BR112023021257A2 - Métodos para a administração combinada de deutetrabenzina e um cyp2d6 - Google Patents
Métodos para a administração combinada de deutetrabenzina e um cyp2d6Info
- Publication number
- BR112023021257A2 BR112023021257A2 BR112023021257A BR112023021257A BR112023021257A2 BR 112023021257 A2 BR112023021257 A2 BR 112023021257A2 BR 112023021257 A BR112023021257 A BR 112023021257A BR 112023021257 A BR112023021257 A BR 112023021257A BR 112023021257 A2 BR112023021257 A2 BR 112023021257A2
- Authority
- BR
- Brazil
- Prior art keywords
- cyp2d6
- deutetrabenzine
- methods
- combined administration
- patient
- Prior art date
Links
- 108010001237 Cytochrome P-450 CYP2D6 Proteins 0.000 title abstract 4
- 102100021704 Cytochrome P450 2D6 Human genes 0.000 title abstract 2
- 239000003112 inhibitor Substances 0.000 abstract 2
- 208000012902 Nervous system disease Diseases 0.000 abstract 1
- 208000025966 Neurological disease Diseases 0.000 abstract 1
- 102000009659 Vesicular Monoamine Transport Proteins Human genes 0.000 abstract 1
- 108010020033 Vesicular Monoamine Transport Proteins Proteins 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 230000000926 neurological effect Effects 0.000 abstract 1
- 208000020016 psychiatric disease Diseases 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4525—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with oxygen as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/49—Cinchonan derivatives, e.g. quinine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Emergency Medicine (AREA)
- Psychology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
métodos para a administração combinada de deutetrabenzina e um cyp2d6. a presente invenção refere-se a um método para tratar uma doença ou distúrbio neurológico ou psiquiátrico em um paciente em necessidade do mesmo, compreendendo: administrar um inibidor do transportador vesicular de monoamina 2 (vmat2) ao paciente em necessidade do mesmo, sendo também administrado ao paciente um forte inibidor de citocromo p450 2d6 (cyp2d6).
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202163175378P | 2021-04-15 | 2021-04-15 | |
US202163189939P | 2021-05-18 | 2021-05-18 | |
US202163238500P | 2021-08-30 | 2021-08-30 | |
PCT/US2022/024840 WO2022221546A1 (en) | 2021-04-15 | 2022-04-14 | Methods for the combined administration of deutetrabenazine and a cyp2d6 inhibitor |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112023021257A2 true BR112023021257A2 (pt) | 2023-12-12 |
Family
ID=81581216
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112023021257A BR112023021257A2 (pt) | 2021-04-15 | 2022-04-14 | Métodos para a administração combinada de deutetrabenzina e um cyp2d6 |
Country Status (6)
Country | Link |
---|---|
US (1) | US20240207247A1 (pt) |
EP (1) | EP4322934A1 (pt) |
JP (1) | JP2024514873A (pt) |
BR (1) | BR112023021257A2 (pt) |
IL (1) | IL307680A (pt) |
WO (1) | WO2022221546A1 (pt) |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4783443A (en) | 1986-03-03 | 1988-11-08 | The University Of Chicago | Amino acyl cephalosporin derivatives |
CN107624067A (zh) * | 2015-03-06 | 2018-01-23 | 奥斯拜客斯制药有限公司 | 用于治疗异常不自主运动障碍的方法 |
US10940141B1 (en) * | 2019-08-23 | 2021-03-09 | Neurocrine Biosciences, Inc. | Methods for the administration of certain VMAT2 inhibitors |
-
2022
- 2022-04-14 IL IL307680A patent/IL307680A/en unknown
- 2022-04-14 EP EP22721568.8A patent/EP4322934A1/en active Pending
- 2022-04-14 WO PCT/US2022/024840 patent/WO2022221546A1/en active Application Filing
- 2022-04-14 US US18/286,935 patent/US20240207247A1/en active Pending
- 2022-04-14 BR BR112023021257A patent/BR112023021257A2/pt unknown
- 2022-04-14 JP JP2023562890A patent/JP2024514873A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
US20240207247A1 (en) | 2024-06-27 |
JP2024514873A (ja) | 2024-04-03 |
IL307680A (en) | 2023-12-01 |
WO2022221546A1 (en) | 2022-10-20 |
EP4322934A1 (en) | 2024-02-21 |
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