BR112018012701A2 - novos compostos de 1,2,3 triazol-tiazol, processo para preparação e utilização dos mesmos - Google Patents
novos compostos de 1,2,3 triazol-tiazol, processo para preparação e utilização dos mesmosInfo
- Publication number
- BR112018012701A2 BR112018012701A2 BR112018012701A BR112018012701A BR112018012701A2 BR 112018012701 A2 BR112018012701 A2 BR 112018012701A2 BR 112018012701 A BR112018012701 A BR 112018012701A BR 112018012701 A BR112018012701 A BR 112018012701A BR 112018012701 A2 BR112018012701 A2 BR 112018012701A2
- Authority
- BR
- Brazil
- Prior art keywords
- novel
- preparation
- processes
- thiazole compounds
- triazole
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Treatment Of Liquids With Adsorbents In General (AREA)
Abstract
?novos compostos de 1,2,3 triazol-tiazol, processo para preparação e utilização dos mesmos?, a presente invenção divulga um novo composto de 1,2,3-triazol-tiazol de fórmula (i) ou sal farmaceuticamente aceitável do mesmo, processo para sua preparação, sua composição farmacêutica e método para o tratamento para impedir a disseminação de vitiligo ou fornecer benefício profilático aos indivíduos com predisposição a vitiligo.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN4189DE2015 | 2015-12-21 | ||
PCT/IN2016/050449 WO2017109793A1 (en) | 2015-12-21 | 2016-12-20 | Novel 1,2,3 triazole-thiazole compounds, process for preparation and use thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112018012701A2 true BR112018012701A2 (pt) | 2018-12-04 |
Family
ID=58191512
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112018012701A BR112018012701A2 (pt) | 2015-12-21 | 2016-12-20 | novos compostos de 1,2,3 triazol-tiazol, processo para preparação e utilização dos mesmos |
Country Status (6)
Country | Link |
---|---|
US (1) | US10246449B2 (pt) |
EP (1) | EP3394054B1 (pt) |
JP (1) | JP6586528B2 (pt) |
BR (1) | BR112018012701A2 (pt) |
SG (1) | SG11201805237TA (pt) |
WO (1) | WO2017109793A1 (pt) |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0028383D0 (en) | 2000-11-21 | 2001-01-03 | Novartis Ag | Organic compounds |
US7259262B2 (en) * | 2003-10-24 | 2007-08-21 | Hoffmann-La Roche Inc. | Arylazole derivatives, their manufacture and use as pharmaceutical agents |
KR20080047591A (ko) * | 2005-09-07 | 2008-05-29 | 플렉시콘, 인코퍼레이티드 | Ppar 조절인자로서 사용하기 위한 1,3-이치환된 인돌유도체 |
WO2007087427A2 (en) * | 2006-01-25 | 2007-08-02 | Synta Pharmaceuticals Corp. | Thiazole and thiadiazole compounds for inflammation and immune-related uses |
EP2464635B1 (en) | 2009-08-11 | 2015-09-16 | The Scripps Research Institute | Copper catalyzed cycloaddition of organic azides and 1-haloalkynes |
US8377970B2 (en) * | 2009-10-08 | 2013-02-19 | Rhizen Pharmaceuticals Sa | Modulators of calcium release-activated calcium channel |
EP3092236B1 (en) * | 2014-01-06 | 2020-08-26 | Rhizen Pharmaceuticals S.A. | Novel glutaminase inhibitors |
-
2016
- 2016-12-20 WO PCT/IN2016/050449 patent/WO2017109793A1/en active Application Filing
- 2016-12-20 SG SG11201805237TA patent/SG11201805237TA/en unknown
- 2016-12-20 EP EP16840334.3A patent/EP3394054B1/en not_active Not-in-force
- 2016-12-20 BR BR112018012701A patent/BR112018012701A2/pt not_active Application Discontinuation
- 2016-12-20 JP JP2018532402A patent/JP6586528B2/ja not_active Expired - Fee Related
- 2016-12-20 US US16/064,415 patent/US10246449B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US10246449B2 (en) | 2019-04-02 |
WO2017109793A1 (en) | 2017-06-29 |
JP2019501168A (ja) | 2019-01-17 |
EP3394054A1 (en) | 2018-10-31 |
EP3394054B1 (en) | 2019-11-06 |
JP6586528B2 (ja) | 2019-10-02 |
US20180370962A1 (en) | 2018-12-27 |
SG11201805237TA (en) | 2018-07-30 |
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Legal Events
Date | Code | Title | Description |
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B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] |
Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS. |
|
B07E | Notice of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] | ||
B06U | Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette] | ||
B11B | Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements |