BR9913052A - Rapamicinas fotocilizadas - Google Patents
Rapamicinas fotocilizadasInfo
- Publication number
- BR9913052A BR9913052A BR9913052-1A BR9913052A BR9913052A BR 9913052 A BR9913052 A BR 9913052A BR 9913052 A BR9913052 A BR 9913052A BR 9913052 A BR9913052 A BR 9913052A
- Authority
- BR
- Brazil
- Prior art keywords
- photocilized
- rapamycin
- antiproliferative
- antiinflammatory
- immunosuppressive
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Engineering & Computer Science (AREA)
- Oncology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Communicable Diseases (AREA)
- Hematology (AREA)
- Transplantation (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Patente de Invenção:<B>"RAPAMICINAS FOTOCICLIZADAS"<D>. A presente invenção refere-se a um composto de estrutura (I) ou (II) ou um éter na posição 31- ou 42- dos mesmos, que é de utilidade como um agente imunossupressor, antiinflamatório, antifungicida e antitumor.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US13542198A | 1998-08-17 | 1998-08-17 | |
PCT/US1999/018564 WO2000009510A1 (en) | 1998-08-17 | 1999-08-16 | Photocyclized rapamycins |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9913052A true BR9913052A (pt) | 2001-05-08 |
Family
ID=22468034
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9913052-1A BR9913052A (pt) | 1998-08-17 | 1999-08-16 | Rapamicinas fotocilizadas |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP1105395B1 (pt) |
JP (1) | JP2002522543A (pt) |
CN (1) | CN1323310A (pt) |
AT (1) | ATE219492T1 (pt) |
AU (1) | AU5487499A (pt) |
BR (1) | BR9913052A (pt) |
CA (1) | CA2340700A1 (pt) |
DE (1) | DE69901907T2 (pt) |
DK (1) | DK1105395T3 (pt) |
ES (1) | ES2179671T3 (pt) |
PT (1) | PT1105395E (pt) |
WO (1) | WO2000009510A1 (pt) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2571710A1 (en) | 2004-06-24 | 2006-11-02 | Nicholas Valiante | Small molecule immunopotentiators and assays for their detection |
ES2380779T3 (es) | 2004-12-20 | 2012-05-18 | Wyeth Llc | Análogos de rapamicina y usos de los mismos en el tratamiento de trastornos neurológicos, proliferativos e inflamatorios |
CN101084226A (zh) | 2004-12-20 | 2007-12-05 | 惠氏公司 | 雷帕霉素衍生物及其治疗神经紊乱的用途 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9221220D0 (en) * | 1992-10-09 | 1992-11-25 | Sandoz Ag | Organic componds |
-
1999
- 1999-08-16 JP JP2000564961A patent/JP2002522543A/ja active Pending
- 1999-08-16 ES ES99941166T patent/ES2179671T3/es not_active Expired - Lifetime
- 1999-08-16 AT AT99941166T patent/ATE219492T1/de not_active IP Right Cessation
- 1999-08-16 AU AU54874/99A patent/AU5487499A/en not_active Abandoned
- 1999-08-16 DK DK99941166T patent/DK1105395T3/da active
- 1999-08-16 BR BR9913052-1A patent/BR9913052A/pt not_active IP Right Cessation
- 1999-08-16 EP EP99941166A patent/EP1105395B1/en not_active Expired - Lifetime
- 1999-08-16 WO PCT/US1999/018564 patent/WO2000009510A1/en active IP Right Grant
- 1999-08-16 DE DE69901907T patent/DE69901907T2/de not_active Expired - Fee Related
- 1999-08-16 PT PT99941166T patent/PT1105395E/pt unknown
- 1999-08-16 CA CA002340700A patent/CA2340700A1/en not_active Abandoned
- 1999-08-16 CN CN99812174A patent/CN1323310A/zh active Pending
Also Published As
Publication number | Publication date |
---|---|
DE69901907D1 (de) | 2002-07-25 |
DE69901907T2 (de) | 2002-12-19 |
PT1105395E (pt) | 2002-09-30 |
DK1105395T3 (da) | 2002-10-14 |
EP1105395A1 (en) | 2001-06-13 |
WO2000009510A1 (en) | 2000-02-24 |
CN1323310A (zh) | 2001-11-21 |
JP2002522543A (ja) | 2002-07-23 |
AU5487499A (en) | 2000-03-06 |
CA2340700A1 (en) | 2000-02-24 |
ATE219492T1 (de) | 2002-07-15 |
EP1105395B1 (en) | 2002-06-19 |
ES2179671T3 (es) | 2003-01-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B25D | Requested change of name of applicant approved | ||
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 5A, 6A, 7A E 8A ANUIDADES |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1911 DE 21/08/2007. |