BR6680359D0 - Um processo para a producao de derivados hidrogenados de tebaina e oripavina - Google Patents

Um processo para a producao de derivados hidrogenados de tebaina e oripavina

Info

Publication number
BR6680359D0
BR6680359D0 BR180359/66A BR18035966A BR6680359D0 BR 6680359 D0 BR6680359 D0 BR 6680359D0 BR 180359/66 A BR180359/66 A BR 180359/66A BR 18035966 A BR18035966 A BR 18035966A BR 6680359 D0 BR6680359 D0 BR 6680359D0
Authority
BR
Brazil
Prior art keywords
tebaina
oripavina
production
hydrogenated derivatives
hydrogenated
Prior art date
Application number
BR180359/66A
Other languages
English (en)
Portuguese (pt)
Inventor
K Bertley
Original Assignee
Reckitt & Sons Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Reckitt & Sons Ltd filed Critical Reckitt & Sons Ltd
Publication of BR6680359D0 publication Critical patent/BR6680359D0/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D489/00Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/09Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems
    • C07D489/10Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems with a bridge between positions 6 and 14
    • C07D489/12Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems with a bridge between positions 6 and 14 the bridge containing only two carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BR180359/66A 1965-06-15 1966-06-14 Um processo para a producao de derivados hidrogenados de tebaina e oripavina BR6680359D0 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB25289/65A GB1136214A (en) 1965-06-15 1965-06-15 Thebaine and oripavine derivatives

Publications (1)

Publication Number Publication Date
BR6680359D0 true BR6680359D0 (pt) 1973-12-26

Family

ID=10225305

Family Applications (1)

Application Number Title Priority Date Filing Date
BR180359/66A BR6680359D0 (pt) 1965-06-15 1966-06-14 Um processo para a producao de derivados hidrogenados de tebaina e oripavina

Country Status (14)

Country Link
AT (1) AT272530B (enrdf_load_stackoverflow)
BE (1) BE682551A (enrdf_load_stackoverflow)
BR (1) BR6680359D0 (enrdf_load_stackoverflow)
CH (1) CH558362A (enrdf_load_stackoverflow)
DE (1) DE1620206A1 (enrdf_load_stackoverflow)
DK (1) DK115926B (enrdf_load_stackoverflow)
ES (1) ES327925A1 (enrdf_load_stackoverflow)
FI (1) FI49724C (enrdf_load_stackoverflow)
FR (1) FR6395M (enrdf_load_stackoverflow)
GB (1) GB1136214A (enrdf_load_stackoverflow)
LU (1) LU51306A1 (enrdf_load_stackoverflow)
NL (1) NL6608255A (enrdf_load_stackoverflow)
NO (1) NO119590B (enrdf_load_stackoverflow)
SE (1) SE325276B (enrdf_load_stackoverflow)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2554816B1 (fr) * 1983-11-16 1986-09-26 Sanofi Sa Nouveau derive de la nororipavine presentant a la fois une activite agoniste et antagoniste des recepteurs morphiniques
KR100204659B1 (ko) * 1996-05-28 1999-06-15 강재헌 신규한 부프레노핀계 진통제용 화합물
RU2138502C1 (ru) * 1999-03-29 1999-09-27 Закрытое акционерное общество "РМА-Фарм" Способ получения 17-циклопропилметил-6,14-эндо-этано-7-(2-гидрокси-3,3-диметилбут-2-ил)тетр агидро-17-норорипавина
AUPQ968300A0 (en) 2000-08-25 2000-09-21 Glaxo Wellcome Australia Ltd Chemical methods
GB2388369B (en) 2002-05-10 2004-05-05 Reckitt Benckiser Healthcare Demethylation of thebaine derivative
GB0421687D0 (en) 2004-09-30 2004-11-03 Johnson Matthey Plc Preparation of opiate analgesics
WO2006091885A2 (en) 2005-02-24 2006-08-31 Dr Pharma Nova, Llc A registry method and control system for dea schedule ii-v medicines
DE102006054731B4 (de) 2006-11-21 2013-02-28 Lts Lohmann Therapie-Systeme Ag Transdermales therapeutisches System zur Verabreichung des Wirkstoffs Buprenorphin und Verwendung desselben in der Schmerztherapie
JP5525524B2 (ja) * 2008-07-30 2014-06-18 パーデュー、ファーマ、リミテッド、パートナーシップ ブプレノルフィン類似体
AU2009300386B2 (en) 2008-09-30 2015-07-02 SpecGx LLC Processes for the alkylation of norbuprenorphine with reduced impurity formation
CA2758231A1 (en) 2009-04-24 2010-10-28 Brock University Processes for the preparation of morphinane and morphinone compounds
GB201111775D0 (en) 2011-07-08 2011-08-24 Univ Bath Compounds and uses thereof
SG11201403162XA (en) 2011-12-12 2014-10-30 Lohmann Therapie Syst Lts Transdermal delivery system comprising buprenorphine
CA2879942C (en) 2012-07-26 2020-06-02 Camurus Ab Opioid formulations
EA034855B1 (ru) 2012-07-26 2020-03-30 Камурус Аб Предшественник депо-препарата, содержащий бупренорфин, и способ лечения путем его введения
US9175000B2 (en) * 2012-12-07 2015-11-03 Purdue Pharma L.P. Buprenorphine analogs
EA201592246A1 (ru) 2013-06-04 2016-05-31 Лтс Лохманн Терапи-Системе Аг Трансдермальная система доставки
EP4448501A1 (en) 2021-12-16 2024-10-23 Arevipharma GmbH Method of making buprenorphine and precursor compounds thereof

Also Published As

Publication number Publication date
GB1136214A (en) 1968-12-11
AT272530B (de) 1969-07-10
DK115926B (da) 1969-11-24
DE1620206A1 (de) 1970-03-19
SE325276B (enrdf_load_stackoverflow) 1970-06-29
CH558362A (de) 1975-01-31
FI49724B (enrdf_load_stackoverflow) 1975-06-02
BE682551A (enrdf_load_stackoverflow) 1966-11-14
FR6395M (enrdf_load_stackoverflow) 1968-10-21
LU51306A1 (enrdf_load_stackoverflow) 1966-08-16
NL6608255A (enrdf_load_stackoverflow) 1966-12-16
FI49724C (fi) 1975-09-10
NO119590B (enrdf_load_stackoverflow) 1970-06-08
ES327925A1 (es) 1967-04-01

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