BR9505571A - Oligômero composto medicamento processo para a produção de um medicamento e uso - Google Patents

Oligômero composto medicamento processo para a produção de um medicamento e uso

Info

Publication number
BR9505571A
BR9505571A BR9505571A BR9505571A BR9505571A BR 9505571 A BR9505571 A BR 9505571A BR 9505571 A BR9505571 A BR 9505571A BR 9505571 A BR9505571 A BR 9505571A BR 9505571 A BR9505571 A BR 9505571A
Authority
BR
Brazil
Prior art keywords
medicine
production
oligomer compound
compound medicine
medicine process
Prior art date
Application number
BR9505571A
Other languages
English (en)
Inventor
Wen-Ren Li
Steve Yik-Kai Tam
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BR9505571A publication Critical patent/BR9505571A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H21/00Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
BR9505571A 1994-11-30 1995-11-29 Oligômero composto medicamento processo para a produção de um medicamento e uso BR9505571A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US34754194A 1994-11-30 1994-11-30

Publications (1)

Publication Number Publication Date
BR9505571A true BR9505571A (pt) 1997-11-04

Family

ID=23364154

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9505571A BR9505571A (pt) 1994-11-30 1995-11-29 Oligômero composto medicamento processo para a produção de um medicamento e uso

Country Status (8)

Country Link
EP (1) EP0714907A1 (pt)
JP (1) JPH08208686A (pt)
CN (1) CN1128269A (pt)
AR (1) AR002003A1 (pt)
BR (1) BR9505571A (pt)
CA (1) CA2163392A1 (pt)
FI (1) FI955767A (pt)
TR (1) TR199501521A2 (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6222025B1 (en) 1995-03-06 2001-04-24 Isis Pharmaceuticals, Inc. Process for the synthesis of 2′-O-substituted pyrimidines and oligomeric compounds therefrom
US6166197A (en) * 1995-03-06 2000-12-26 Isis Pharmaceuticals, Inc. Oligomeric compounds having pyrimidine nucleotide (S) with 2'and 5 substitutions
AU3340797A (en) * 1996-06-28 1998-01-21 Novartis Ag Modified oligonucleotides
DE60024906T2 (de) * 1999-03-05 2006-09-14 Tosoh Corp., Shinnanyo Eine am 3'-Ende modifizierte Nukleinsäuresonde, geeignet zur Hybridisierung und Detektion über Fluoreszenz
FR2804960B1 (fr) * 2000-02-11 2005-06-24 Lvmh Rech Nouveaux oligonucleotides et utilisation d'oligonucleotides modulant l'expression de la tyrosinase et de la tyrosinase- related-protein 1 comme agents depigmentants
WO2005092907A2 (en) * 2004-03-26 2005-10-06 Ranbaxy Laboratories Limited Monosaccharide derivatives as anti-cancer and anti-inflammatory agents
FR2864540B1 (fr) * 2005-02-22 2010-10-22 Lvmh Rech Nouveaux oligonucleotides et utilisation d'oligonucleotides modulant l'expression de la tyrosinase et de la tyrosinase-related-protein 1 comme agents depigmentants
US7820810B2 (en) 2007-03-19 2010-10-26 Isis Pharmaceuticals, Inc. Process for the synthesis of 2′-O-substituted purine nulceosides
GB201700595D0 (en) * 2017-01-13 2017-03-01 Univ Oxford Innovation Ltd Oligonucleotide ligation

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5378825A (en) * 1990-07-27 1995-01-03 Isis Pharmaceuticals, Inc. Backbone modified oligonucleotide analogs
EP0691977B1 (en) * 1993-03-31 1997-11-26 Sanofi Oligonucleotides with amide linkages replacing phosphodiester linkages

Also Published As

Publication number Publication date
AR002003A1 (es) 1998-01-07
CA2163392A1 (en) 1996-05-31
TR199501521A2 (tr) 1996-07-21
EP0714907A1 (en) 1996-06-05
FI955767A (fi) 1996-05-31
FI955767A0 (fi) 1995-11-30
CN1128269A (zh) 1996-08-07
JPH08208686A (ja) 1996-08-13

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Legal Events

Date Code Title Description
FA10 Dismissal: dismissal - article 33 of industrial property law
B15K Others concerning applications: alteration of classification

Ipc: C07H 19/06 (2006.01), C07H 19/04 (2006.0