BR112023019309A2 - Tratamento de hidradenite supurativa com orismilaste - Google Patents

Tratamento de hidradenite supurativa com orismilaste

Info

Publication number
BR112023019309A2
BR112023019309A2 BR112023019309A BR112023019309A BR112023019309A2 BR 112023019309 A2 BR112023019309 A2 BR 112023019309A2 BR 112023019309 A BR112023019309 A BR 112023019309A BR 112023019309 A BR112023019309 A BR 112023019309A BR 112023019309 A2 BR112023019309 A2 BR 112023019309A2
Authority
BR
Brazil
Prior art keywords
treatment
hidradenitis suppurativa
orismilaste
suppurativa
hidradenitis
Prior art date
Application number
BR112023019309A
Other languages
English (en)
Inventor
Anne Weiss
Hjardem Taudorf Elisabeth
B E Jemec Gregor
Kim Kjøller
Morten Sommer
Philippe Andres
Original Assignee
Union Therapeutics As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB2103975.5A external-priority patent/GB202103975D0/en
Application filed by Union Therapeutics As filed Critical Union Therapeutics As
Publication of BR112023019309A2 publication Critical patent/BR112023019309A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/10Spiro-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4436Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/2853Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4866Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4891Coated capsules; Multilayered drug free capsule shells
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/10Anti-acne agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Treatments Of Macromolecular Shaped Articles (AREA)
  • Medicinal Preparation (AREA)

Abstract

tratamento de hidradenite supurativa com orismilaste. um composto de fórmula ou um sal, solvato ou hidrato farmaceuticamente aceitável do mesmo, para uso no tratamento de hidradenite supurativa (hs) em um indivíduo.
BR112023019309A 2021-03-22 2022-03-22 Tratamento de hidradenite supurativa com orismilaste BR112023019309A2 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GBGB2103975.5A GB202103975D0 (en) 2021-03-22 2021-03-22 Treatment of HS
GB202118420 2021-12-17
GB202201381 2022-02-03
PCT/EP2022/057472 WO2022200339A1 (en) 2021-03-22 2022-03-22 Treatment of hidradenitis suppurativa with orismilast

Publications (1)

Publication Number Publication Date
BR112023019309A2 true BR112023019309A2 (pt) 2023-10-31

Family

ID=81346285

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112023019309A BR112023019309A2 (pt) 2021-03-22 2022-03-22 Tratamento de hidradenite supurativa com orismilaste

Country Status (8)

Country Link
EP (1) EP4313043A1 (pt)
JP (1) JP2024511141A (pt)
KR (1) KR20230159485A (pt)
AU (1) AU2022245186A1 (pt)
BR (1) BR112023019309A2 (pt)
CA (1) CA3212316A1 (pt)
IL (1) IL306020A (pt)
WO (1) WO2022200339A1 (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB202205715D0 (en) * 2022-04-19 2022-06-01 Union Therapeutics As Treatment of neutrophilic dermatoses

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2585469B1 (en) 2010-06-24 2016-05-25 Leo Pharma A/S Benzodioxole or benzodioxepine heterocyclic compounds as phosphodiesterase inhibitors
JP6785666B2 (ja) 2014-06-23 2020-11-18 レオ ファーマ アクティーゼルスカブ 1,3−ベンゾジオキソール複素環化合物の調製方法
ES2961237T3 (es) 2015-12-18 2024-03-11 Union Therapeutics As Métodos para la preparación de compuestos heterocíclicos de 1,3-benzodioxol
CA3064033A1 (en) 2017-06-20 2018-12-27 Leo Pharma A/S Methods for the preparation of 1,3-benzodioxole heterocyclic compounds
EP3911304B1 (en) 2019-01-15 2023-09-06 UNION therapeutics A/S Modified release tablet formulations containing phosphodiesterase inhibitors

Also Published As

Publication number Publication date
WO2022200339A1 (en) 2022-09-29
EP4313043A1 (en) 2024-02-07
AU2022245186A1 (en) 2023-10-05
IL306020A (en) 2023-11-01
CA3212316A1 (en) 2022-09-29
KR20230159485A (ko) 2023-11-21
JP2024511141A (ja) 2024-03-12

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