BR0315046A - Intermediários na preparação de aminoácidos bicìclicos fundidos terapêuticos - Google Patents
Intermediários na preparação de aminoácidos bicìclicos fundidos terapêuticosInfo
- Publication number
- BR0315046A BR0315046A BR0315046-1A BR0315046A BR0315046A BR 0315046 A BR0315046 A BR 0315046A BR 0315046 A BR0315046 A BR 0315046A BR 0315046 A BR0315046 A BR 0315046A
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- amino acids
- fused bicyclic
- intermediates
- bicyclic amino
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/608—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a ring other than a six-membered aromatic ring in the acid moiety
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/347—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups
- C07C51/353—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups by isomerisation; by change of size of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C53/00—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
- C07C53/132—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen containing rings
- C07C53/136—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen containing rings containing condensed ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
- C07C57/26—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing rings other than six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C67/00—Preparation of carboxylic acid esters
- C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
- C07C67/333—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton
- C07C67/343—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/14—All rings being cycloaliphatic
- C07C2602/20—All rings being cycloaliphatic the ring system containing seven carbon atoms
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
"INTERMEDIáRIOS NA PREPARAçãO DE AMINOáCIDOS BICìCLICOS FUNDIDOS TERAPêUTICOS". A invenção apresenta compostos com a fórmula (I), em que R representa H ou um grupo protetor de ácido carboxílico adequado, que são intermediários na preparação de aminoácidos bicíclicos fundidos terapêuticos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0223070.4A GB0223070D0 (en) | 2002-10-04 | 2002-10-04 | Intermediates in the preparation of therapeutic fused bicyclic amino acids |
PCT/IB2003/004179 WO2004031115A1 (en) | 2002-10-04 | 2003-09-22 | Intermediates in the preparation of therapeutic fused bicyclic amino acids |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0315046A true BR0315046A (pt) | 2005-08-16 |
Family
ID=9945336
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0315046-1A BR0315046A (pt) | 2002-10-04 | 2003-09-22 | Intermediários na preparação de aminoácidos bicìclicos fundidos terapêuticos |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP1551789A1 (pt) |
JP (1) | JP2006501296A (pt) |
AU (1) | AU2003263487A1 (pt) |
BR (1) | BR0315046A (pt) |
CA (1) | CA2499863A1 (pt) |
GB (1) | GB0223070D0 (pt) |
MX (1) | MXPA05003638A (pt) |
WO (1) | WO2004031115A1 (pt) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN110818550A (zh) * | 2019-11-25 | 2020-02-21 | 东华理工大学 | 一种选择性酶促水解反应制备右旋异丁苯丙酸的方法 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PL366406A1 (en) * | 2001-04-19 | 2005-01-24 | Warner-Lambert Company Llc | Fused bicyclic or tricyclic amino acids |
-
2002
- 2002-10-04 GB GBGB0223070.4A patent/GB0223070D0/en not_active Ceased
-
2003
- 2003-09-22 CA CA002499863A patent/CA2499863A1/en not_active Abandoned
- 2003-09-22 BR BR0315046-1A patent/BR0315046A/pt not_active IP Right Cessation
- 2003-09-22 JP JP2004541065A patent/JP2006501296A/ja not_active Withdrawn
- 2003-09-22 EP EP03799019A patent/EP1551789A1/en not_active Withdrawn
- 2003-09-22 AU AU2003263487A patent/AU2003263487A1/en not_active Abandoned
- 2003-09-22 MX MXPA05003638A patent/MXPA05003638A/es unknown
- 2003-09-22 WO PCT/IB2003/004179 patent/WO2004031115A1/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
EP1551789A1 (en) | 2005-07-13 |
CA2499863A1 (en) | 2004-04-15 |
AU2003263487A1 (en) | 2004-04-23 |
MXPA05003638A (es) | 2005-06-03 |
WO2004031115A1 (en) | 2004-04-15 |
GB0223070D0 (en) | 2002-11-13 |
JP2006501296A (ja) | 2006-01-12 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application fees: dismissal - article 86 of industrial property law |
Free format text: REFERENTE 6A. E 7A. ANUIDADES. |
|
B08K | Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87) |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2069 DE 31/08/2010. |