AU656217B2 - Use of quinozilinederivatives as orexigenics - Google Patents

Use of quinozilinederivatives as orexigenics

Info

Publication number
AU656217B2
AU656217B2 AU23719/92A AU2371992A AU656217B2 AU 656217 B2 AU656217 B2 AU 656217B2 AU 23719/92 A AU23719/92 A AU 23719/92A AU 2371992 A AU2371992 A AU 2371992A AU 656217 B2 AU656217 B2 AU 656217B2
Authority
AU
Australia
Prior art keywords
alkyl
endo
hydrogen
compounds
quinolizin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU23719/92A
Other languages
English (en)
Other versions
AU2371992A (en
Inventor
John T Burke
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharmaceuticals Inc
Original Assignee
Merrell Dow Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharmaceuticals Inc filed Critical Merrell Dow Pharmaceuticals Inc
Publication of AU2371992A publication Critical patent/AU2371992A/en
Application granted granted Critical
Publication of AU656217B2 publication Critical patent/AU656217B2/en
Assigned to MERRELL PHARMACEUTICALS INC. reassignment MERRELL PHARMACEUTICALS INC. Request to Amend Deed and Register Assignors: MERRELL DOW PHARMACEUTICALS INC.
Assigned to AVENTIS INC. reassignment AVENTIS INC. Alteration of Name(s) in Register under S187 Assignors: MERRELL PHARMACEUTICALS INC.
Assigned to AVENTISUB II INC. reassignment AVENTISUB II INC. Alteration of Name(s) in Register under S187 Assignors: AVENTIS INC.
Anticipated expiration legal-status Critical
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Child & Adolescent Psychology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Compounds Of Alkaline-Earth Elements, Aluminum Or Rare-Earth Metals (AREA)
  • Manufacture And Refinement Of Metals (AREA)
AU23719/92A 1991-08-09 1992-07-09 Use of quinozilinederivatives as orexigenics Expired AU656217B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US74295191A 1991-08-09 1991-08-09
US742951 1991-08-09
PCT/US1992/005809 WO1993002678A1 (fr) 1991-08-09 1992-07-09 Utilisation de derives de quinoziline en tant qu'orexigenes

Publications (2)

Publication Number Publication Date
AU2371992A AU2371992A (en) 1993-03-02
AU656217B2 true AU656217B2 (en) 1995-01-27

Family

ID=24986902

Family Applications (1)

Application Number Title Priority Date Filing Date
AU23719/92A Expired AU656217B2 (en) 1991-08-09 1992-07-09 Use of quinozilinederivatives as orexigenics

Country Status (8)

Country Link
US (1) US5352686A (fr)
EP (1) EP0599878A1 (fr)
JP (1) JPH06509795A (fr)
AU (1) AU656217B2 (fr)
HU (1) HUT66138A (fr)
NZ (1) NZ243833A (fr)
PT (1) PT100743B (fr)
WO (1) WO1993002678A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0831835B1 (fr) * 1995-06-01 2002-10-30 Eli Lilly And Company Traitement de l'anorexie

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4906755A (en) * 1986-11-03 1990-03-06 Merrell Dow Pharmaceuticals Inc. Esters of hexahydro-8-hydroxy-2,6-methano-2H-quinolizin-3-(4H)-one and related compounds

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4906755A (en) * 1986-11-03 1990-03-06 Merrell Dow Pharmaceuticals Inc. Esters of hexahydro-8-hydroxy-2,6-methano-2H-quinolizin-3-(4H)-one and related compounds

Also Published As

Publication number Publication date
AU2371992A (en) 1993-03-02
EP0599878A1 (fr) 1994-06-08
JPH06509795A (ja) 1994-11-02
PT100743A (pt) 1993-10-29
NZ243833A (en) 1997-03-24
US5352686A (en) 1994-10-04
HUT66138A (en) 1994-09-28
HU9400358D0 (en) 1994-05-30
WO1993002678A1 (fr) 1993-02-18
PT100743B (pt) 1999-10-29

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Legal Events

Date Code Title Description
HB Alteration of name in register

Owner name: MERRELL PHARMACEUTICALS INC.

Free format text: FORMER NAME WAS: MERRELL DOW PHARMACEUTICALS INC.

MK14 Patent ceased section 143(a) (annual fees not paid) or expired
NA Applications received for extensions of time, section 223

Free format text: AN APPLICATION TO EXTEND THE TIME FROM 20010709 TO 20040609 IN WHICH TO PAY A RENEWAL FEE HAS BEEN LODGED

NB Applications allowed - extensions of time section 223(2)

Free format text: THE TIME IN WHICH TO PAY A RENEWAL FEE HAS BEEN EXTENDED TO 20040609