BE901336A - NOVEL PYRAZOLO [1,5-A] PYRIDINE DERIVATIVES, THEIR PREPARATION AND THE THERAPEUTIC COMPOSITIONS CONTAINING THEM. - Google Patents
NOVEL PYRAZOLO [1,5-A] PYRIDINE DERIVATIVES, THEIR PREPARATION AND THE THERAPEUTIC COMPOSITIONS CONTAINING THEM.Info
- Publication number
- BE901336A BE901336A BE0/214208A BE214208A BE901336A BE 901336 A BE901336 A BE 901336A BE 0/214208 A BE0/214208 A BE 0/214208A BE 214208 A BE214208 A BE 214208A BE 901336 A BE901336 A BE 901336A
- Authority
- BE
- Belgium
- Prior art keywords
- aryl
- preparation
- compositions containing
- therapeutic compositions
- pyridine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Pharmacology & Pharmacy (AREA)
- Rheumatology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Nouveaux dérivés de formule I dans laquelle R1 = COOH, alcoyloxycarbonyle, CONH2, alcoylcarbamoyle ou dialcoylcarbamoyle, R2= halogène, alcoyle, CN, alcoyloxycarbonyle, COOH, CONH2, alcoylcarbamoyle, dialcoylcarbamoyle, NO2, OH, alcoyloxy, aryloxy, aralcoyle, CF3, alcoylthio, alcoylsulfinyle, alcoylsulfonyle, arylthio, arylsulfinyle, arylsulfonyle, alcanoyle, aroyle ou aryle, ou un radical amino qui peut etre substitué et n = 1, 2, 3 ou 4, sauf restrictions particulières. Les produits permettent d'envisager une utilisation dans le traitement des maladies arthritiques.New derivatives of formula I in which R1 = COOH, alkyloxycarbonyl, CONH2, alkylcarbamoyl or dialcoylcarbamoyl, R2 = halogen, alkyl, CN, alkyloxycarbonyl, COOH, CONH2, alkylcarbamoyl, CFloyl, arylcoyl, aryl, arylalkyl, NO2, aralkyl, aryloyl, aryl, aryl, aryl, NO2, alkyl , alkylsulfinyl, alkylsulfonyl, arylthio, arylsulfinyl, arylsulfonyl, alkanoyl, aroyl or aryl, or an amino radical which can be substituted and n = 1, 2, 3 or 4, unless there are special restrictions. The products make it possible to envisage a use in the treatment of arthritic diseases.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB838334001A GB8334001D0 (en) | 1983-12-21 | 1983-12-21 | Compositions of matter |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE901336A true BE901336A (en) | 1985-06-20 |
Family
ID=10553616
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE0/214208A BE901336A (en) | 1983-12-21 | 1984-12-20 | NOVEL PYRAZOLO [1,5-A] PYRIDINE DERIVATIVES, THEIR PREPARATION AND THE THERAPEUTIC COMPOSITIONS CONTAINING THEM. |
Country Status (18)
| Country | Link |
|---|---|
| JP (1) | JPS60172979A (en) |
| KR (1) | KR850004758A (en) |
| AT (1) | ATA404684A (en) |
| AU (1) | AU3690684A (en) |
| BE (1) | BE901336A (en) |
| DE (1) | DE3447730A1 (en) |
| DK (1) | DK616784A (en) |
| ES (2) | ES8605516A1 (en) |
| FI (1) | FI845022L (en) |
| FR (1) | FR2556723A1 (en) |
| GB (2) | GB8334001D0 (en) |
| GR (1) | GR82507B (en) |
| IL (1) | IL73860A0 (en) |
| IT (1) | IT1178768B (en) |
| LU (1) | LU85690A1 (en) |
| NL (1) | NL8403874A (en) |
| SE (1) | SE8406478L (en) |
| ZA (1) | ZA849903B (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20070155738A1 (en) | 2005-05-20 | 2007-07-05 | Alantos Pharmaceuticals, Inc. | Heterobicyclic metalloprotease inhibitors |
| AU2008273050A1 (en) * | 2007-07-11 | 2009-01-15 | Auckland Uniservices Limited | Pyrazolo[1,5-a]pyridines and their use in cancer therapy |
| JP6816287B2 (en) * | 2016-09-07 | 2021-01-20 | シャンハイ ハイヘ ファーマシューティカル カンパニー リミテッドＳｈａｎｇｈａｉ Ｈａｉｈｅ Ｐｈａｒｍａｃｅｕｔｉｃａｌ Ｃｏ．， Ｌｔｄ | Pyridine and 5-membered aromatic ring compounds, their production methods and uses |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5154583A (en) * | 1974-11-01 | 1976-05-13 | Kyorin Seiyaku Kk | Shinkipirazoro * 1 55a * pirijinjudotaino seizoho |
| JPS5610114A (en) * | 1979-07-05 | 1981-02-02 | Grelan Pharmaceut Co Ltd | Novel analgesic and anti-inflammatory agent |
| GB2121799B (en) * | 1982-06-16 | 1985-07-10 | May & Baker Ltd | New pyrazolopyridine derivative |
-
1983
- 1983-12-21 GB GB838334001A patent/GB8334001D0/en active Pending
-
1984
- 1984-12-18 LU LU85690A patent/LU85690A1/en unknown
- 1984-12-19 KR KR1019840008098A patent/KR850004758A/en not_active Application Discontinuation
- 1984-12-19 JP JP59268203A patent/JPS60172979A/en active Pending
- 1984-12-19 AU AU36906/84A patent/AU3690684A/en not_active Abandoned
- 1984-12-19 IL IL73860A patent/IL73860A0/en unknown
- 1984-12-19 ZA ZA849903A patent/ZA849903B/en unknown
- 1984-12-19 GR GR82507A patent/GR82507B/en unknown
- 1984-12-19 GB GB08431986A patent/GB2153818B/en not_active Expired
- 1984-12-19 FI FI845022A patent/FI845022L/en not_active Application Discontinuation
- 1984-12-19 SE SE8406478A patent/SE8406478L/en not_active Application Discontinuation
- 1984-12-20 AT AT0404684A patent/ATA404684A/en not_active IP Right Cessation
- 1984-12-20 NL NL8403874A patent/NL8403874A/en not_active Application Discontinuation
- 1984-12-20 BE BE0/214208A patent/BE901336A/en not_active IP Right Cessation
- 1984-12-20 DK DK616784A patent/DK616784A/en not_active Application Discontinuation
- 1984-12-20 FR FR8419522A patent/FR2556723A1/en not_active Withdrawn
- 1984-12-21 ES ES538957A patent/ES8605516A1/en not_active Expired
- 1984-12-21 DE DE19843447730 patent/DE3447730A1/en not_active Withdrawn
- 1984-12-21 IT IT24176/84A patent/IT1178768B/en active
-
1985
- 1985-04-22 ES ES542457A patent/ES8603426A1/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| ES538957A0 (en) | 1986-03-16 |
| SE8406478D0 (en) | 1984-12-19 |
| DE3447730A1 (en) | 1985-07-04 |
| GR82507B (en) | 1985-04-22 |
| IT8424176A0 (en) | 1984-12-21 |
| SE8406478L (en) | 1985-06-22 |
| GB8431986D0 (en) | 1985-01-30 |
| LU85690A1 (en) | 1986-07-17 |
| AU3690684A (en) | 1985-07-04 |
| JPS60172979A (en) | 1985-09-06 |
| NL8403874A (en) | 1985-07-16 |
| ES542457A0 (en) | 1985-12-16 |
| FR2556723A1 (en) | 1985-06-21 |
| ES8603426A1 (en) | 1985-12-16 |
| ZA849903B (en) | 1985-08-28 |
| DK616784A (en) | 1985-06-22 |
| IT1178768B (en) | 1987-09-16 |
| FI845022A0 (en) | 1984-12-19 |
| DK616784D0 (en) | 1984-12-20 |
| FI845022L (en) | 1985-06-22 |
| ES8605516A1 (en) | 1986-03-16 |
| KR850004758A (en) | 1985-07-27 |
| IL73860A0 (en) | 1985-03-31 |
| ATA404684A (en) | 1987-08-15 |
| GB2153818B (en) | 1987-07-29 |
| GB8334001D0 (en) | 1984-02-01 |
| GB2153818A (en) | 1985-08-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RE | Patent lapsed |
Owner name: MAY & BAKER LTD Effective date: 19871231 |