BR112015025816A2 - processo para a preparação de drospirenona - Google Patents

processo para a preparação de drospirenona

Info

Publication number
BR112015025816A2
BR112015025816A2 BR112015025816A BR112015025816A BR112015025816A2 BR 112015025816 A2 BR112015025816 A2 BR 112015025816A2 BR 112015025816 A BR112015025816 A BR 112015025816A BR 112015025816 A BR112015025816 A BR 112015025816A BR 112015025816 A2 BR112015025816 A2 BR 112015025816A2
Authority
BR
Brazil
Prior art keywords
drospirenone
preparation
ÿþr
Prior art date
Application number
BR112015025816A
Other languages
English (en)
Other versions
BR112015025816B1 (pt
Inventor
Barbieri Francesco
Giovanna Luoni Maria
Noseda Monica
Lenna Roberto
Original Assignee
Ind Chimica Srl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ind Chimica Srl filed Critical Ind Chimica Srl
Publication of BR112015025816A2 publication Critical patent/BR112015025816A2/pt
Publication of BR112015025816B1 publication Critical patent/BR112015025816B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • C07J53/004—3 membered carbocyclic rings
    • C07J53/008—3 membered carbocyclic rings in position 15/16
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Reproductive Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Endocrinology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

ÿþr
BR112015025816-6A 2013-04-12 2013-04-12 processo para a preparação de drospirenona BR112015025816B1 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/IB2013/052918 WO2014167386A1 (en) 2013-04-12 2013-04-12 Process for the preparation of drospirenone

Publications (2)

Publication Number Publication Date
BR112015025816A2 true BR112015025816A2 (pt) 2017-07-25
BR112015025816B1 BR112015025816B1 (pt) 2021-02-02

Family

ID=48539320

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015025816-6A BR112015025816B1 (pt) 2013-04-12 2013-04-12 processo para a preparação de drospirenona

Country Status (14)

Country Link
US (1) US9556220B2 (pt)
EP (1) EP2984100B1 (pt)
JP (1) JP6469078B2 (pt)
CN (1) CN105164144B (pt)
AR (1) AR095833A1 (pt)
BR (1) BR112015025816B1 (pt)
CA (1) CA2909087C (pt)
DK (1) DK2984100T3 (pt)
ES (1) ES2630331T3 (pt)
HU (1) HUE032858T2 (pt)
MX (1) MX356791B (pt)
PL (1) PL2984100T3 (pt)
PT (1) PT2984100T (pt)
WO (1) WO2014167386A1 (pt)

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3042136A1 (de) 1980-11-03 1982-06-09 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur herstellung von 3 (beta), 7 (beta) -dihydroxy- (delta) (pfeil hoch)5(pfeil hoch) -steroiden
EP0075189B1 (en) 1981-09-21 1985-08-28 Schering Aktiengesellschaft 3-beta,7-beta,15-alpha-trihydroxy-5-androsten-17-one, its 3,15-dipivalate, and its preparation
DE19633685C1 (de) * 1996-08-12 1997-10-09 Schering Ag Verfahren zur Herstellung von Drospirenon (6beta,7beta;15 beta,16beta-Dimethyl-en-3-oxo-17alpha-pregn-4-en-21,17-carbolacton, DRSP) sowie 7alpha-(3-Hydroxy-1-propyl)-6beta,7beta;15beta, 16beta-dimethylen-5beta-androstan-3beta,5,17beta-triol (ZK 92836) und 6beta,7beta;15beta,16beta-dimethylen-5beta-hydroxy-3-oxo-17alpha-androstan-21,17-carbolacton (90965) als Zwischenprodukte des Verfahrens
JP4645779B2 (ja) * 2000-05-16 2011-03-09 日産化学工業株式会社 キノリンカルボアルデヒドの製造法
ITMI20040367A1 (it) * 2004-03-01 2004-06-01 Ind Chimica Srl Processo per la preparazione di drospirenone
ITMI20042338A1 (it) 2004-12-06 2005-03-06 Ind Chimica Srl Processo per la preparazione di drospirenone
DE502005004948D1 (de) * 2005-07-21 2008-09-18 Bayer Schering Pharma Ag Verfahren zur Herstellung von 3-Oxo-pregn-4-en-21,17-carbolactonen durch die metallfreie Oxidation von 17-(3-hydroxypropyl)-3,17-dihydroxyandrostanen
CN100480256C (zh) * 2006-06-21 2009-04-22 上海迪赛诺医药发展有限公司 合成曲螺酮的方法
WO2008137050A2 (en) * 2007-05-01 2008-11-13 Sicor Inc. A process for preparing drospirenone and intermediate thereof
RS51892B (en) * 2007-07-26 2012-02-29 Newchem S.P.A. DROSPIRENON PREPARATION PROCESS
CN101503455B (zh) 2009-03-11 2011-02-16 药源药物化学（上海）有限公司 一种制备屈螺酮的方法及中间体
ES2432063T3 (es) 2009-06-16 2013-11-29 Crystal Pharma, S.A.U. Procedimiento para la obtención de 17-espirolactonas en esteroides
ES2419663T3 (es) * 2010-08-03 2013-08-21 Newchem S.P.A. Métodos para la preparación de Drospirenona y productos intermedios de la misma

Also Published As

Publication number Publication date
US20160052960A1 (en) 2016-02-25
JP6469078B2 (ja) 2019-02-13
BR112015025816B1 (pt) 2021-02-02
CN105164144A (zh) 2015-12-16
PT2984100T (pt) 2017-07-14
AR095833A1 (es) 2015-11-11
WO2014167386A1 (en) 2014-10-16
HUE032858T2 (en) 2017-11-28
JP2016516095A (ja) 2016-06-02
CA2909087A1 (en) 2014-10-16
PL2984100T3 (pl) 2017-10-31
DK2984100T3 (en) 2017-07-10
ES2630331T3 (es) 2017-08-21
US9556220B2 (en) 2017-01-31
CN105164144B (zh) 2017-03-08
EP2984100B1 (en) 2017-04-05
MX356791B (es) 2018-06-12
CA2909087C (en) 2020-01-07
MX2015014331A (es) 2015-12-08
EP2984100A1 (en) 2016-02-17

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according art. 34 industrial property law
B07E Notice of approval relating to section 229 industrial property law
B06U Preliminary requirement: requests with searches performed by other patent offices: suspension of the patent application procedure
B09A Decision: intention to grant
B16A Patent or certificate of addition of invention granted

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 12/04/2013, OBSERVADAS AS CONDICOES LEGAIS.