BE837878A - 4-arylpiperidines et procedes pour les preparer - Google Patents

4-arylpiperidines et procedes pour les preparer

Info

Publication number
BE837878A
BE837878A BE163778A BE163778A BE837878A BE 837878 A BE837878 A BE 837878A BE 163778 A BE163778 A BE 163778A BE 163778 A BE163778 A BE 163778A BE 837878 A BE837878 A BE 837878A
Authority
BE
Belgium
Prior art keywords
arylpiperidines
preparing
methods
Prior art date
Application number
BE163778A
Other languages
English (en)
French (fr)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to US05/533,642 priority Critical patent/US4048314A/en
Priority to FI753525A priority patent/FI753525A7/fi
Priority to SE7514177A priority patent/SE7514177L/xx
Priority to CA242,119A priority patent/CA1053230A/en
Priority to AU10381/76A priority patent/AU1038176A/en
Application filed filed Critical
Priority to BE163778A priority patent/BE837878A/xx
Publication of BE837878A publication Critical patent/BE837878A/xx
Priority to US05/832,567 priority patent/US4146629A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D211/62—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
    • C07D211/64—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4 having an aryl radical as the second substituent in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE163778A 1974-12-17 1976-01-23 4-arylpiperidines et procedes pour les preparer BE837878A (fr)

Priority Applications (7)

Application Number Priority Date Filing Date Title
US05/533,642 US4048314A (en) 1974-12-17 1974-12-17 Morpholino containing 4-arylpiperidine derivatives
FI753525A FI753525A7 (enExample) 1974-12-17 1975-12-15
SE7514177A SE7514177L (sv) 1974-12-17 1975-12-16 Nya 4-arylpiperidinderivat och forfaranden for deras framstellning
CA242,119A CA1053230A (en) 1974-12-17 1975-12-17 4-arylpiperidine derivatives and processes for the production thereof
AU10381/76A AU1038176A (en) 1974-12-17 1976-01-19 4-arylpiperidine derivatives
BE163778A BE837878A (fr) 1974-12-17 1976-01-23 4-arylpiperidines et procedes pour les preparer
US05/832,567 US4146629A (en) 1974-12-17 1977-09-12 4-arylpiperidine derivatives

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/533,642 US4048314A (en) 1974-12-17 1974-12-17 Morpholino containing 4-arylpiperidine derivatives
BE163778A BE837878A (fr) 1974-12-17 1976-01-23 4-arylpiperidines et procedes pour les preparer

Publications (1)

Publication Number Publication Date
BE837878A true BE837878A (fr) 1976-05-14

Family

ID=25649081

Family Applications (1)

Application Number Title Priority Date Filing Date
BE163778A BE837878A (fr) 1974-12-17 1976-01-23 4-arylpiperidines et procedes pour les preparer

Country Status (6)

Country Link
US (2) US4048314A (enExample)
AU (1) AU1038176A (enExample)
BE (1) BE837878A (enExample)
CA (1) CA1053230A (enExample)
FI (1) FI753525A7 (enExample)
SE (1) SE7514177L (enExample)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4286095A (en) * 1976-08-05 1981-08-25 Canada Packers Inc. 4-Arylpiperidine derivatives
USRE46117E1 (en) 1999-12-22 2016-08-23 Teva Pharmaceuticals International Gmbh Modulators of dopamine neurotransmission
SE0401465D0 (sv) * 2004-06-08 2004-06-08 Carlsson A Research Ab New substituted piperdines as modulators of dopamine neurotransmission
CA2584831C (en) * 2004-10-13 2013-09-17 Neurosearch Sweden Ab Process for the synthesis of 4-(3-methanesulfonylphenyl)-1-n-propyl-piperidine
MX2007004216A (es) * 2004-10-13 2007-10-10 Neurosearch Sweden Ab Proceso para la sintesis de 4-(3-sulfonil)-piperidinas.
IL165365A0 (en) 2004-11-24 2006-01-15 Q Core Ltd Finger-type peristaltic pump
CN102766079B (zh) * 2011-05-06 2015-04-08 上海医药工业研究院 一类吡咯烷衍生物、其制备方法及应用
WO2013086425A1 (en) 2011-12-08 2013-06-13 IVAX International GmbH The hydrobromide salt of pridopidine
US20130267552A1 (en) 2012-04-04 2013-10-10 IVAX International GmbH Pharmaceutical compositions for combination therapy
TR201911032T4 (tr) 2015-05-18 2019-08-21 Tolero Pharmaceuticals Inc Artırılmış biyoyararlanıma sahip alvocıdıb ön ilaçları.
US11279694B2 (en) 2016-11-18 2022-03-22 Sumitomo Dainippon Pharma Oncology, Inc. Alvocidib prodrugs and their use as protein kinase inhibitors
US11497756B2 (en) 2017-09-12 2022-11-15 Sumitomo Pharma Oncology, Inc. Treatment regimen for cancers that are insensitive to BCL-2 inhibitors using the MCL-1 inhibitor alvocidib
US11542084B2 (en) 2018-07-20 2023-01-03 The Procter & Gamble Company Flexible package and method of manufacture
KR20210099066A (ko) 2018-12-04 2021-08-11 스미토모 다이니폰 파마 온콜로지, 인크. 암의 치료를 위한 작용제로서 사용하기 위한 cdk9 억제제 및 그의 다형체
US11793802B2 (en) 2019-03-20 2023-10-24 Sumitomo Pharma Oncology, Inc. Treatment of acute myeloid leukemia (AML) with venetoclax failure

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3125574A (en) * 1964-03-17 I-aroylpropylx-acyl-x-amino-
US2167351A (en) * 1937-08-07 1939-07-25 Winthrop Chem Co Inc Piperidine compounds and a process of preparing them
US2748140A (en) * 1954-10-07 1956-05-29 Rohm & Haas 3-hydroxymethyl-4-phenyltetrahydro-pyridines and their esters
US3080372A (en) * 1960-03-25 1963-03-05 Res Lab Dr C Janssen 1-aroylalkyl-4-arylpiperidine derivatives
US3371094A (en) * 1961-08-08 1968-02-27 Sterling Drug Inc N-(amidoximino-lower-alkyl)-and n-amidino-n-[(1-piperidyl)-lower-alkyl]amines
US3158616A (en) * 1962-03-16 1964-11-24 Boehringer Sohn Ingelheim Nu-substituted 4-aryl-4-alkanoyloxypiperidines
US3845064A (en) * 1972-10-24 1974-10-29 Wyeth John & Brother Ltd Piperidinethioamides

Also Published As

Publication number Publication date
SE7514177L (sv) 1976-06-18
US4048314A (en) 1977-09-13
AU1038176A (en) 1977-07-28
FI753525A7 (enExample) 1976-06-18
US4146629A (en) 1979-03-27
CA1053230A (en) 1979-04-24

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