BR0115809A - Processo de ciclização para sìntese de compostos derivados de pirolidina - Google Patents
Processo de ciclização para sìntese de compostos derivados de pirolidinaInfo
- Publication number
- BR0115809A BR0115809A BR0115809-0A BR0115809A BR0115809A BR 0115809 A BR0115809 A BR 0115809A BR 0115809 A BR0115809 A BR 0115809A BR 0115809 A BR0115809 A BR 0115809A
- Authority
- BR
- Brazil
- Prior art keywords
- synthesis
- cyclization process
- pyrolidine
- derivatives
- pyrolidine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/12—Oxygen or sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pyrrole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
"PROCESSO DE CICLIZAçãO PARA SìNTESE DE COMPOSTOS DERIVADOS DE PIROLIDINA". A presente invenção diz respeito a um processo de preparação de derivados de pirolidina o qual consiste numa reação de ciclização do composto de fórmula (1) na presença de um catalisador, uma amina primária ou uma base.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0015626A FR2817550B1 (fr) | 2000-12-01 | 2000-12-01 | Procede de preparation de derives de pyrrolidine substituee |
PCT/FR2001/003796 WO2002044146A1 (fr) | 2000-12-01 | 2001-11-30 | Procede de cyclisation pour la synthese de composes derives de pyrrolidine |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0115809A true BR0115809A (pt) | 2003-09-16 |
Family
ID=8857165
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0115809-0A BR0115809A (pt) | 2000-12-01 | 2001-11-30 | Processo de ciclização para sìntese de compostos derivados de pirolidina |
Country Status (9)
Country | Link |
---|---|
US (1) | US6861535B2 (pt) |
EP (1) | EP1347956A1 (pt) |
JP (1) | JP2004514710A (pt) |
AU (1) | AU2002222087A1 (pt) |
BR (1) | BR0115809A (pt) |
CA (1) | CA2430302A1 (pt) |
FR (1) | FR2817550B1 (pt) |
IL (1) | IL156078A0 (pt) |
WO (1) | WO2002044146A1 (pt) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7968734B2 (en) * | 2004-07-01 | 2011-06-28 | Stc.Unm | Organocatalysts and methods of use in chemical synthesis |
KR101072479B1 (ko) | 2008-12-01 | 2011-10-11 | 엔자이텍 주식회사 | 라세믹 또는 광학적으로 활성이 있는 3―하이드록시피롤리딘 및 그의 유도체의 제조방법 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS60104061A (ja) * | 1983-11-08 | 1985-06-08 | Sankyo Co Ltd | ピロリジン誘導体の製法 |
JPH0776209B2 (ja) * | 1990-04-11 | 1995-08-16 | 高砂香料工業株式会社 | 光学活性3―ヒドロキシピロリジン誘導体の製造方法 |
US5977381A (en) * | 1998-01-12 | 1999-11-02 | Hoffmann-La Roche Inc. | Process for making 3-amino-pyrolidine derivatives |
-
2000
- 2000-12-01 FR FR0015626A patent/FR2817550B1/fr not_active Expired - Fee Related
-
2001
- 2001-11-30 BR BR0115809-0A patent/BR0115809A/pt not_active IP Right Cessation
- 2001-11-30 JP JP2002546516A patent/JP2004514710A/ja active Pending
- 2001-11-30 CA CA002430302A patent/CA2430302A1/fr not_active Abandoned
- 2001-11-30 AU AU2002222087A patent/AU2002222087A1/en not_active Abandoned
- 2001-11-30 IL IL15607801A patent/IL156078A0/xx unknown
- 2001-11-30 EP EP01998536A patent/EP1347956A1/fr not_active Withdrawn
- 2001-11-30 WO PCT/FR2001/003796 patent/WO2002044146A1/fr active Application Filing
-
2003
- 2003-05-30 US US10/449,377 patent/US6861535B2/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
US20040034235A1 (en) | 2004-02-19 |
CA2430302A1 (fr) | 2002-06-06 |
IL156078A0 (en) | 2003-12-23 |
EP1347956A1 (fr) | 2003-10-01 |
US6861535B2 (en) | 2005-03-01 |
AU2002222087A1 (en) | 2002-06-11 |
WO2002044146A1 (fr) | 2002-06-06 |
JP2004514710A (ja) | 2004-05-20 |
FR2817550B1 (fr) | 2005-04-29 |
FR2817550A1 (fr) | 2002-06-07 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 6A , 7A E 8A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 DA RPI 2021 DE 29/09/2009. |