BE848696A - Derives de la 3,4-dihydro-quinazoline a activite antiallergique et procede pour leur preparation, - Google Patents
Derives de la 3,4-dihydro-quinazoline a activite antiallergique et procede pour leur preparation,Info
- Publication number
- BE848696A BE848696A BE172653A BE172653A BE848696A BE 848696 A BE848696 A BE 848696A BE 172653 A BE172653 A BE 172653A BE 172653 A BE172653 A BE 172653A BE 848696 A BE848696 A BE 848696A
- Authority
- BE
- Belgium
- Prior art keywords
- quinazoline
- dihydro
- derivatives
- preparation
- antiallergic activity
- Prior art date
Links
- LGACUMPRRMLUFZ-UHFFFAOYSA-N 1,4-dihydroquinazoline Chemical class C1=CC=C2CN=CNC2=C1 LGACUMPRRMLUFZ-UHFFFAOYSA-N 0.000 title 1
- 230000003266 anti-allergic effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
- C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
- C07D239/90—Oxygen atoms with acyclic radicals attached in position 2 or 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/93—Sulfur atoms
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Pulmonology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Immunology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT29998/75A IT1050750B (it) | 1975-12-05 | 1975-12-05 | Derivati della 3.4 di idro chinazolina |
Publications (1)
Publication Number | Publication Date |
---|---|
BE848696A true BE848696A (fr) | 1977-03-16 |
Family
ID=11228830
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE172653A BE848696A (fr) | 1975-12-05 | 1976-11-24 | Derives de la 3,4-dihydro-quinazoline a activite antiallergique et procede pour leur preparation, |
Country Status (22)
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4419357A (en) | 1982-01-18 | 1983-12-06 | The Dow Chemical Company | 3-(1H-Tetrazol-5-yl)-4(3H)-quinazolinones |
IL69274A (en) * | 1982-08-05 | 1986-08-31 | Erba Farmitalia | (substituted amino)derivatives of 3-benzylidene-pyrrolo(2,1-b)quinazolin-9-ones and 6-benzylidene-pyrido(2,1-b)quinazolin-11-ones,their preparation and pharmaceutical compositions containing them |
US4666913A (en) * | 1985-11-22 | 1987-05-19 | William H. Rorer, Inc. | Hydroxy and aminothiazolyl-benzodiazinone compounds, cardiotonic compositions including the same, and their uses |
GB8827988D0 (en) * | 1988-11-30 | 1989-01-05 | Smith Kline French Lab | Chemical compounds |
US5430148A (en) * | 1992-03-31 | 1995-07-04 | Agouron Pharmaceuticals, Inc. | Antiproliferative quinazolines |
US6632961B1 (en) * | 1998-05-22 | 2003-10-14 | Abbott Laboratories | Antiangiogenic drug to treat cancer, arthritis and retinopathy |
DE69934113T2 (de) * | 1998-05-22 | 2007-06-06 | Abbott Laboratories, Abbott Park | Antiangiogene substanz zur behandlung von krebs, arthritis und netzhauterkrankungen |
CO5170498A1 (es) * | 1999-05-28 | 2002-06-27 | Abbott Lab | Biaril sulfonamidas son utiles como inhibidores de proliferacion celular |
US7893071B2 (en) * | 2001-04-23 | 2011-02-22 | University Of Virginia Patent Foundation | Synthesis and evaluation of novel phthalimide mimics as anti-angiogenic |
CN100518740C (zh) * | 2003-06-06 | 2009-07-29 | 阿里克斯股份公司 | 杂环化合物作为scce抑制剂的制药用途 |
EP1631295B1 (en) * | 2003-06-06 | 2010-03-03 | Arexis AB | Use of condensed heterocyclic compounds as scce inhibitors for the treatment of skin diseases |
CN101501007B (zh) * | 2006-08-08 | 2014-01-29 | Aska制药株式会社 | 喹唑啉衍生物 |
SI2118074T1 (sl) | 2007-02-01 | 2014-05-30 | Resverlogix Corp. | Spojine za preprečevanje in zdravljenje kardiovaskularnih bolezni |
CA3146333A1 (en) | 2009-03-18 | 2010-09-23 | Resverlogix Corp. | Phenyl-quinazolin-4(3h)-one and phenyl-pyrido[2,3-d]pyrimidin-4(3h)-one derivatives and compositions thereof useful as anti-inflammatory agents |
MX352614B (es) | 2009-04-22 | 2017-12-01 | Resverlogix Corp | Nuevos agentes anti-inflamatorios. |
JP6903585B2 (ja) | 2015-03-13 | 2021-07-14 | レスバーロジックス コーポレイション | 補体関連疾患の治療のための組成物および治療方法 |
GB201510254D0 (en) * | 2015-06-12 | 2015-07-29 | Syngenta Participations Ag | Improvements in or relating to organic compounds |
US12012410B2 (en) * | 2018-06-27 | 2024-06-18 | Reborna Biosciences, Inc. | Substituted pyrazolo[1,5-a]pyrazines for spinal muscular atrophy |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3696102A (en) * | 1970-03-09 | 1972-10-03 | Pfizer & Co C | Process for the synthesis of substituted quinazolin-4-ones |
GB1301319A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1970-07-13 | 1972-12-29 |
-
1975
- 1975-12-05 IT IT29998/75A patent/IT1050750B/it active
-
1976
- 1976-11-02 US US05/738,221 patent/US4251531A/en not_active Expired - Lifetime
- 1976-11-04 IL IL50849A patent/IL50849A/xx unknown
- 1976-11-10 ZA ZA766745A patent/ZA766745B/xx unknown
- 1976-11-10 AU AU19472/76A patent/AU505660B2/en not_active Expired
- 1976-11-24 BE BE172653A patent/BE848696A/xx not_active IP Right Cessation
- 1976-11-25 FI FI763391A patent/FI64359C/fi not_active IP Right Cessation
- 1976-11-30 DE DE19762654215 patent/DE2654215A1/de not_active Withdrawn
- 1976-12-01 GB GB50164/76A patent/GB1523081A/en not_active Expired
- 1976-12-01 NZ NZ182778A patent/NZ182778A/xx unknown
- 1976-12-02 NL NL7613450A patent/NL7613450A/xx not_active Application Discontinuation
- 1976-12-02 AT AT894376A patent/AT355029B/de not_active IP Right Cessation
- 1976-12-02 FR FR7636343A patent/FR2333511A1/fr active Granted
- 1976-12-03 SE SE7613588A patent/SE7613588L/xx not_active Application Discontinuation
- 1976-12-03 DK DK546776A patent/DK147855C/da not_active IP Right Cessation
- 1976-12-03 HU HU76EA167A patent/HU177817B/hu unknown
- 1976-12-03 CS CS767886A patent/CS194786B2/cs unknown
- 1976-12-03 SU SU762426155A patent/SU786894A3/ru active
- 1976-12-03 NO NO764135A patent/NO146095C/no unknown
- 1976-12-03 CA CA267,090A patent/CA1084051A/en not_active Expired
- 1976-12-03 CH CH1527276A patent/CH626073A5/de not_active IP Right Cessation
- 1976-12-06 JP JP51146444A patent/JPS5271485A/ja active Granted
-
1980
- 1980-11-28 CH CH885580A patent/CH626075A5/de not_active IP Right Cessation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BE849794A (fr) | Derives de carbostyrile et leur procede de preparation | |
FR2315930A1 (fr) | Derives de 1,4-dihydropyridine et leur procede de preparation | |
BE848696A (fr) | Derives de la 3,4-dihydro-quinazoline a activite antiallergique et procede pour leur preparation, | |
FR2349579A1 (fr) | Derives de 1,2-dihydronaphtalene et leur procede de preparation | |
BE823027A (fr) | Derives d'isoquinoleine et leur procede de preparation | |
BE848659A (fr) | Nouveau catalyseur d'eposydation et procede de sa preparation, | |
BE818975A (fr) | Derives d'acides phenoxypropioniques et leur procede de preparation | |
FR2299032A1 (fr) | Derives de tetrahydroisoquinoleine et leur procede de preparation | |
BE861289A (fr) | Procede de preparation de derives des acides perfluoroalcane-carboxyliques et perfluoroalcane-sulfiniques | |
BE847347A (fr) | Nouveaux derives d'acides phenoxy-alkyl-carboxyliques et procede pour leur preparation, | |
FR2319345A1 (fr) | Derives de thiazolidine, leur procede de preparation et leur application | |
BE855236A (fr) | Derives omega-nor-aromatiques de 13,14-dehydro-prostaglandines et procede pour leur preparation | |
BE827870A (fr) | Derives d'emidazole et leur procede de preparation | |
BE858157A (fr) | Derives d'acides heterocyclyl-carboxyliques acyles et procede pour leur preparation | |
FR2343724A1 (fr) | Nouveaux derives hydrosolubles de nitrosouree doues d'activite antitumorale et leur procede de preparation | |
BE841538A (fr) | Procede de preparation de derives de carbanate et d'uree | |
FR2317930A1 (fr) | Nouveaux derives d'apovincaminol, leur procede de preparation et leur application | |
BE841165A (fr) | Derives d'acides 8-aza-prostanoiques et leur procede de preparation | |
BE859081A (fr) | Derives de l'anthraquinone et leur procede de preparation | |
BE843576A (fr) | Derives de 1,4-dihydropyridine et leur procede de preparation | |
BE821893A (fr) | Derives d'adenine et leur procede de preparation | |
BE848627A (fr) | Derives substitues d'aminobenzaldehydes et leur procede de preparation, | |
BE872594A (fr) | Derives d'acides 1-hydrocarbyl-pyrrole-2-acetiques et leur procede de production | |
BE862095A (fr) | Derives de l'imidazole, leur procede de preparation et leur application | |
BE777849A (fr) | Nouveaux derives gem.-diaryl-ethyleniques doues d'activite anti-histaminique et leur procede de preparation |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: CARLO ERBA S.P.A. Effective date: 19851130 |