BR112023019309A2 - Tratamento de hidradenite supurativa com orismilaste - Google Patents
Tratamento de hidradenite supurativa com orismilasteInfo
- Publication number
- BR112023019309A2 BR112023019309A2 BR112023019309A BR112023019309A BR112023019309A2 BR 112023019309 A2 BR112023019309 A2 BR 112023019309A2 BR 112023019309 A BR112023019309 A BR 112023019309A BR 112023019309 A BR112023019309 A BR 112023019309A BR 112023019309 A2 BR112023019309 A2 BR 112023019309A2
- Authority
- BR
- Brazil
- Prior art keywords
- treatment
- hidradenitis suppurativa
- orismilaste
- suppurativa
- hidradenitis
- Prior art date
Links
- 208000002557 hidradenitis Diseases 0.000 title abstract 3
- 201000007162 hidradenitis suppurativa Diseases 0.000 title abstract 3
- ZININGNRPUGNSL-UHFFFAOYSA-N 2-(3,5-dichloro-1-oxidopyridin-1-ium-4-yl)-1-[7-(difluoromethoxy)-1',1'-dioxospiro[1,3-benzodioxole-2,4'-thiane]-4-yl]ethanone Chemical compound ClC1=C[N+]([O-])=CC(Cl)=C1CC(=O)C1=CC=C(OC(F)F)C2=C1OC1(CCS(=O)(=O)CC1)O2 ZININGNRPUGNSL-UHFFFAOYSA-N 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 229940016320 orismilast Drugs 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/10—Spiro-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4436—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/2853—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4891—Coated capsules; Multilayered drug free capsule shells
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Dermatology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Treatments Of Macromolecular Shaped Articles (AREA)
- Medicinal Preparation (AREA)
Abstract
tratamento de hidradenite supurativa com orismilaste. um composto de fórmula ou um sal, solvato ou hidrato farmaceuticamente aceitável do mesmo, para uso no tratamento de hidradenite supurativa (hs) em um indivíduo.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB2103975.5A GB202103975D0 (en) | 2021-03-22 | 2021-03-22 | Treatment of HS |
GB202118420 | 2021-12-17 | ||
GB202201381 | 2022-02-03 | ||
PCT/EP2022/057472 WO2022200339A1 (en) | 2021-03-22 | 2022-03-22 | Treatment of hidradenitis suppurativa with orismilast |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112023019309A2 true BR112023019309A2 (pt) | 2023-10-31 |
Family
ID=81346285
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112023019309A BR112023019309A2 (pt) | 2021-03-22 | 2022-03-22 | Tratamento de hidradenite supurativa com orismilaste |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP4313043A1 (pt) |
JP (1) | JP2024511141A (pt) |
KR (1) | KR20230159485A (pt) |
AU (1) | AU2022245186A1 (pt) |
BR (1) | BR112023019309A2 (pt) |
CA (1) | CA3212316A1 (pt) |
IL (1) | IL306020A (pt) |
WO (1) | WO2022200339A1 (pt) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB202205715D0 (en) * | 2022-04-19 | 2022-06-01 | Union Therapeutics As | Treatment of neutrophilic dermatoses |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2585469B1 (en) | 2010-06-24 | 2016-05-25 | Leo Pharma A/S | Benzodioxole or benzodioxepine heterocyclic compounds as phosphodiesterase inhibitors |
JP6785666B2 (ja) | 2014-06-23 | 2020-11-18 | レオ ファーマ アクティーゼルスカブ | 1,3−ベンゾジオキソール複素環化合物の調製方法 |
ES2961237T3 (es) | 2015-12-18 | 2024-03-11 | Union Therapeutics As | Métodos para la preparación de compuestos heterocíclicos de 1,3-benzodioxol |
CA3064033A1 (en) | 2017-06-20 | 2018-12-27 | Leo Pharma A/S | Methods for the preparation of 1,3-benzodioxole heterocyclic compounds |
EP3911304B1 (en) | 2019-01-15 | 2023-09-06 | UNION therapeutics A/S | Modified release tablet formulations containing phosphodiesterase inhibitors |
-
2022
- 2022-03-22 BR BR112023019309A patent/BR112023019309A2/pt unknown
- 2022-03-22 IL IL306020A patent/IL306020A/en unknown
- 2022-03-22 WO PCT/EP2022/057472 patent/WO2022200339A1/en active Application Filing
- 2022-03-22 CA CA3212316A patent/CA3212316A1/en active Pending
- 2022-03-22 EP EP22717748.2A patent/EP4313043A1/en active Pending
- 2022-03-22 AU AU2022245186A patent/AU2022245186A1/en active Pending
- 2022-03-22 KR KR1020237035255A patent/KR20230159485A/ko unknown
- 2022-03-22 JP JP2023558591A patent/JP2024511141A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
WO2022200339A1 (en) | 2022-09-29 |
EP4313043A1 (en) | 2024-02-07 |
AU2022245186A1 (en) | 2023-10-05 |
IL306020A (en) | 2023-11-01 |
CA3212316A1 (en) | 2022-09-29 |
KR20230159485A (ko) | 2023-11-21 |
JP2024511141A (ja) | 2024-03-12 |
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