BE867994A - Procede de preparation de derives de l'acide methoxy-7,alpha-(dithietane-1,3-carboxamido-2)-cephalosporanique - Google Patents

Procede de preparation de derives de l'acide methoxy-7,alpha-(dithietane-1,3-carboxamido-2)-cephalosporanique

Info

Publication number
BE867994A
BE867994A BE188469A BE188469A BE867994A BE 867994 A BE867994 A BE 867994A BE 188469 A BE188469 A BE 188469A BE 188469 A BE188469 A BE 188469A BE 867994 A BE867994 A BE 867994A
Authority
BE
Belgium
Prior art keywords
dithietane
carboxamido
methoxy
alpha
derivatives
Prior art date
Application number
BE188469A
Other languages
English (en)
Inventor
M Iwanami
T Maeda
Y Nagano
M Fujimoto
N Nagano
A Yamazaki
Original Assignee
Yamanouchi Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yamanouchi Pharma Co Ltd filed Critical Yamanouchi Pharma Co Ltd
Publication of BE867994A publication Critical patent/BE867994A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D339/00—Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/57—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with a further substituent in position 7, e.g. cephamycines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE188469A 1977-06-10 1978-06-09 Procede de preparation de derives de l'acide methoxy-7,alpha-(dithietane-1,3-carboxamido-2)-cephalosporanique BE867994A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP52068699A JPS5854157B2 (ja) 1977-06-10 1977-06-10 セフアロスポリン化合物の新規誘導体ならびにその製造方法

Publications (1)

Publication Number Publication Date
BE867994A true BE867994A (fr) 1978-12-11

Family

ID=13381266

Family Applications (1)

Application Number Title Priority Date Filing Date
BE188469A BE867994A (fr) 1977-06-10 1978-06-09 Procede de preparation de derives de l'acide methoxy-7,alpha-(dithietane-1,3-carboxamido-2)-cephalosporanique

Country Status (10)

Country Link
JP (1) JPS5854157B2 (fr)
AU (1) AU518620B2 (fr)
BE (1) BE867994A (fr)
DE (1) DE2857816C2 (fr)
FR (1) FR2405953A1 (fr)
GB (1) GB1604740A (fr)
HU (1) HU184788B (fr)
SE (1) SE454512B (fr)
SU (2) SU843752A3 (fr)
UA (2) UA5924A1 (fr)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0187355A1 (fr) 1981-09-23 1986-07-16 E.R. Squibb & Sons, Inc. Procédé de préparation d'antibiotiques bêta-lactames
EP0251330A2 (fr) 1986-07-03 1988-01-07 F. Hoffmann-La Roche Ag Dérivés de céphalosporine, leur procédé de préparation et les compositions pharmaceutiques les contenant
LT3289B (en) 1993-04-16 1995-06-26 Hoffmann La Roche Cephalosporin derivatives with antibacterial activity
US5811419A (en) * 1996-01-16 1998-09-22 Hoffmann-La Roche Inc. Isooxacephem-derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL29235A (en) * 1967-01-05 1971-10-20 Bristol Myers Co 7-(pyridylthioacetamido)cephalosporanic acid derivatives and their preparation
JPS5165789A (en) * 1974-11-30 1976-06-07 Sankyo Co 77 metokishisefuarosuhorinkagobutsuno seiho
CA1088049A (fr) * 1975-06-03 1980-10-21 Takashi Masugi Procedes d'obtention de derives d'acides alcanamido substitues en 3 et substitues en 7-3-cephem-4 carboxyliques
DE2539214C2 (de) * 1975-09-03 1984-03-29 E.R. Squibb & Sons, Inc., 08540 Princeton, N.J. 7-Methoxythienyl-ureido-cephalosporin und dieses enthaltendes Arzneimittel

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0187355A1 (fr) 1981-09-23 1986-07-16 E.R. Squibb & Sons, Inc. Procédé de préparation d'antibiotiques bêta-lactames
EP0251330A2 (fr) 1986-07-03 1988-01-07 F. Hoffmann-La Roche Ag Dérivés de céphalosporine, leur procédé de préparation et les compositions pharmaceutiques les contenant
LT3289B (en) 1993-04-16 1995-06-26 Hoffmann La Roche Cephalosporin derivatives with antibacterial activity
US5811419A (en) * 1996-01-16 1998-09-22 Hoffmann-La Roche Inc. Isooxacephem-derivatives

Also Published As

Publication number Publication date
DE2857816C2 (de) 1985-05-09
SE454512B (sv) 1988-05-09
JPS5854157B2 (ja) 1983-12-02
AU518620B2 (en) 1981-10-08
AU3698878A (en) 1979-12-13
HU184788B (en) 1984-10-29
SU843752A3 (ru) 1981-06-30
SU904525A3 (ru) 1982-02-07
UA5922A1 (uk) 1994-12-29
SE8306298L (sv) 1983-11-16
FR2405953A1 (fr) 1979-05-11
JPS543090A (en) 1979-01-11
UA5924A1 (uk) 1994-12-29
FR2405953B1 (fr) 1983-07-18
SE8306298D0 (sv) 1983-11-16
GB1604740A (en) 1981-12-16

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Legal Events

Date Code Title Description
CCPA Application for a supplementary protection certificate

Free format text: 093C0113

CCPV Grant of a supplementary protection certificate

Free format text: 093C0113, EXPIRES 19991204

RE20 Patent expired

Owner name: YAMANOUCHI PHARMACEUTICAL CO. LTD

Effective date: 19980609