BE798170A - Procede de preparation d'acides 6-(alpha-(guanyl-ureido- alcanoylamino)aracylamino) penicillaniques - Google Patents

Procede de preparation d'acides 6-(alpha-(guanyl-ureido- alcanoylamino)aracylamino) penicillaniques

Info

Publication number
BE798170A
BE798170A BE1004965A BE1004965A BE798170A BE 798170 A BE798170 A BE 798170A BE 1004965 A BE1004965 A BE 1004965A BE 1004965 A BE1004965 A BE 1004965A BE 798170 A BE798170 A BE 798170A
Authority
BE
Belgium
Prior art keywords
aracylamino
alcanoylamino
guanyl
ureido
alpha
Prior art date
Application number
BE1004965A
Other languages
English (en)
French (fr)
Inventor
E S Hamanaka
D S Patton
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of BE798170A publication Critical patent/BE798170A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/04—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms
    • C07C275/06—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an acyclic and saturated carbon skeleton
    • C07C275/16—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an acyclic and saturated carbon skeleton being further substituted by carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/28—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to cyano groups, e.g. cyanoguanidines, dicyandiamides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C335/30—Isothioureas
    • C07C335/34—Isothioureas having sulfur atoms of isothiourea groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C335/30—Isothioureas
    • C07C335/38—Isothioureas containing any of the groups, X being a hetero atom, Y being any atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/30—Oxygen or sulfur atoms
    • C07D233/42—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44—Nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44—Nitrogen atoms not forming part of a nitro radical
    • C07D233/46—Nitrogen atoms not forming part of a nitro radical with only hydrogen atoms attached to said nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BE1004965A 1972-05-16 1973-04-13 Procede de preparation d'acides 6-(alpha-(guanyl-ureido- alcanoylamino)aracylamino) penicillaniques BE798170A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US00253856A US3838153A (en) 1972-05-16 1972-05-16 6-(alpha-(guanylureidoalkanoylamino)aracylamino)penicillanic acids

Publications (1)

Publication Number Publication Date
BE798170A true BE798170A (fr) 1973-10-15

Family

ID=22961983

Family Applications (1)

Application Number Title Priority Date Filing Date
BE1004965A BE798170A (fr) 1972-05-16 1973-04-13 Procede de preparation d'acides 6-(alpha-(guanyl-ureido- alcanoylamino)aracylamino) penicillaniques

Country Status (23)

Country Link
US (1) US3838153A (en:Method)
JP (1) JPS5533712B2 (en:Method)
AR (1) AR195914A1 (en:Method)
AT (1) AT325767B (en:Method)
AU (1) AU475922B2 (en:Method)
BE (1) BE798170A (en:Method)
CA (1) CA1010444A (en:Method)
CH (1) CH573434A5 (en:Method)
DE (1) DE2318986A1 (en:Method)
DK (1) DK137046B (en:Method)
ES (1) ES413937A1 (en:Method)
FI (1) FI56534C (en:Method)
FR (1) FR2184609B1 (en:Method)
GB (1) GB1404469A (en:Method)
IE (1) IE37491B1 (en:Method)
IL (1) IL41937A (en:Method)
NL (1) NL7305355A (en:Method)
PH (1) PH10024A (en:Method)
PL (1) PL89245B1 (en:Method)
SE (1) SE415976B (en:Method)
SU (1) SU504491A3 (en:Method)
YU (1) YU36965B (en:Method)
ZA (1) ZA732343B (en:Method)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1462421A (en) * 1973-12-14 1977-01-26 Pfizer 6-a-amidino-and -'midoylaminoalkanoylamino aracylamino-penicillanic acids and their preparation
US3994965A (en) * 1974-08-09 1976-11-30 Pfizer Inc. D-N-(guanylureidoacetyl)-α-aminophenyl acetic acid and D-N-(guanylureidoacetyl)-α-aminophenyl acetyl chloride
JPS5562537U (en:Method) * 1978-10-20 1980-04-28
DE3014353A1 (de) * 1980-04-15 1982-01-21 Bayer Ag, 5090 Leverkusen Trisubstituierte cyanguanidine, verfahren zu ihrer herstellung sowie ihre verwendung als fungizide
JPS56161152A (en) * 1980-05-12 1981-12-11 Tachikawa Spring Co Manufacture of steel band with resin
IL134298A0 (en) 1997-08-21 2001-04-30 Quark Biotech Inc Hypoxia-regulating genes
US20030104973A1 (en) * 1997-08-21 2003-06-05 Quark Biotech, Inc. Hypoxia-regulated genes
US7973156B2 (en) * 1997-08-21 2011-07-05 Quark Pharmaceuticals Inc. Hypoxia-regulated genes

Also Published As

Publication number Publication date
AR195914A1 (es) 1973-11-15
SU504491A3 (ru) 1976-02-25
FI56534C (fi) 1980-02-11
IE37491L (en) 1973-11-16
ZA732343B (en) 1974-01-30
AT325767B (de) 1975-11-10
AU5428373A (en) 1974-10-10
ES413937A1 (es) 1976-06-01
FI56534B (fi) 1979-10-31
FR2184609A1 (en:Method) 1973-12-28
IL41937A (en) 1976-10-31
US3838153A (en) 1974-09-24
CH573434A5 (en:Method) 1976-03-15
CA1010444A (en) 1977-05-17
DK137046B (da) 1978-01-09
IL41937A0 (en) 1973-06-29
YU36965B (en) 1984-08-31
DE2318986A1 (de) 1973-12-06
JPS5533712B2 (en:Method) 1980-09-02
NL7305355A (en:Method) 1973-11-20
FR2184609B1 (en:Method) 1976-10-22
AU475922B2 (en) 1976-09-09
SE415976B (sv) 1980-11-17
PL89245B1 (en:Method) 1976-11-30
ATA341573A (de) 1975-01-15
IE37491B1 (en) 1977-08-03
PH10024A (en) 1976-07-13
DK137046C (en:Method) 1978-06-12
YU97773A (en) 1982-06-18
GB1404469A (en) 1975-08-28
JPS4924991A (en:Method) 1974-03-05

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