BE833291A - NEW CYCLOAKLYL DERIVATIVES OF 1-ARYLOXY-3-AMINO-2-PROPANOLS, THEIR PREPARATION METHODS, AND THEIR THERAPEUTIC USES - Google Patents
NEW CYCLOAKLYL DERIVATIVES OF 1-ARYLOXY-3-AMINO-2-PROPANOLS, THEIR PREPARATION METHODS, AND THEIR THERAPEUTIC USESInfo
- Publication number
- BE833291A BE833291A BE159930A BE159930A BE833291A BE 833291 A BE833291 A BE 833291A BE 159930 A BE159930 A BE 159930A BE 159930 A BE159930 A BE 159930A BE 833291 A BE833291 A BE 833291A
- Authority
- BE
- Belgium
- Prior art keywords
- cycloaklyl
- propanols
- aryloxy
- derivatives
- amino
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/096—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/12—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
- C07D303/18—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by etherified hydroxyl radicals
- C07D303/20—Ethers with hydroxy compounds containing no oxirane rings
- C07D303/22—Ethers with hydroxy compounds containing no oxirane rings with monohydroxy compounds
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US50540874A | 1974-09-12 | 1974-09-12 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE833291A true BE833291A (en) | 1976-03-11 |
Family
ID=24010183
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE159930A BE833291A (en) | 1974-09-12 | 1975-09-11 | NEW CYCLOAKLYL DERIVATIVES OF 1-ARYLOXY-3-AMINO-2-PROPANOLS, THEIR PREPARATION METHODS, AND THEIR THERAPEUTIC USES |
Country Status (9)
Country | Link |
---|---|
JP (1) | JPS51125038A (en) |
BE (1) | BE833291A (en) |
DD (1) | DD122519A5 (en) |
DE (1) | DE2540552A1 (en) |
DK (1) | DK405775A (en) |
ES (1) | ES440890A1 (en) |
FR (1) | FR2284321A1 (en) |
NL (1) | NL7510781A (en) |
SE (1) | SE7510153L (en) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4665094A (en) * | 1985-08-29 | 1987-05-12 | Merck & Co., Inc. | Oculoselective beta-blockers for treatment of elevated intraocular pressure |
US4945182A (en) * | 1985-12-24 | 1990-07-31 | Merck & Co., Inc. | Oculoselective beta-blockers |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2522325B1 (en) * | 1982-02-26 | 1985-08-09 | Delalande Sa | NOVEL ARYLIC DERIVATIVES OF PIPERAZINE, HOMOPIPERAZINE AND N, N'-DIALKYL DIAMINO-1,2 ETHANE, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION |
JP3441665B2 (en) * | 1999-02-04 | 2003-09-02 | 株式会社資生堂 | (2-Substituted oxyphenyl) alkaneamide derivatives, hair tonics, skin external preparations |
PL209602B1 (en) | 2005-10-20 | 2011-09-30 | Inst Chemii Bioorg Pan | Synthesis of amide of the 3- (4-hydroxyphenyl)propane acid |
EP2118080B1 (en) | 2007-02-09 | 2016-08-31 | Ocera Therapeutics, Inc. | Macrocyclic ghrelin receptor modulators and methods of using the same |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1937477C3 (en) * | 1969-07-23 | 1980-04-10 | C.H. Boehringer Sohn, 6507 Ingelheim | I-phenoxy-2-hydroxy-3- (l -methylcycloalkylamino) propane, process for their preparation and medicaments containing them |
GB1391444A (en) * | 1971-07-13 | 1975-04-23 | Ici Ltd | Chemical process for the manufacture of alkanolamine derivatives |
-
1975
- 1975-09-11 DK DK405775A patent/DK405775A/en unknown
- 1975-09-11 BE BE159930A patent/BE833291A/en unknown
- 1975-09-11 SE SE7510153A patent/SE7510153L/en unknown
- 1975-09-11 DE DE19752540552 patent/DE2540552A1/en active Pending
- 1975-09-12 FR FR7528137A patent/FR2284321A1/en active Granted
- 1975-09-12 JP JP50110138A patent/JPS51125038A/en active Pending
- 1975-09-12 NL NL7510781A patent/NL7510781A/en unknown
- 1975-09-12 ES ES440890A patent/ES440890A1/en not_active Expired
- 1975-09-12 DD DD188308A patent/DD122519A5/xx unknown
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4665094A (en) * | 1985-08-29 | 1987-05-12 | Merck & Co., Inc. | Oculoselective beta-blockers for treatment of elevated intraocular pressure |
US4945182A (en) * | 1985-12-24 | 1990-07-31 | Merck & Co., Inc. | Oculoselective beta-blockers |
Also Published As
Publication number | Publication date |
---|---|
DK405775A (en) | 1976-03-13 |
ES440890A1 (en) | 1977-04-01 |
NL7510781A (en) | 1976-03-16 |
DE2540552A1 (en) | 1976-03-25 |
SE7510153L (en) | 1976-05-07 |
FR2284321B1 (en) | 1978-07-28 |
FR2284321A1 (en) | 1976-04-09 |
JPS51125038A (en) | 1976-11-01 |
DD122519A5 (en) | 1976-10-12 |
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