BR0116657A - Composto, processo para a preparação do mesmo, composição para controlar e proteger contra microrganismos fitopatogênicos, uso de um composto, e, método para controlar e evitar a infestação por microrganismos fitopatogênicos em plantações - Google Patents

Composto, processo para a preparação do mesmo, composição para controlar e proteger contra microrganismos fitopatogênicos, uso de um composto, e, método para controlar e evitar a infestação por microrganismos fitopatogênicos em plantações

Info

Publication number
BR0116657A
BR0116657A BR0116657-3A BR0116657A BR0116657A BR 0116657 A BR0116657 A BR 0116657A BR 0116657 A BR0116657 A BR 0116657A BR 0116657 A BR0116657 A BR 0116657A
Authority
BR
Brazil
Prior art keywords
sub
alkyl
controlling
hydrogen
haloalkyl
Prior art date
Application number
BR0116657-3A
Other languages
English (en)
Other versions
BR0116657B1 (pt
Inventor
Martin Eberle
Hugo Ziegler
Fredrik Cederbaum
Peter Ackermann
Anita Schnyder
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of BR0116657A publication Critical patent/BR0116657A/pt
Publication of BR0116657B1 publication Critical patent/BR0116657B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D419/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms
    • C07D419/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

"COMPOSTO, PROCESSO PARA A PREPARAçãO DO MESMO, COMPOSIçãO PARA CONTROLAR E PROTEGER CONTRA MICRORGANISMOS FITOPATOGêNICOS, USO DE UM COMPOSTO, E, MéTODO PARA CONTROLAR E EVITAR A INFESTAçãO POR MICRORGANISMOS FITOPATOGêNICOS EM PLANTAçõES". A invenção está relacionada a novos derivados de N-fenil-4-(4-piridil)-2-pirimidinoamina com a fórmula (I) onde a soma de (m+p) juntos é 0, 1, 2 ou 3; n e q são independentemente um do outro 0 ou 1, e a soma de (m+p+q) juntos é 1, 2, 3 ou 4; R~ 1~ é hidrogênio, halogênio, alcóxi, haloalquila, haloalcóxi ou alquila; R~ 2~ é hidrogênio, C~ 1~-C~ 6~ alquila, C~ 1~-C~ 6~ haloalquila ou C~ 1~-C~ 6~ alcóxi; R~ 2A~ é hidrogênio, C~ 1~-C~ 6~ alquila, C~ 3~-C~ 4~ alquenila ou C~ 3~-C~ 4~ alquinila; cada um de R~ 3~, R~ 4~, R~ 5~ e R~ 6~ é, independentemente dos outros, hidrogênio, C~ 1~-C~ 6~ alquila, C~ 1~-C~ 6~ haloalquila, hidróxi-C~ 1~-C~ 6~ alquila ou C~ 1~-C~ 6~-alcóxi-C~ 1~-C~ 6~-alquila, ou os membros do anel CR~ 3~R~ 4~ ou CR~ 5~R~ 6~ ou CR~ 2~R~ 2A~ são independentemente dos outros um grupo carbonila (C=O) ou um grupo C=S; X é C=O, C=S, S=O ou O=S=O; Y é O, S, C=O, CH~ 2~, -N(R~ 8~)-, -O-N(R~ 8~)-, -N(R~ 8~)-O- ou -NH-; R~ 7~ é hidrogênio, C~ 1~-C~ 4~ alquila, C~ 3~-C~ 4~ alquenila, C~ 3~-C~ 4~ alquinila, -CH~ 2~OR~ 8~, CH~ 2~SR~ 8~, -C(O)R~ 8~, -C(O)OR~ 8~, SO~ 2~R~ 8~, SOR8 ou SR~ 8~; e R~ 8~ é C~ 1~-C~ 8~ alquila, C~ 1~-C~ 8~ alcoxialquila, C~ 1~-C~ 8~ haloalquila ou fenil-C~ 1~-C~ 2~ alquila, onde a fenila pode ser substituído por até três grupos selecionados de halo ou C~ 1~-C~ 4~ alquila; ou um sal do mesmo. A invenção está relacionada também à preparação dos compostos e a composições agroquímicas que compreendem pelo menos um desses compostos como o ingrediente ativo, bem como à preparação das ditas composições e ao uso dos compostos ou das composições para o controle ou a prevenção da infestação em plantas por microrganismos fitopatogênicos, em especial os fungos.
BRPI0116657-3A 2001-01-03 2001-12-20 composto, processo para a preparaÇço do mesmo, composiÇço para controlar e proteger contra microrganismos fitopatogÊnicos, uso de um composto, e, mÉtodo para controlar e evitar a infestaÇço por microrganismos fitopatogÊnicos em plantaÇÕes. BR0116657B1 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0100102.3A GB0100102D0 (en) 2001-01-03 2001-01-03 Organic compounds
PCT/IB2001/002821 WO2002053560A1 (en) 2001-01-03 2001-12-20 Microbiocidal n-phenyl-n-[4-(4-pyridyl-2-pyrimidin-2-yl]-amine derivatives

Publications (2)

Publication Number Publication Date
BR0116657A true BR0116657A (pt) 2004-01-06
BR0116657B1 BR0116657B1 (pt) 2012-08-07

Family

ID=9906185

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0116657-3A BR0116657B1 (pt) 2001-01-03 2001-12-20 composto, processo para a preparaÇço do mesmo, composiÇço para controlar e proteger contra microrganismos fitopatogÊnicos, uso de um composto, e, mÉtodo para controlar e evitar a infestaÇço por microrganismos fitopatogÊnicos em plantaÇÕes.

Country Status (17)

Country Link
US (1) US7074787B2 (pt)
EP (1) EP1349849B1 (pt)
JP (1) JP4274795B2 (pt)
KR (1) KR100838796B1 (pt)
CN (1) CN100374434C (pt)
AT (1) ATE276243T1 (pt)
AU (1) AU2002236101B2 (pt)
BR (1) BR0116657B1 (pt)
CA (1) CA2428604C (pt)
DE (1) DE60105646T2 (pt)
ES (1) ES2223938T3 (pt)
GB (1) GB0100102D0 (pt)
IL (2) IL155939A0 (pt)
MX (1) MXPA03006000A (pt)
PL (1) PL204272B1 (pt)
WO (1) WO2002053560A1 (pt)
ZA (1) ZA200303743B (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0129391D0 (en) * 2001-12-07 2002-01-30 Syngenta Participations Ag Microbiocidal n-phenyl-n-[4-(4-pyridyl)-2-pyrimidin-2-yl]-amine derivatives
MXPA04012577A (es) 2002-07-31 2005-03-23 Ciba Sc Holding Ag Derivados de piridin-triacina como sustancias microbicidas activas.
BRPI0408332A (pt) 2003-03-14 2006-03-21 Ono Pharmaceutical Co derivados heterocìclicos contendo nitrogênio e medicamentos contendo os mesmos como ingrediente ativo
GB0307268D0 (en) * 2003-03-28 2003-05-07 Syngenta Ltd Organic compounds
GB0307269D0 (en) * 2003-03-28 2003-05-07 Syngenta Ltd Fungicidal compositions
EP2492264A3 (en) * 2003-06-03 2012-12-19 Rib-X Pharmaceuticals, Inc. Biaryl Heterocyclic Compounds And Methods Of Making And Using The Same
US8324398B2 (en) 2003-06-03 2012-12-04 Rib-X Pharmaceuticals, Inc. Process for the synthesis of biaryl oxazolidinones
CN101775013A (zh) * 2004-09-13 2010-07-14 小野药品工业株式会社 含氮杂环衍生物及含有其作为活性成分的药物
WO2006133397A2 (en) 2005-06-08 2006-12-14 Rib-X Pharmaceuticals, Inc. Process for the synthesis of triazoles
WO2007105637A1 (ja) 2006-03-10 2007-09-20 Ono Pharmaceutical Co., Ltd. 含窒素複素環誘導体およびそれらを有効成分とする薬剤
CL2008001460A1 (es) * 2007-05-16 2008-11-21 Bayer Cropscience Sa Compuestos derivados de fenil-pirimidin-amino; compuestos intermediarios; composicion fungicida que comprende a dichos compuestos; y metodo para controlar hongos fitopatogenos de cultivos agricolas.
AU2013206248B2 (en) * 2008-06-27 2016-06-23 Xenon Pharmaceuticals Inc. Organic compounds
CA2738787A1 (en) * 2008-11-13 2010-05-20 Bayer Cropscience Ag Substituted (pyridyl)-azinylamine derivatives as fungicides
EP3442961B1 (en) * 2016-04-13 2021-03-24 Redag Crop Protection Ltd Agricultural chemicals
WO2018019574A1 (en) * 2016-07-28 2018-02-01 Basf Se Herbicidal pyrimidine compounds

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0388838B1 (de) * 1989-03-22 1996-01-10 Ciba-Geigy Ag Schädlingsbekämpfungsmittel
DE4034762A1 (de) * 1990-11-02 1992-05-07 Hoechst Ag Pyridylpyrimidine, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als fungizide
DE69429078T2 (de) * 1993-10-01 2002-07-11 Novartis Ag Pharmacologisch wirksame pyridinderivate und verfahren zu deren herstellung
JP3588116B2 (ja) * 1993-10-01 2004-11-10 ノバルティス アクチェンゲゼルシャフト 薬理活性のピリミジンアミン誘導体およびその製造方法
GB9622363D0 (en) * 1996-10-28 1997-01-08 Celltech Therapeutics Ltd Chemical compounds
GB0014022D0 (en) 2000-06-08 2000-08-02 Novartis Ag Organic compounds

Also Published As

Publication number Publication date
GB0100102D0 (en) 2001-02-14
IL155939A (en) 2008-07-08
WO2002053560A1 (en) 2002-07-11
JP2004517122A (ja) 2004-06-10
CN100374434C (zh) 2008-03-12
DE60105646T2 (de) 2005-11-17
ATE276243T1 (de) 2004-10-15
DE60105646D1 (de) 2004-10-21
MXPA03006000A (es) 2005-02-14
EP1349849B1 (en) 2004-09-15
KR100838796B1 (ko) 2008-06-17
IL155939A0 (en) 2003-12-23
EP1349849A1 (en) 2003-10-08
PL362143A1 (en) 2004-10-18
US20040063937A1 (en) 2004-04-01
ES2223938T3 (es) 2005-03-01
PL204272B1 (pl) 2009-12-31
ZA200303743B (en) 2004-03-31
CA2428604A1 (en) 2002-07-11
BR0116657B1 (pt) 2012-08-07
US7074787B2 (en) 2006-07-11
KR20030066676A (ko) 2003-08-09
CA2428604C (en) 2009-05-12
CN1484641A (zh) 2004-03-24
AU2002236101B2 (en) 2006-09-14
JP4274795B2 (ja) 2009-06-10

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 07/08/2012, OBSERVADAS AS CONDICOES LEGAIS.

B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE A 13A ANUIDADE.

B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)

Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2285 DE 21-10-2014 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.