BRPI0412898A - unsubstituted indolyl-3-glyoxylic acid amides, their use as a medicament, and process for their production - Google Patents
unsubstituted indolyl-3-glyoxylic acid amides, their use as a medicament, and process for their productionInfo
- Publication number
- BRPI0412898A BRPI0412898A BRPI0412898-2A BRPI0412898A BRPI0412898A BR PI0412898 A BRPI0412898 A BR PI0412898A BR PI0412898 A BRPI0412898 A BR PI0412898A BR PI0412898 A BRPI0412898 A BR PI0412898A
- Authority
- BR
- Brazil
- Prior art keywords
- production
- medicament
- acid amides
- glyoxylic acid
- unsubstituted indolyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
"AMIDAS DE áCIDO INDOLIL-3-GLIOXìLICO N-SUBSTITUìDAS, SEU USO COMO UM MEDICAMENTO, E PROCESSO PARA SUA PRODUçãO". A invenção refere-se a novas amidas de ácido indolil-3-glioxílico N-substituídas de fórmula geral (I), sua produção, e seu uso como um medicamento, especialmente para o tratamento de tumores."N-REPLACED INDOLYL-3-GLIOXYLIC ACID AMIDS, ITS USE AS A MEDICINAL PRODUCT, AND PROCESS FOR THEIR PRODUCTION". The invention relates to novel N-substituted indolyl-3-glyoxylic acid amides of formula (I), their production, and their use as a medicament, especially for the treatment of tumors.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10334040A DE10334040A1 (en) | 2003-07-25 | 2003-07-25 | Novel N-substituted indolyl-3-glyoxylic acid amides, their use as medicaments and process for their preparation |
PCT/EP2004/007573 WO2005014542A2 (en) | 2003-07-25 | 2004-07-09 | Novel n-substituted indolyl-3-glyoxylic acid amides, use thereof as a medicament against cancer, and method for the production thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0412898A true BRPI0412898A (en) | 2006-10-03 |
Family
ID=34129467
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0412898-2A BRPI0412898A (en) | 2003-07-25 | 2004-07-09 | unsubstituted indolyl-3-glyoxylic acid amides, their use as a medicament, and process for their production |
Country Status (18)
Country | Link |
---|---|
EP (1) | EP1651600A2 (en) |
JP (1) | JP2007503376A (en) |
KR (1) | KR20060037398A (en) |
CN (1) | CN1839129A (en) |
AR (1) | AR045928A1 (en) |
AU (1) | AU2004263238A1 (en) |
BR (1) | BRPI0412898A (en) |
CA (1) | CA2533433A1 (en) |
DE (1) | DE10334040A1 (en) |
IL (1) | IL173335A0 (en) |
MX (1) | MXPA06000995A (en) |
NO (1) | NO20060697L (en) |
RS (1) | RS20060049A (en) |
RU (1) | RU2317293C9 (en) |
TW (1) | TW200524863A (en) |
UA (1) | UA83498C2 (en) |
WO (1) | WO2005014542A2 (en) |
ZA (1) | ZA200601300B (en) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP5406716B2 (en) | 2006-08-07 | 2014-02-05 | アイアンウッド ファーマシューティカルズ インコーポレイテッド | Indole compounds |
AR084433A1 (en) | 2010-12-22 | 2013-05-15 | Ironwood Pharmaceuticals Inc | FAAH INHIBITORS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2005504790A (en) * | 2001-09-13 | 2005-02-17 | シンタ ファーマスーティカルズ コーポレイション | 3-glyoxylylamidoindole for treating cancer |
-
2003
- 2003-07-25 DE DE10334040A patent/DE10334040A1/en not_active Withdrawn
-
2004
- 2004-07-09 RS YUP-2006/0049A patent/RS20060049A/en unknown
- 2004-07-09 BR BRPI0412898-2A patent/BRPI0412898A/en not_active IP Right Cessation
- 2004-07-09 KR KR1020067001636A patent/KR20060037398A/en not_active Application Discontinuation
- 2004-07-09 WO PCT/EP2004/007573 patent/WO2005014542A2/en active Application Filing
- 2004-07-09 EP EP04740854A patent/EP1651600A2/en not_active Withdrawn
- 2004-07-09 RU RU2006105708/04A patent/RU2317293C9/en not_active IP Right Cessation
- 2004-07-09 CA CA002533433A patent/CA2533433A1/en not_active Abandoned
- 2004-07-09 CN CNA2004800240832A patent/CN1839129A/en active Pending
- 2004-07-09 JP JP2006521430A patent/JP2007503376A/en not_active Withdrawn
- 2004-07-09 AU AU2004263238A patent/AU2004263238A1/en not_active Abandoned
- 2004-07-09 MX MXPA06000995A patent/MXPA06000995A/en unknown
- 2004-07-19 TW TW093121509A patent/TW200524863A/en unknown
- 2004-07-23 AR ARP040102632A patent/AR045928A1/en not_active Application Discontinuation
- 2004-09-07 UA UAA200601216A patent/UA83498C2/en unknown
-
2006
- 2006-01-24 IL IL173335A patent/IL173335A0/en unknown
- 2006-02-13 ZA ZA200601300A patent/ZA200601300B/en unknown
- 2006-02-14 NO NO20060697A patent/NO20060697L/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO2005014542A2 (en) | 2005-02-17 |
TW200524863A (en) | 2005-08-01 |
RU2317293C2 (en) | 2008-02-20 |
RS20060049A (en) | 2008-08-07 |
DE10334040A1 (en) | 2005-03-10 |
ZA200601300B (en) | 2007-03-28 |
EP1651600A2 (en) | 2006-05-03 |
AU2004263238A1 (en) | 2005-02-17 |
RU2006105708A (en) | 2006-06-27 |
NO20060697L (en) | 2006-02-14 |
KR20060037398A (en) | 2006-05-03 |
RU2317293C9 (en) | 2008-05-10 |
CN1839129A (en) | 2006-09-27 |
WO2005014542A3 (en) | 2006-10-19 |
IL173335A0 (en) | 2006-06-11 |
CA2533433A1 (en) | 2005-02-17 |
AR045928A1 (en) | 2005-11-16 |
MXPA06000995A (en) | 2006-04-11 |
JP2007503376A (en) | 2007-02-22 |
UA83498C2 (en) | 2008-07-25 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B15K | Others concerning applications: alteration of classification |
Free format text: PARA: INT. CL. C07D 209/00; A61P 35/00 Ipc: C07D 209/00 (2011.01), A61P 35/00 (2011.01) |
|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 7A E 8A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2159 DE 22/05/2012. |