AU753476B2 - Taste masking rapid release coating system - Google Patents
Taste masking rapid release coating system Download PDFInfo
- Publication number
- AU753476B2 AU753476B2 AU19220/00A AU1922000A AU753476B2 AU 753476 B2 AU753476 B2 AU 753476B2 AU 19220/00 A AU19220/00 A AU 19220/00A AU 1922000 A AU1922000 A AU 1922000A AU 753476 B2 AU753476 B2 AU 753476B2
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- AU
- Australia
- Prior art keywords
- core
- taste masking
- weight
- patient
- drug
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- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
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- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Emergency Medicine (AREA)
- Zoology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US11003298P | 1998-11-25 | 1998-11-25 | |
| US60/110032 | 1998-11-25 | ||
| PCT/US1999/027981 WO2000030617A1 (en) | 1998-11-25 | 1999-11-24 | Taste masking rapid release coating system |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU1922000A AU1922000A (en) | 2000-06-13 |
| AU753476B2 true AU753476B2 (en) | 2002-10-17 |
Family
ID=22330879
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU19220/00A Ceased AU753476B2 (en) | 1998-11-25 | 1999-11-24 | Taste masking rapid release coating system |
Country Status (6)
| Country | Link |
|---|---|
| EP (2) | EP2260836B1 (enExample) |
| JP (1) | JP2002530322A (enExample) |
| AU (1) | AU753476B2 (enExample) |
| CA (1) | CA2351720C (enExample) |
| ES (1) | ES2601855T3 (enExample) |
| WO (1) | WO2000030617A1 (enExample) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0027357D0 (en) | 2000-11-09 | 2000-12-27 | Bradford Particle Design Plc | Particle formation methods and their products |
| AR034813A1 (es) * | 2001-07-20 | 2004-03-17 | Novartis Ag | Composiciones farmaceuticas y uso de las mismas |
| GB0208742D0 (en) | 2002-04-17 | 2002-05-29 | Bradford Particle Design Ltd | Particulate materials |
| US6753009B2 (en) | 2002-03-13 | 2004-06-22 | Mcneil-Ppc, Inc. | Soft tablet containing high molecular weight polyethylene oxide |
| US7582284B2 (en) | 2002-04-17 | 2009-09-01 | Nektar Therapeutics | Particulate materials |
| US9339459B2 (en) | 2003-04-24 | 2016-05-17 | Nektar Therapeutics | Particulate materials |
| AU2002368090A1 (en) * | 2002-07-17 | 2004-02-09 | Eurand Pharmaceuticals Ltd | Process for the preparation of pharmaceutical microcapsules with enhanced tastemasking and high dissolution rate |
| US20040258752A1 (en) * | 2003-01-31 | 2004-12-23 | Paruthi Manoj Kumar | Taste masking pharmaceutical composition and process for its preparation |
| WO2004098561A2 (en) | 2003-05-08 | 2004-11-18 | Nektar Therapeutics Uk Ltd | Particulate materials |
| US20040265372A1 (en) | 2003-06-27 | 2004-12-30 | David Wynn | Soft tablet containing high molecular weight cellulosics |
| MX2007008320A (es) * | 2005-01-06 | 2007-09-07 | Cima Labs Inc | Sistema enmascarador de sabor para farmacos no plastificantes. |
| US20070098746A1 (en) * | 2005-11-02 | 2007-05-03 | Nichols William M | Multi-layered coating technology for taste masking |
| WO2007143131A2 (en) * | 2006-06-01 | 2007-12-13 | Cima Labs, Inc. | Prednisolone sodium phosphate formulations |
| US8637076B2 (en) | 2006-06-01 | 2014-01-28 | Cima Labs Inc. | Prednisolone salt formulations |
| EA017832B1 (ru) * | 2006-08-04 | 2013-03-29 | Этифарм | Гранулы и орально дезинтегрируемые таблетки, содержащие оксикодон |
| KR101408315B1 (ko) * | 2006-08-04 | 2014-06-20 | 에씨팜 | 다층 경구 붕해 정제 |
| ES2691033T3 (es) | 2007-02-11 | 2018-11-23 | Map Pharmaceuticals Inc. | Método de administración terapéutica de DHE para activar el alivio rápido de la migraña a la vez que se reduce al mínimo el perfil de los efectos secundarios |
| UY32836A (es) | 2009-08-12 | 2011-03-31 | Bayer Schering Pharma Ag | Partículas estabilizadas que comprenden 5-metil-(6s)-tetrahidrofolato |
| KR20120056824A (ko) | 2009-08-19 | 2012-06-04 | 바이엘 파마 악티엔게젤샤프트 | 소아과 용도를 위한 약물 전달 시스템 （웨이퍼） |
| WO2011042897A1 (en) * | 2009-10-05 | 2011-04-14 | Yissum Research Development Company Of The Hebrew University Of Jerusalem, Ltd | Liquid precursor compositions and uses thereof for a ph-dependant sustained release treatment of oral disorders |
| MX350838B (es) | 2011-02-11 | 2017-09-18 | Grain Proc Corporation * | Composicion de sal. |
| FR3078630B1 (fr) | 2018-03-08 | 2021-05-14 | Karim Ioualalen | Mode de formulation sous forme de solide divise hydrophobe |
| FR3079146B1 (fr) | 2018-03-23 | 2020-04-17 | Karim Ioualalen | Formulation gastroprotectrice de complexes d’enzymes permettant de restaurer la fonction digestive. |
| CN110755404B (zh) * | 2019-12-04 | 2022-03-08 | 长春雷允上药业有限公司 | 一种阿奇霉素药物组合物及其制备方法 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5516524A (en) * | 1993-12-20 | 1996-05-14 | The Procter & Gamble Company | Laxative compositions containing bulk fiber |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8623557D0 (en) * | 1986-10-01 | 1986-11-05 | Boots Co Plc | Therapeutic agents |
| SE8605515D0 (sv) * | 1986-12-22 | 1986-12-22 | Astra Laekemedel Ab | A liquid dosage form for oral administration of a pharmaceutically active substance |
| US5004595A (en) * | 1986-12-23 | 1991-04-02 | Warner-Lambert Company | Multiple encapsulated flavor delivery system and method of preparation |
| US4874613A (en) * | 1987-03-06 | 1989-10-17 | Baker Cummins Pharmaceuticals, Inc. | Taste concealing pharmaceutical dosage unit |
| US5234957A (en) | 1991-02-27 | 1993-08-10 | Noven Pharmaceuticals, Inc. | Compositions and methods for topical administration of pharmaceutically active agents |
| US5026559A (en) * | 1989-04-03 | 1991-06-25 | Kinaform Technology, Inc. | Sustained-release pharmaceutical preparation |
| US4966770A (en) * | 1989-07-26 | 1990-10-30 | Himedics, Inc. | Prednisone microencapsulated granules |
| US5527545A (en) * | 1989-09-18 | 1996-06-18 | Recordati S.A. Chemical And Pharmaceutical Company | Liquid-suspension controlled-release pharmaceutical composition |
| US5614222A (en) * | 1994-10-25 | 1997-03-25 | Kaplan; Milton R. | Stable aqueous drug suspensions and methods for preparation thereof |
| US5529783A (en) * | 1994-12-19 | 1996-06-25 | Mcneil-Ppc, Inc. | Rotor granulation and coating of acetaminophen, pseudoephedrine, chlorpheniramine, and, optionally dextromethorphan |
| CN1244119A (zh) * | 1997-01-06 | 2000-02-09 | 辉瑞大药厂 | 迅速释放和掩蔽味觉的药物剂型 |
| US6289180B1 (en) * | 1997-12-08 | 2001-09-11 | Intel Corporation | Photoflash charging circuit with current and voltage monitor |
-
1999
- 1999-11-24 EP EP10010237.5A patent/EP2260836B1/en not_active Expired - Lifetime
- 1999-11-24 AU AU19220/00A patent/AU753476B2/en not_active Ceased
- 1999-11-24 WO PCT/US1999/027981 patent/WO2000030617A1/en not_active Ceased
- 1999-11-24 JP JP2000583501A patent/JP2002530322A/ja active Pending
- 1999-11-24 CA CA002351720A patent/CA2351720C/en not_active Expired - Fee Related
- 1999-11-24 ES ES10010237.5T patent/ES2601855T3/es not_active Expired - Lifetime
- 1999-11-24 EP EP99962868A patent/EP1133282A4/en not_active Withdrawn
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5516524A (en) * | 1993-12-20 | 1996-05-14 | The Procter & Gamble Company | Laxative compositions containing bulk fiber |
Also Published As
| Publication number | Publication date |
|---|---|
| HK1146901A1 (en) | 2011-07-22 |
| CA2351720A1 (en) | 2000-06-02 |
| EP1133282A4 (en) | 2006-03-29 |
| EP2260836B1 (en) | 2016-08-10 |
| EP2260836A3 (en) | 2012-02-01 |
| EP1133282A1 (en) | 2001-09-19 |
| JP2002530322A (ja) | 2002-09-17 |
| AU1922000A (en) | 2000-06-13 |
| CA2351720C (en) | 2006-11-21 |
| ES2601855T3 (es) | 2017-02-16 |
| EP2260836A2 (en) | 2010-12-15 |
| WO2000030617A9 (en) | 2000-11-23 |
| WO2000030617A1 (en) | 2000-06-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FGA | Letters patent sealed or granted (standard patent) | ||
| NB | Applications allowed - extensions of time section 223(2) |
Free format text: THE TIME IN WHICH TO PROVIDE SEARCH RESULTS UNDER S45(3) HAS BEEN EXTENDED TO 20040401 |
|
| MK14 | Patent ceased section 143(a) (annual fees not paid) or expired |