BE898943A - Composes pour le traitement des psychoses et leur utilisation - Google Patents

Composes pour le traitement des psychoses et leur utilisation

Info

Publication number
BE898943A
BE898943A BE0/212415A BE212415A BE898943A BE 898943 A BE898943 A BE 898943A BE 0/212415 A BE0/212415 A BE 0/212415A BE 212415 A BE212415 A BE 212415A BE 898943 A BE898943 A BE 898943A
Authority
BE
Belgium
Prior art keywords
treatment
psychoses
compounds
triazolobenzodiazepines
schizophrenics
Prior art date
Application number
BE0/212415A
Other languages
English (en)
Inventor
R Lahti
R Pyka
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of BE898943A publication Critical patent/BE898943A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Abstract

Certaines amino-triazolobenzodiazépines, telles que, par exemple, l'adinazolam (I) s'avèrent intéressantes pour le traitement des états psychotiques, y compris schizophréniques, chez l'etre humain.
BE0/212415A 1983-02-18 1984-02-17 Composes pour le traitement des psychoses et leur utilisation BE898943A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/467,691 US4472397A (en) 1983-02-18 1983-02-18 Use of certain 1-substituted-triazolo-benzodiazepines to treat psychoses

Publications (1)

Publication Number Publication Date
BE898943A true BE898943A (fr) 1984-08-17

Family

ID=23856728

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/212415A BE898943A (fr) 1983-02-18 1984-02-17 Composes pour le traitement des psychoses et leur utilisation

Country Status (9)

Country Link
US (1) US4472397A (fr)
EP (1) EP0117140A1 (fr)
JP (1) JPS59157022A (fr)
AU (1) AU560215B2 (fr)
BE (1) BE898943A (fr)
DE (1) DE3401290A1 (fr)
IT (1) IT1175942B (fr)
PH (1) PH20776A (fr)
ZA (1) ZA8430B (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5706829A (en) * 1996-06-06 1998-01-13 Creighton University Method for treating neurocardiogenic syncope

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4250094A (en) * 1971-04-28 1981-02-10 The Upjohn Company 1-(Aminoalkyl) substituted-6-phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines
US4264615A (en) * 1971-04-28 1981-04-28 The Upjohn Company Compositions and process
US4012413A (en) * 1973-05-17 1977-03-15 The Upjohn Company Organic compounds and process
US4082761A (en) * 1973-09-04 1978-04-04 The Upjohn Company Triazolo[4,3-a][1,4]benzodiazepinium quaternary salts
US3894025A (en) * 1974-03-21 1975-07-08 Upjohn Co 1-Piperazino-6-phenyl-4H-s-triazolo{8 4,3-a{9 {8 1,4{9 -benzodiazepine compounds
US3996230A (en) * 1975-03-28 1976-12-07 The Upjohn Company 1-Piperazino-6-(2-pyridyl)-4H-s-triazolo[4,3-a][1,4]benzodiazepines
US4001262A (en) * 1975-10-20 1977-01-04 The Upjohn Company Process for the production of 1-[(dimethylamino)methyl]-6-phenyl-4H-triazolo[4,3-a][1,4]-benzodiazepine
JPS5259193A (en) * 1975-11-07 1977-05-16 Upjohn Co Production of aminotriazobenzodiazepine
US4180668A (en) * 1977-06-08 1979-12-25 The Upjohn Company Piperidino-4H-s-triazolo[4,3-a][1,4]benzodiazepines
US4179510A (en) * 1977-10-31 1979-12-18 The Upjohn Company Methods of treating psychosis

Also Published As

Publication number Publication date
JPS59157022A (ja) 1984-09-06
US4472397A (en) 1984-09-18
ZA8430B (en) 1984-08-29
IT1175942B (it) 1987-08-12
EP0117140A1 (fr) 1984-08-29
AU2377084A (en) 1984-08-23
DE3401290A1 (de) 1984-08-23
AU560215B2 (en) 1987-04-02
PH20776A (en) 1987-04-14
IT8419659A0 (it) 1984-02-16

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: THE UPJOHN CY

Effective date: 19930228