BE873195A - NEW DERIVATIVES OF (1,2-A) PYRIMIDINE AND PROCESS FOR THEIR PREPARATION - Google Patents
NEW DERIVATIVES OF (1,2-A) PYRIMIDINE AND PROCESS FOR THEIR PREPARATIONInfo
- Publication number
- BE873195A BE873195A BE192660A BE192660A BE873195A BE 873195 A BE873195 A BE 873195A BE 192660 A BE192660 A BE 192660A BE 192660 A BE192660 A BE 192660A BE 873195 A BE873195 A BE 873195A
- Authority
- BE
- Belgium
- Prior art keywords
- pyrimidine
- preparation
- new derivatives
- derivatives
- new
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Neurosurgery (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Anesthesiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
HU77CI1796A HU180701B (en) | 1977-12-29 | 1977-12-29 | Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering |
Publications (1)
Publication Number | Publication Date |
---|---|
BE873195A true BE873195A (en) | 1979-04-17 |
Family
ID=10994685
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE192660A BE873195A (en) | 1977-12-29 | 1978-12-29 | NEW DERIVATIVES OF (1,2-A) PYRIMIDINE AND PROCESS FOR THEIR PREPARATION |
Country Status (8)
Country | Link |
---|---|
JP (1) | JPS5498797A (en) |
BE (1) | BE873195A (en) |
CH (1) | CH642368A5 (en) |
DE (1) | DE2853273A1 (en) |
FR (1) | FR2413375A1 (en) |
GB (1) | GB2011410B (en) |
HU (1) | HU180701B (en) |
SU (1) | SU1022659A3 (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4310526A (en) | 1979-05-08 | 1982-01-12 | Farmitalia Carlo Erba S.P.A. | Substituted 6,7-methylene pyrido[1,2-a]pyrimidines useful as anti-allergic and anti-ulcer agents |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN101628913B (en) * | 2008-07-18 | 2013-01-23 | 中国科学院广州生物医药与健康研究院 | Compound as estrogen-related receptor modulator and application thereof |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
HU168014B (en) * | 1973-03-30 | 1976-02-28 | ||
US3898224A (en) * | 1974-09-09 | 1975-08-05 | Squibb & Sons Inc | 1,6,7,8-Tetrahydro-4-oxo-4H-pyrido {8 1,2-A{9 pyrimidine-9-carboalkoxy compounds |
HU173438B (en) * | 1975-11-27 | 1979-05-28 | Chinoin Gyogyszer Es Vegyeszet | Process for preparing new 4-oxo-1,6,7,8-tetrahydro-4h-pyrido-/1,2-a/pyrimidine derivatives with antiinflammatory and anticoagulant activity |
HU174693B (en) * | 1976-02-12 | 1980-03-28 | Chinoin Gyogyszer Es Vegyeszet | Process for producing condensed pyrimidine derivatives |
HU178910B (en) * | 1977-08-19 | 1982-07-28 | Chinoin Gyogyszer Es Vegyeszet | Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines |
-
1977
- 1977-12-29 HU HU77CI1796A patent/HU180701B/en unknown
-
1978
- 1978-12-09 DE DE19782853273 patent/DE2853273A1/en not_active Ceased
- 1978-12-25 SU SU782700554A patent/SU1022659A3/en active
- 1978-12-27 JP JP16453378A patent/JPS5498797A/en active Pending
- 1978-12-27 FR FR7836463A patent/FR2413375A1/en active Granted
- 1978-12-28 GB GB7850108A patent/GB2011410B/en not_active Expired
- 1978-12-28 CH CH1323178A patent/CH642368A5/en not_active IP Right Cessation
- 1978-12-29 BE BE192660A patent/BE873195A/en not_active IP Right Cessation
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4310526A (en) | 1979-05-08 | 1982-01-12 | Farmitalia Carlo Erba S.P.A. | Substituted 6,7-methylene pyrido[1,2-a]pyrimidines useful as anti-allergic and anti-ulcer agents |
US4341780A (en) | 1979-05-08 | 1982-07-27 | Farmitalia Carlo Erba S.P.A. | Substituted pyrido [1,2-a] pyrimidines useful as anti-allergic, anti-ulcer and anti-diabetic agents |
Also Published As
Publication number | Publication date |
---|---|
FR2413375A1 (en) | 1979-07-27 |
CH642368A5 (en) | 1984-04-13 |
SU1022659A3 (en) | 1983-06-07 |
HU180701B (en) | 1983-04-29 |
GB2011410B (en) | 1982-09-22 |
GB2011410A (en) | 1979-07-11 |
JPS5498797A (en) | 1979-08-03 |
DE2853273A1 (en) | 1979-07-12 |
FR2413375B1 (en) | 1983-08-05 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT Effective date: 19861231 |