BR0308060A - Base de citalopram, métodos para purificar a base de citalopram, para fabricar um sal de citalopram e para fabricar uma base de citalopram amorfa, sal de citalopram, e, composição farmacêutica - Google Patents

Base de citalopram, métodos para purificar a base de citalopram, para fabricar um sal de citalopram e para fabricar uma base de citalopram amorfa, sal de citalopram, e, composição farmacêutica

Info

Publication number
BR0308060A
BR0308060A BR0308060-9A BR0308060A BR0308060A BR 0308060 A BR0308060 A BR 0308060A BR 0308060 A BR0308060 A BR 0308060A BR 0308060 A BR0308060 A BR 0308060A
Authority
BR
Brazil
Prior art keywords
citalopram
base
salt
making
purifying
Prior art date
Application number
BR0308060-9A
Other languages
English (en)
Inventor
Yusuf Khwaja Hamied
Rajendra N Kankan
Dharmaraj R Rao
Original Assignee
Cipla Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cipla Ltd filed Critical Cipla Ltd
Publication of BR0308060A publication Critical patent/BR0308060A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87Benzo [c] furans; Hydrogenated benzo [c] furans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

"BASE DE CITALOPRAM , MéTODOS PARA PURIFICAR A BASE DE CITALOPRAM, PARA FABRICAR UM SAL DE CITALOPRAM E PARA FABRICAR UMA BASE DE CITALOPRAM AMORFA, SAL DE CITALOPRAM, E, COMPOSIçãO FARMACêUTICA". Base de citalopram é purificada e isolada por cromatografia.
BR0308060-9A 2002-02-27 2003-02-26 Base de citalopram, métodos para purificar a base de citalopram, para fabricar um sal de citalopram e para fabricar uma base de citalopram amorfa, sal de citalopram, e, composição farmacêutica BR0308060A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB0204680A GB2386118A (en) 2002-02-27 2002-02-27 Citalopram
PCT/GB2003/000810 WO2003072562A1 (en) 2002-02-27 2003-02-26 Amorphous citalopram

Publications (1)

Publication Number Publication Date
BR0308060A true BR0308060A (pt) 2004-12-28

Family

ID=9931949

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0308060-9A BR0308060A (pt) 2002-02-27 2003-02-26 Base de citalopram, métodos para purificar a base de citalopram, para fabricar um sal de citalopram e para fabricar uma base de citalopram amorfa, sal de citalopram, e, composição farmacêutica

Country Status (6)

Country Link
EP (1) EP1478636B1 (pt)
AU (1) AU2003207348A1 (pt)
BR (1) BR0308060A (pt)
DE (1) DE60324772D1 (pt)
GB (1) GB2386118A (pt)
WO (1) WO2003072562A1 (pt)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS617267A (ja) * 1984-06-20 1986-01-13 Otsuka Pharmaceut Co Ltd 新規フタライド誘導体
GB2357762B (en) * 2000-03-13 2002-01-30 Lundbeck & Co As H Crystalline base of citalopram

Also Published As

Publication number Publication date
EP1478636B1 (en) 2008-11-19
WO2003072562A1 (en) 2003-09-04
DE60324772D1 (de) 2009-01-02
AU2003207348A1 (en) 2003-09-09
GB0204680D0 (en) 2002-04-17
EP1478636A1 (en) 2004-11-24
GB2386118A (en) 2003-09-10

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Legal Events

Date Code Title Description
B11Y Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired