BE866841A - Procede de preparation d'imidazoazines et -diazines substituees et leur utilisation - Google Patents

Procede de preparation d'imidazoazines et -diazines substituees et leur utilisation

Info

Publication number
BE866841A
BE866841A BE187505A BE187505A BE866841A BE 866841 A BE866841 A BE 866841A BE 187505 A BE187505 A BE 187505A BE 187505 A BE187505 A BE 187505A BE 866841 A BE866841 A BE 866841A
Authority
BE
Belgium
Prior art keywords
imidazoazines
diazines
substituted
preparation
Prior art date
Application number
BE187505A
Other languages
English (en)
French (fr)
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of BE866841A publication Critical patent/BE866841A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61Halogen atoms or nitro radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BE187505A 1977-05-16 1978-05-09 Procede de preparation d'imidazoazines et -diazines substituees et leur utilisation BE866841A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/796,958 US4166851A (en) 1977-05-16 1977-05-16 Certain imidazo(1,2a)pyridine derivatives

Publications (1)

Publication Number Publication Date
BE866841A true BE866841A (fr) 1978-11-09

Family

ID=25169498

Family Applications (1)

Application Number Title Priority Date Filing Date
BE187505A BE866841A (fr) 1977-05-16 1978-05-09 Procede de preparation d'imidazoazines et -diazines substituees et leur utilisation

Country Status (13)

Country Link
US (1) US4166851A (is)
JP (1) JPS53141292A (is)
BE (1) BE866841A (is)
CH (1) CH639662A5 (is)
DE (1) DE2820938A1 (is)
DK (1) DK180878A (is)
FR (1) FR2391215A1 (is)
GB (1) GB1601041A (is)
IE (1) IE46882B1 (is)
IT (1) IT1156737B (is)
LU (1) LU79651A1 (is)
NL (1) NL7804345A (is)
SE (1) SE7804777L (is)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0006614A3 (en) * 1978-06-27 1980-01-23 Merck & Co. Inc. Pyridyl- and imidazopyridyloxypropanolamines, process for preparing the same and pharmaceutical compositions containing the same

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4233301A (en) * 1977-05-16 1980-11-11 Merck & Co., Inc. Novel imidazoazines and imidazodiazines
US4330543A (en) * 1978-12-14 1982-05-18 Merck & Co., Inc. Imidazoazines and imidazodiazines
US4349673A (en) * 1980-12-23 1982-09-14 Merck & Co., Inc. Benzoxazines
US4656168A (en) * 1980-12-23 1987-04-07 Merck & Co., Inc. (3-aralkylamino-2-or-propoxy)heterocyclic compounds in method of effecting bronchodilation
US4331679A (en) * 1980-12-23 1982-05-25 Merck Sharp & Dohme (I.A.) Corp. (3-Aralkylamino-2-or-propoxy) heterocyclic compounds
US4442094A (en) * 1980-12-23 1984-04-10 Merck & Co., Inc. (3-Aralkylamino-2-or-propoxy)heterocyclic compounds
US4391806A (en) * 1982-07-12 1983-07-05 The Dow Chemical Company Substituted tetrahydropyridazino-(1,6-A)benzimidazoles and use as bronchodilators
ZA839398B (en) * 1982-12-27 1985-08-28 Lilly Co Eli Substituted imidazopyrimidines-pyrazines,and-triazines
US4636502A (en) * 1982-12-27 1987-01-13 Eli Lilly And Company Methods of producing a positive inotropic effect or vasodilation by administration of 2-phenyl imidazo pyrimidines and pyrazines
US4537889A (en) * 1982-12-27 1985-08-27 Eli Lilly And Company Inotropic agents
DE3446778A1 (de) * 1984-12-21 1986-07-03 Dr. Karl Thomae Gmbh, 7950 Biberach Neue imidazoderivate, ihre herstellung und diese verbindungen enthaltende arzneimittel
GB8719368D0 (en) * 1987-08-15 1987-09-23 Wellcome Found Heterocyclic compounds
PH27291A (en) * 1989-01-31 1993-05-04 Takeda Chemical Industries Ltd Imidazolpyrimidazines their production and use
EP0440119A1 (en) * 1990-01-31 1991-08-07 Takeda Chemical Industries, Ltd. Imidazopyridazine compounds, their production and use
ATE119774T1 (de) * 1990-07-30 1995-04-15 Takeda Chemical Industries Ltd Imidazopyridinderivate und ihre verwendung.
US5420133A (en) * 1993-03-19 1995-05-30 Merck & Co., Inc. Quinazolinones substituted with phenoxyphenylacetic acid derivatives
DE10145457A1 (de) * 2001-09-14 2003-04-03 Basf Ag Substituierte Imidazo[1,2-a]-5,6,7,8-tetrahydropyridin-8-one, Verfahren zu ihrer Herstellung, sowie deren Verwendung zur Herstellung von Imidazo[1,2,-a]pyridinen
US20070078136A1 (en) 2005-09-22 2007-04-05 Bristol-Myers Squibb Company Fused heterocyclic compounds useful as kinase modulators
AU2009279936A1 (en) * 2008-08-05 2010-02-11 Banyu Pharmaceutical Co., Ltd. Therapeutic compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR208397A1 (es) * 1973-02-20 1976-12-27 Ciba Geigy Ag Procedimiento para la elaboracion de compuestos de 1-piridiloxi-2-hidroxi-3-amino-propano1-piraziniloxi-2-hidroxi-3-amino-propano y 1-pirimidiniloxi-2-hidroxi-3-amino-propan
US4071630A (en) * 1975-04-08 1978-01-31 Sandoz Ltd. 1-Substituted-amino-3-(4-furo[3,2-c]pyridinyloxy)-2-propanols
CH614711A5 (is) * 1975-04-08 1979-12-14 Sandoz Ag

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0006614A3 (en) * 1978-06-27 1980-01-23 Merck & Co. Inc. Pyridyl- and imidazopyridyloxypropanolamines, process for preparing the same and pharmaceutical compositions containing the same

Also Published As

Publication number Publication date
JPS53141292A (en) 1978-12-08
DK180878A (da) 1978-11-17
FR2391215B1 (is) 1981-12-11
FR2391215A1 (fr) 1978-12-15
DE2820938A1 (de) 1978-11-23
IE780923L (en) 1978-11-16
IT7849338A0 (it) 1978-05-12
JPS623153B2 (is) 1987-01-23
NL7804345A (nl) 1978-11-20
IE46882B1 (en) 1983-10-19
CH639662A5 (de) 1983-11-30
LU79651A1 (fr) 1979-02-02
IT1156737B (it) 1987-02-04
GB1601041A (en) 1981-10-21
SE7804777L (sv) 1978-11-17
US4166851A (en) 1979-09-04

Similar Documents

Publication Publication Date Title
FR2449699B1 (fr) Polyetherpolyamides et leur procede de preparation
BE891094Q (fr) N-benzoyl-n'-pyridyloxy-phenylurees et leur procede de preparation
BE866841A (fr) Procede de preparation d'imidazoazines et -diazines substituees et leur utilisation
BE866226A (fr) Procede pour la preparation de thymosine alpha1 et d'un analogue
BE866660A (fr) Procede de preparation de n-alkyl-n-acyl-thienamycines et leur utilisation
BE869163A (fr) Thioethers basiques et leur procede de preparation
BE863872A (fr) Steroides-11 beta-substitues et procede de leur preparation
BE866957A (fr) Procede de preparation d'homopolymerisats et de copolymerisats d'alpha-mono-olefines
BE850855A (fr) Procede de preparation d'homopolymeres et copolymeres d'alpha-mono-olefines
BE865136A (fr) Composes de 2-phenoxy-5-trifluoromethylpyridine et leur procede de preparation
BE869074A (fr) Diurethannes, leur procede de preparation et leur utilisation
BE865805A (fr) 1,2,3-thiadiazol-3-in-5-ylidene-urees, leur procede de preparation et leur utilisation
BE856220A (fr) Polyether-polyureides et procede de leur preparation
BE884286A (fr) Acylurees, leur procede de preparation et leur utilisation
BE885946A (fr) Nouvelles pyridothienotriazines et leur procede de preparation
FR2305416A1 (fr) Procede de preparation de tricosene-(9) et d'heneicosene-(9)
BE857100A (fr) Procede de preparation d'homopolymeres et de copolymeres d'&-mono-olefines
BE872294A (fr) Procede de preparation de 3-iodorifamycine s et de 3-bromorifamycine s
BE878127A (fr) Amides 1,2,3-triazolecarboxyliques, leur procede de preparation et leur utilisation
BE884652R (fr) Phenoxyalcoyl trialcoxysilanes et leur procede de preparation
BE858806A (fr) Procede pour la preparation de glycol-aldehyde et d'ethylene-glycol
BE867086A (fr) Composes d'azacyclyle et procede pour leur preparation
RO78342A (ro) Procedeu de preparare a unor imino-eteri de benztiazoline si benzoxazoline
FR2424281B1 (fr) Phenoxyalcoyl trialcoxysilanes et leur procede de preparation
LU79551A1 (fr) Procede de preparation de nouvelles 3-amino-2-or-propoxy-naphtyridines et leur utilisation

Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: MERCK & CO. INC.

Effective date: 19850509