BR112017010602A2 - análogos de ureia ligados em ponte substituídos como moduladores de sirtuína - Google Patents

análogos de ureia ligados em ponte substituídos como moduladores de sirtuína

Info

Publication number
BR112017010602A2
BR112017010602A2 BR112017010602A BR112017010602A BR112017010602A2 BR 112017010602 A2 BR112017010602 A2 BR 112017010602A2 BR 112017010602 A BR112017010602 A BR 112017010602A BR 112017010602 A BR112017010602 A BR 112017010602A BR 112017010602 A2 BR112017010602 A2 BR 112017010602A2
Authority
BR
Brazil
Prior art keywords
disorders
diseases
sirtuin
modulators
substituted bridged
Prior art date
Application number
BR112017010602A
Other languages
English (en)
Portuguese (pt)
Inventor
Lamond Ellis James
Anderson Evans Karen
Andrew Seefeld Mark
Michael Fox Ryan
Henry Miller William
Original Assignee
Glaxosmithkline Ip No 2 Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Ip No 2 Ltd filed Critical Glaxosmithkline Ip No 2 Ltd
Publication of BR112017010602A2 publication Critical patent/BR112017010602A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/18Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/18Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4995Pyrazines or piperazines forming part of bridged ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/55131,4-Benzodiazepines, e.g. diazepam or clozapine
    • A61K31/55171,4-Benzodiazepines, e.g. diazepam or clozapine condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Obesity (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
BR112017010602A 2014-11-19 2015-11-19 análogos de ureia ligados em ponte substituídos como moduladores de sirtuína BR112017010602A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201462081916P 2014-11-19 2014-11-19
PCT/IB2015/058978 WO2016079710A1 (en) 2014-11-19 2015-11-19 Substituted bridged urea analogs as sirtuin modulators

Publications (1)

Publication Number Publication Date
BR112017010602A2 true BR112017010602A2 (pt) 2017-12-26

Family

ID=54705247

Family Applications (4)

Application Number Title Priority Date Filing Date
BR112017010602A BR112017010602A2 (pt) 2014-11-19 2015-11-19 análogos de ureia ligados em ponte substituídos como moduladores de sirtuína
BR112017010599A BR112017010599A2 (pt) 2014-11-19 2015-11-19 análogos de ureia ligada substituída como moduladores sirtuin
BR112017010601A BR112017010601A2 (pt) 2014-11-19 2015-11-19 análogos de ureia substituídos em ponte como moduladores de sirtuínas
BR112017010595-0A BR112017010595A2 (pt) 2014-11-19 2015-11-19 análogos de ureia com ligações por pontes substituídas como moduladores de sirtuína

Family Applications After (3)

Application Number Title Priority Date Filing Date
BR112017010599A BR112017010599A2 (pt) 2014-11-19 2015-11-19 análogos de ureia ligada substituída como moduladores sirtuin
BR112017010601A BR112017010601A2 (pt) 2014-11-19 2015-11-19 análogos de ureia substituídos em ponte como moduladores de sirtuínas
BR112017010595-0A BR112017010595A2 (pt) 2014-11-19 2015-11-19 análogos de ureia com ligações por pontes substituídas como moduladores de sirtuína

Country Status (21)

Country Link
US (4) US20170355705A1 (enExample)
EP (4) EP3221317B1 (enExample)
JP (4) JP2017534663A (enExample)
KR (4) KR20170087907A (enExample)
CN (4) CN107207520A (enExample)
AU (4) AU2015348944A1 (enExample)
BR (4) BR112017010602A2 (enExample)
CA (4) CA2968032A1 (enExample)
CL (1) CL2017001275A1 (enExample)
CO (1) CO2017004994A2 (enExample)
CR (1) CR20170209A (enExample)
DO (1) DOP2017000123A (enExample)
EA (1) EA201791074A1 (enExample)
ES (1) ES2823748T3 (enExample)
IL (1) IL252252A0 (enExample)
MX (1) MX2017006658A (enExample)
PE (1) PE20171257A1 (enExample)
PH (1) PH12017500913A1 (enExample)
RU (3) RU2017120855A (enExample)
SG (1) SG11201703824QA (enExample)
WO (4) WO2016079712A1 (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016086088A2 (en) 2014-11-25 2016-06-02 Northwestern University Wound healing through sirt1 overexpression
CN108329388A (zh) * 2018-01-18 2018-07-27 天津市湖滨盘古基因科学发展有限公司 一种人的沉默配型信息调节蛋白突变蛋白及其应用
CN108707150B (zh) * 2018-05-14 2021-04-16 江苏惠利生物科技有限公司 一种咪唑并吡嗪医药中间体的制备方法
CN108395436B (zh) * 2018-05-14 2021-01-12 鹤壁市人民医院 一种咪唑并吡嗪医药中间体的制备方法
CN110478339A (zh) * 2019-08-12 2019-11-22 昆明理工大学 紫铆因在制备靶向恢复突变p53构象药物中的应用
EP4025566A1 (de) * 2019-09-02 2022-07-13 Merck Patent GmbH Materialien für organische elektrolumineszenzvorrichtungen
BR112022009649A2 (pt) * 2019-11-19 2022-08-16 Lupin Ltd Processo, intermediários e métodos para preparar compostos de cromano
FI4090654T3 (fi) * 2020-01-17 2025-09-30 Lupin Ltd Menetelmiä, prosesseja ja välituotteita kromaaniyhdisteiden valmistamiseksi
CN114890955A (zh) * 2022-06-23 2022-08-12 江西瑞威尔生物科技有限公司 一种n取代吗啉类有机化合物的制备工艺

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4727064A (en) 1984-04-25 1988-02-23 The United States Of America As Represented By The Department Of Health And Human Services Pharmaceutical preparations containing cyclodextrin derivatives
US4683195A (en) 1986-01-30 1987-07-28 Cetus Corporation Process for amplifying, detecting, and/or-cloning nucleic acid sequences
WO2006094210A2 (en) * 2005-03-03 2006-09-08 Sirtris Pharmaceuticals, Inc. Tetrahydroquinoxalinone sirtuin modulators
UA108596C2 (xx) 2007-11-09 2015-05-25 Інгібітори пептиддеформілази
CA2779303A1 (en) * 2009-10-29 2011-05-19 Sirtris Pharmaceuticals, Inc. Bicyclic pyridines and analogs as sirtuin modulators
AU2012352442A1 (en) * 2011-12-12 2014-07-03 Smb Innovation Aps Novel heterocyclic compounds useful in sirtuin binding and modulation
WO2014186313A1 (en) * 2013-05-13 2014-11-20 Glaxosmithkline Llc Substituted bridged urea analogs as sirtuin modulators

Also Published As

Publication number Publication date
CA2968030A1 (en) 2016-05-26
WO2016079709A1 (en) 2016-05-26
BR112017010601A2 (pt) 2017-12-26
RU2017120857A (ru) 2018-12-19
CN107108627A (zh) 2017-08-29
JP6806679B2 (ja) 2021-01-06
BR112017010595A2 (pt) 2018-01-02
EP3221317B1 (en) 2020-07-22
US20190048016A1 (en) 2019-02-14
WO2016079711A1 (en) 2016-05-26
DOP2017000123A (es) 2017-08-15
AU2015348944A1 (en) 2017-06-01
KR20170087907A (ko) 2017-07-31
CA2968027A1 (en) 2016-05-26
CA2968029A1 (en) 2016-05-26
US20170355705A1 (en) 2017-12-14
RU2017120855A (ru) 2018-12-19
CN107207509B (zh) 2020-04-21
AU2015348942B2 (en) 2018-07-05
PE20171257A1 (es) 2017-08-28
CO2017004994A2 (es) 2017-09-20
RU2017120858A (ru) 2018-12-19
EP3221322A1 (en) 2017-09-27
US10072011B2 (en) 2018-09-11
MX2017006658A (es) 2018-01-15
JP2017534665A (ja) 2017-11-24
CR20170209A (es) 2017-07-17
CN107207520A (zh) 2017-09-26
WO2016079712A1 (en) 2016-05-26
AU2015348942A1 (en) 2017-06-01
EP3220918A1 (en) 2017-09-27
ES2823748T3 (es) 2021-05-10
EP3221317A1 (en) 2017-09-27
CN107207509A (zh) 2017-09-26
KR20170083133A (ko) 2017-07-17
IL252252A0 (en) 2017-07-31
US20170362234A1 (en) 2017-12-21
KR20170083135A (ko) 2017-07-17
JP2017534664A (ja) 2017-11-24
PH12017500913A1 (en) 2017-12-04
JP2017534662A (ja) 2017-11-24
CN107207521A (zh) 2017-09-26
BR112017010599A2 (pt) 2017-12-26
CA2968032A1 (en) 2016-05-26
CL2017001275A1 (es) 2017-12-15
EA201791074A1 (ru) 2017-10-31
WO2016079710A1 (en) 2016-05-26
AU2015348943A1 (en) 2017-06-01
KR20170083134A (ko) 2017-07-17
AU2015348941A1 (en) 2017-06-01
JP2017534663A (ja) 2017-11-24
US20180319810A1 (en) 2018-11-08
EP3221316A1 (en) 2017-09-27
SG11201703824QA (en) 2017-06-29

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements