Sc Ag | Novel bifunctional compounds which inhibit protein kinases and histone deacetylases |
CA2753637A1 (en) * | 2009-03-06 | 2010-09-10 | Novartis Ag | Use of pyrimidylaminobenzamide derivatives for the treatment of disorders mediated by the leucine zipper- and sterile alpha motif-containing kinase (zak) |
AU2012319188B2 (en) * | 2011-10-03 | 2016-11-24 | Sloan-Kettering Institute For Cancer Research | Novel molecules that selectively inhibit histone deacetylase 6 relative to histone deacetylase 1 |
WO2015100363A1 (en) | 2013-12-23 | 2015-07-02 | The Trustees Of Columbia University In The City Of New York | Selective hdac6 inhibitors |
JP6531312B2 (ja) * | 2014-10-17 | 2019-06-19 | 東洋鋼鈑株式会社 | Bcr−abl阻害剤耐性関連変異の検出方法及びこれを用いたbcr−abl阻害剤耐性を予測するためのデータ取得方法 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PE20020354A1 (es) * | 2000-09-01 | 2002-06-12 | Novartis Ag | Compuestos de hidroxamato como inhibidores de histona-desacetilasa (hda) |
GB0215676D0 (en) * | 2002-07-05 | 2002-08-14 | Novartis Ag | Organic compounds |
JP2006501267A (ja) * | 2002-09-13 | 2006-01-12 | バージニア コモンウェルス ユニバーシティー | 白血病の処置のためのa)N−{5−[4−(4−メチル−ピペラジノ−メチル)−ベンゾイルアミド]−2−メチルフェニル}−4−(3−ピリジル)−2−ピリミジン−アミンおよびb)ヒストンデアセチラーゼインヒビターの組合せ剤 |
US20040127571A1 (en) * | 2002-09-19 | 2004-07-01 | University Of South Florida | Method of Treating Leukemia with a Combination of Suberoylanilide Hydromaxic Acid and Imatinib Mesylate |
-
2006
- 2006-08-10 CA CA002617979A patent/CA2617979A1/en not_active Abandoned
- 2006-08-10 MX MX2008001971A patent/MX2008001971A/es active IP Right Grant
- 2006-08-10 US US12/063,172 patent/US20080200489A1/en not_active Abandoned
- 2006-08-10 EP EP06801378A patent/EP1915154A2/en not_active Withdrawn
- 2006-08-10 RU RU2008108911/15A patent/RU2008108911A/ru not_active Application Discontinuation
- 2006-08-10 JP JP2008526270A patent/JP2009504674A/ja not_active Withdrawn
- 2006-08-10 BR BRPI0614810-7A patent/BRPI0614810A2/pt not_active IP Right Cessation
- 2006-08-10 AU AU2006279781A patent/AU2006279781A1/en not_active Abandoned
- 2006-08-10 WO PCT/US2006/031563 patent/WO2007022044A2/en active Application Filing
- 2006-08-10 KR KR1020087005782A patent/KR20080044277A/ko not_active Application Discontinuation
- 2006-08-10 CN CNA2006800375839A patent/CN101282728A/zh active Pending
-
2010
- 2010-10-20 AU AU2010235917A patent/AU2010235917A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
EP1915154A2 (en) | 2008-04-30 |
AU2006279781A1 (en) | 2007-02-22 |
JP2009504674A (ja) | 2009-02-05 |
CA2617979A1 (en) | 2007-02-22 |
WO2007022044A3 (en) | 2007-05-24 |
RU2008108911A (ru) | 2009-09-20 |
CN101282728A (zh) | 2008-10-08 |
MX2008001971A (es) | 2008-03-26 |
WO2007022044A2 (en) | 2007-02-22 |
US20080200489A1 (en) | 2008-08-21 |
AU2010235917A1 (en) | 2010-11-11 |
KR20080044277A (ko) | 2008-05-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A ANUI DADE. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2214 DE 11/06/2013. |