BE899399A - Derives d'acide quinolone-carboxylique. - Google Patents
Derives d'acide quinolone-carboxylique. Download PDFInfo
- Publication number
- BE899399A BE899399A BE0/212743A BE212743A BE899399A BE 899399 A BE899399 A BE 899399A BE 0/212743 A BE0/212743 A BE 0/212743A BE 212743 A BE212743 A BE 212743A BE 899399 A BE899399 A BE 899399A
- Authority
- BE
- Belgium
- Prior art keywords
- emi
- formula
- acid
- carboxylic acid
- methyl
- Prior art date
Links
- XOQQVKDBGLYPGH-UHFFFAOYSA-N 2-oxo-1h-quinoline-3-carboxylic acid Chemical class C1=CC=C2NC(=O)C(C(=O)O)=CC2=C1 XOQQVKDBGLYPGH-UHFFFAOYSA-N 0.000 title 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical group FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 229910052801 chlorine Inorganic materials 0.000 abstract 1
- 239000000460 chlorine Substances 0.000 abstract 1
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 1
- 229910052731 fluorine Inorganic materials 0.000 abstract 1
- 239000011737 fluorine Chemical group 0.000 abstract 1
- 150000004677 hydrates Chemical class 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- -1 p-aminobenzyl Chemical group 0.000 abstract 1
- LOAUVZALPPNFOQ-UHFFFAOYSA-N quinaldic acid Chemical class C1=CC=CC2=NC(C(=O)O)=CC=C21 LOAUVZALPPNFOQ-UHFFFAOYSA-N 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- G—PHYSICS
- G03—PHOTOGRAPHY; CINEMATOGRAPHY; ANALOGOUS TECHNIQUES USING WAVES OTHER THAN OPTICAL WAVES; ELECTROGRAPHY; HOLOGRAPHY
- G03C—PHOTOSENSITIVE MATERIALS FOR PHOTOGRAPHIC PURPOSES; PHOTOGRAPHIC PROCESSES, e.g. CINE, X-RAY, COLOUR, STEREO-PHOTOGRAPHIC PROCESSES; AUXILIARY PROCESSES IN PHOTOGRAPHY
- G03C1/00—Photosensitive materials
- G03C1/005—Silver halide emulsions; Preparation thereof; Physical treatment thereof; Incorporation of additives therein
- G03C1/06—Silver halide emulsions; Preparation thereof; Physical treatment thereof; Incorporation of additives therein with non-macromolecular additives
- G03C1/34—Fog-inhibitors; Stabilisers; Agents inhibiting latent image regression
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Physics & Mathematics (AREA)
- Spectroscopy & Molecular Physics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Materials Engineering (AREA)
- General Physics & Mathematics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP23257083A JPS60123837A (ja) | 1983-12-09 | 1983-12-09 | ハロゲン化銀写真乳剤 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE899399A true BE899399A (fr) | 1984-07-31 |
Family
ID=16941409
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE0/212743A BE899399A (fr) | 1983-12-09 | 1984-04-12 | Derives d'acide quinolone-carboxylique. |
Country Status (2)
Country | Link |
---|---|
JP (1) | JPS60123837A (enrdf_load_stackoverflow) |
BE (1) | BE899399A (enrdf_load_stackoverflow) |
Cited By (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0167763A1 (de) * | 1984-06-04 | 1986-01-15 | Bayer Ag | 7-Amino-1-cyclopropyl-6,8-dihalogen-1,4-dihydro-4-oxo-3-chinolincarbonsäuren, Verfahren zur ihrer Herstellung sowie diese enthaltende antibakterielle Mittel |
EP0178388A1 (en) * | 1984-10-11 | 1986-04-23 | Kyorin Pharmaceutical Co., Ltd. | Quinolinecarboxylic acid derivatives |
EP0195316A1 (en) * | 1985-03-08 | 1986-09-24 | Kyorin Pharmaceutical Co., Ltd. | Quinolonecarboxylic acid derivatives |
EP0195841A1 (en) * | 1985-03-08 | 1986-10-01 | Kyorin Pharmaceutical Co., Ltd. | Quinolinecarboxylic acid derivatives and process for their preparation |
EP0198678A3 (en) * | 1985-04-15 | 1987-03-25 | Warner-Lambert Company | A process for preparing substituted quinoline-3-carboxylic acids |
US4668680A (en) * | 1985-12-12 | 1987-05-26 | Warner-Lambert Company | 5-amino-6,8-difluoroquinolones as antibacterial agents |
US4689423A (en) * | 1986-04-01 | 1987-08-25 | Warner-Lambert Company | Process for the preparation of 2,3,4,5-tetrafluorobenzoyl acetates |
US4772706A (en) * | 1986-01-13 | 1988-09-20 | Warner-Lambert Company | Process for quinoline-3-carboxylic acid antibacterial agents |
US4874764A (en) * | 1986-02-25 | 1989-10-17 | Otsuka Pharmaceutical Company, Limited | Benzoheterocyclic compounds |
EP0287951A3 (en) * | 1987-04-16 | 1990-06-13 | Otsuka Pharmaceutical Co., Ltd. | Benzoheterocyclic compounds |
US5290934A (en) * | 1987-04-16 | 1994-03-01 | Otsuka Pharmaceutical Company, Limited | Benzoheterocyclic compounds |
WO1995021603A1 (de) * | 1994-02-10 | 1995-08-17 | Henkel Kommanditgesellschaft Auf Aktien | 2-fluor-6-nitroaniline |
US5468861A (en) * | 1984-06-04 | 1995-11-21 | Bayer Aktiengesellschaft | 8-chloro-1-cyclopropyl-6,7-difluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid and alkyl esters thereof |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS63220130A (ja) * | 1987-03-09 | 1988-09-13 | Mitsubishi Paper Mills Ltd | ハロゲン化銀写真乳剤 |
-
1983
- 1983-12-09 JP JP23257083A patent/JPS60123837A/ja active Granted
-
1984
- 1984-04-12 BE BE0/212743A patent/BE899399A/fr not_active IP Right Cessation
Cited By (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0167763A1 (de) * | 1984-06-04 | 1986-01-15 | Bayer Ag | 7-Amino-1-cyclopropyl-6,8-dihalogen-1,4-dihydro-4-oxo-3-chinolincarbonsäuren, Verfahren zur ihrer Herstellung sowie diese enthaltende antibakterielle Mittel |
US5571812A (en) * | 1984-06-04 | 1996-11-05 | Bayer Aktiengesellschaft | 7-amino-1-cyclopropyl-6,8-dihalogeno-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid antibacterial agents |
US5969141A (en) * | 1984-06-04 | 1999-10-19 | Bayer Aktiengesellschaft | Intermediates for 7-amino-1-cyclopropyl-6,8-dihalogeno-1,4-dihydro-4-oxo-3-quinolinecarbox ylic acid antibacterial agents |
US5468861A (en) * | 1984-06-04 | 1995-11-21 | Bayer Aktiengesellschaft | 8-chloro-1-cyclopropyl-6,7-difluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid and alkyl esters thereof |
EP0178388A1 (en) * | 1984-10-11 | 1986-04-23 | Kyorin Pharmaceutical Co., Ltd. | Quinolinecarboxylic acid derivatives |
EP0195316A1 (en) * | 1985-03-08 | 1986-09-24 | Kyorin Pharmaceutical Co., Ltd. | Quinolonecarboxylic acid derivatives |
EP0195841A1 (en) * | 1985-03-08 | 1986-10-01 | Kyorin Pharmaceutical Co., Ltd. | Quinolinecarboxylic acid derivatives and process for their preparation |
EP0198678A3 (en) * | 1985-04-15 | 1987-03-25 | Warner-Lambert Company | A process for preparing substituted quinoline-3-carboxylic acids |
US4668680A (en) * | 1985-12-12 | 1987-05-26 | Warner-Lambert Company | 5-amino-6,8-difluoroquinolones as antibacterial agents |
US4772706A (en) * | 1986-01-13 | 1988-09-20 | Warner-Lambert Company | Process for quinoline-3-carboxylic acid antibacterial agents |
US4880806A (en) * | 1986-02-25 | 1989-11-14 | Otsuka Pharmaceutical Company, Limited | 1-Cyclopropyl-6-fluoro-7-piperazinyl-1,4-Dihydro-4-oxo-quinoline-3-carboxylic acid derivatives |
US4874764A (en) * | 1986-02-25 | 1989-10-17 | Otsuka Pharmaceutical Company, Limited | Benzoheterocyclic compounds |
US4689423A (en) * | 1986-04-01 | 1987-08-25 | Warner-Lambert Company | Process for the preparation of 2,3,4,5-tetrafluorobenzoyl acetates |
EP0287951A3 (en) * | 1987-04-16 | 1990-06-13 | Otsuka Pharmaceutical Co., Ltd. | Benzoheterocyclic compounds |
US5563138A (en) * | 1987-04-16 | 1996-10-08 | Otsuka Pharmaceutical Company, Limited | Benzoheterocyclic compounds |
EP0565132A3 (en) * | 1987-04-16 | 1994-05-18 | Otsuka Pharma Co Ltd | Benzoheterocyclic compounds |
US5591744A (en) * | 1987-04-16 | 1997-01-07 | Otsuka Pharmaceutical Company, Limited | Benzoheterocyclic compounds |
US5723648A (en) * | 1987-04-16 | 1998-03-03 | Otsuka Pharmaceutical Company, Limited | Intermediates for anti-microbial benzoheterocyclic compounds |
US5811576A (en) * | 1987-04-16 | 1998-09-22 | Otsuka Pharmaceutical Company, Limited | Intermediates for anti-microbial quinolone carboxylic acids |
US5290934A (en) * | 1987-04-16 | 1994-03-01 | Otsuka Pharmaceutical Company, Limited | Benzoheterocyclic compounds |
WO1995021603A1 (de) * | 1994-02-10 | 1995-08-17 | Henkel Kommanditgesellschaft Auf Aktien | 2-fluor-6-nitroaniline |
Also Published As
Publication number | Publication date |
---|---|
JPS60123837A (ja) | 1985-07-02 |
JPH0222934B2 (enrdf_load_stackoverflow) | 1990-05-22 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE20 | Patent expired |
Owner name: *KYORIN PHARMACEUTICAL CO. LTD Effective date: 20040412 |