BG20799A3 - Метод за получаване на бензодиазепинови производни - Google Patents

Метод за получаване на бензодиазепинови производни

Info

Publication number
BG20799A3
BG20799A3 BG018690A BG1869071A BG20799A3 BG 20799 A3 BG20799 A3 BG 20799A3 BG 018690 A BG018690 A BG 018690A BG 1869071 A BG1869071 A BG 1869071A BG 20799 A3 BG20799 A3 BG 20799A3
Authority
BG
Bulgaria
Prior art keywords
obtaining
benzodiazepine derivatives
benzodiazepine
derivatives
obtaining benzodiazepine
Prior art date
Application number
BG018690A
Other languages
Bulgarian (bg)
English (en)
Inventor
Roland Jannin
Josepf Hellerbach
Original Assignee
F. Hoffmann - La Roche Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F. Hoffmann - La Roche Ag filed Critical F. Hoffmann - La Roche Ag
Publication of BG20799A3 publication Critical patent/BG20799A3/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
BG018690A 1970-10-07 1971-10-05 Метод за получаване на бензодиазепинови производни BG20799A3 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH1490570A CH538492A (de) 1970-10-07 1970-10-07 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Publications (1)

Publication Number Publication Date
BG20799A3 true BG20799A3 (bg) 1975-12-20

Family

ID=4404720

Family Applications (6)

Application Number Title Priority Date Filing Date
BG020775A BG21030A3 (bg) 1970-10-07 1971-10-05 Метод за получаване на бензодиазепинови производни
BG018690A BG20799A3 (bg) 1970-10-07 1971-10-05 Метод за получаване на бензодиазепинови производни
BG020778A BG20111A3 (bg) 1970-10-07 1971-10-05 Метод за получаване на бензодиазепинови производни
BG020774A BG20597A3 (bg) 1970-10-07 1971-10-05 Метод за получаване на бензодиазепинови производни
BG020776A BG20598A3 (bg) 1970-10-07 1971-10-05 Метод за получаване на бензодиазепинови производни
BG20777A BG19599A3 (pt) 1970-10-07 1971-10-05

Family Applications Before (1)

Application Number Title Priority Date Filing Date
BG020775A BG21030A3 (bg) 1970-10-07 1971-10-05 Метод за получаване на бензодиазепинови производни

Family Applications After (4)

Application Number Title Priority Date Filing Date
BG020778A BG20111A3 (bg) 1970-10-07 1971-10-05 Метод за получаване на бензодиазепинови производни
BG020774A BG20597A3 (bg) 1970-10-07 1971-10-05 Метод за получаване на бензодиазепинови производни
BG020776A BG20598A3 (bg) 1970-10-07 1971-10-05 Метод за получаване на бензодиазепинови производни
BG20777A BG19599A3 (pt) 1970-10-07 1971-10-05

Country Status (26)

Country Link
US (1) US3757008A (pt)
JP (1) JPS5614667B1 (pt)
AT (6) AT317900B (pt)
AU (1) AU456526B2 (pt)
BE (1) BE773547A (pt)
BG (6) BG21030A3 (pt)
BR (1) BR7106395D0 (pt)
CA (1) CA972754A (pt)
CH (1) CH538492A (pt)
CS (1) CS174165B2 (pt)
DE (1) DE2150075A1 (pt)
DK (1) DK138797B (pt)
ES (1) ES395762A1 (pt)
FR (1) FR2110275B1 (pt)
GB (2) GB1357547A (pt)
HU (1) HU164060B (pt)
IE (1) IE35685B1 (pt)
IL (1) IL37645A (pt)
MY (1) MY7500047A (pt)
NL (1) NL7113023A (pt)
PH (1) PH10182A (pt)
PL (1) PL82734B1 (pt)
RO (1) RO71264A (pt)
SE (2) SE388611B (pt)
SU (1) SU520917A3 (pt)
ZA (1) ZA715787B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT314541B (de) * 1970-10-19 1974-04-10 Sumitomo Chemical Co Verfahren zur Herstellung von neuen Benzodiazepinen und ihren Salzen
HU171033B (hu) * 1974-05-29 1977-10-28 Richter Gedeon Vegyeszet Sposob poluchenija proizvodnykh benzodiazepina
ES2084577T3 (es) * 1986-10-24 1996-05-16 Abbott Lab Ensayo, trazadores, inmunogenos y anticuerpos para benzodiazepinas.
FR2630109B1 (fr) * 1988-04-19 1991-11-29 Synthelabo Derives de ((n-(amino-2 oxo-2 ethyl)methylamino)-2 ethyl)-5 hydroxy-3 (methoxy-4 phenyl)-2 dihydro-2,3 5h-benzothiazepine-1,5 one-4, leur preparation et leur application en therapeutique
FR2653122B1 (fr) * 1989-10-17 1994-04-15 Synthelabo Derives de 5-[2-[[2-amino-2-oxoethyl]methylamino]ethyl]-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-1,5(5h)-benzothiazepine-4-one, leur preparation et leur application en therapeutique.
US5302715A (en) * 1992-04-06 1994-04-12 Biosite Diagnostics, Inc. Benzodiazepine derivatives
HU227319B1 (en) * 2005-12-08 2011-03-28 Egis Gyogyszergyar Nyrt Process for the production of (2-chloro-ethoxy)-acetic acid-n,n-dimethylamide and its intermediate and the novel intermediate

Also Published As

Publication number Publication date
AT315180B (de) 1974-05-10
PL82734B1 (pt) 1975-10-31
CA972754A (en) 1975-08-12
BG20111A3 (bg) 1975-10-30
IE35685B1 (en) 1976-04-28
GB1357548A (en) 1974-06-26
HU164060B (pt) 1973-12-28
DK138797B (da) 1978-10-30
FR2110275B1 (pt) 1974-11-15
SE7513089L (sv) 1975-11-20
BG21030A3 (bg) 1976-01-20
AT317901B (de) 1974-09-25
JPS5614667B1 (pt) 1981-04-06
BG20597A3 (bg) 1975-12-05
FR2110275A1 (pt) 1972-06-02
BG20598A3 (bg) 1975-12-05
CH538492A (de) 1973-06-30
CS174165B2 (pt) 1977-03-31
BG19599A3 (pt) 1975-06-25
SU520917A3 (ru) 1976-07-05
PH10182A (en) 1976-09-23
IL37645A (en) 1974-11-29
ZA715787B (en) 1972-05-31
AU3296671A (en) 1973-03-08
US3757008A (en) 1973-09-04
GB1357547A (en) 1974-06-26
ES395762A1 (es) 1974-10-16
NL7113023A (pt) 1972-04-11
IE35685L (en) 1972-04-07
DK138797C (pt) 1979-04-09
AT317900B (de) 1974-09-25
BE773547A (fr) 1972-04-06
MY7500047A (en) 1975-12-31
IL37645A0 (en) 1971-11-29
RO71264A (ro) 1980-07-15
SE388611B (sv) 1976-10-11
AT315859B (de) 1974-06-10
AU456526B2 (en) 1974-12-19
AT317902B (de) 1974-09-25
BR7106395D0 (pt) 1973-04-12
AT315860B (de) 1974-06-10
DE2150075A1 (de) 1972-04-13

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