AU6178894A - Alkanesulfonamido-1-indanone derivatives as inhibitors of cyclooxygenase - Google Patents

Alkanesulfonamido-1-indanone derivatives as inhibitors of cyclooxygenase

Info

Publication number
AU6178894A
AU6178894A AU61788/94A AU6178894A AU6178894A AU 6178894 A AU6178894 A AU 6178894A AU 61788/94 A AU61788/94 A AU 61788/94A AU 6178894 A AU6178894 A AU 6178894A AU 6178894 A AU6178894 A AU 6178894A
Authority
AU
Australia
Prior art keywords
alkanesulfonamido
cyclooxygenase
inhibitors
indanone derivatives
indanone
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU61788/94A
Inventor
Cameron W Black
Daniel Guay
Chun-Sing Li
Petpiboon Prasit
Patrick Roy
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Frosst Canada and Co
Original Assignee
Merck Frosst Canada and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Frosst Canada and Co filed Critical Merck Frosst Canada and Co
Publication of AU6178894A publication Critical patent/AU6178894A/en
Priority to AU36139/95A priority Critical patent/AU715676B2/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/38—One sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/36—Sulfur atoms
AU61788/94A 1993-03-12 1994-03-10 Alkanesulfonamido-1-indanone derivatives as inhibitors of cyclooxygenase Abandoned AU6178894A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU36139/95A AU715676B2 (en) 1993-03-12 1995-10-09 Use of inhibitors of cyclooxygenase in the treatment of neurodegenerative diseases

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/030,924 US5409944A (en) 1993-03-12 1993-03-12 Alkanesulfonamido-1-indanone derivatives as inhibitors of cyclooxygenase
US030924 1993-03-12
PCT/CA1994/000135 WO1994020480A1 (en) 1993-03-12 1994-03-10 Alkanesulfonamido-1-indanone derivatives as inhibitors of cyclooxygenase

Related Child Applications (1)

Application Number Title Priority Date Filing Date
AU36139/95A Division AU715676B2 (en) 1993-03-12 1995-10-09 Use of inhibitors of cyclooxygenase in the treatment of neurodegenerative diseases

Publications (1)

Publication Number Publication Date
AU6178894A true AU6178894A (en) 1994-09-26

Family

ID=21856726

Family Applications (1)

Application Number Title Priority Date Filing Date
AU61788/94A Abandoned AU6178894A (en) 1993-03-12 1994-03-10 Alkanesulfonamido-1-indanone derivatives as inhibitors of cyclooxygenase

Country Status (4)

Country Link
US (1) US5409944A (en)
AU (1) AU6178894A (en)
CA (1) CA2157107C (en)
WO (1) WO1994020480A1 (en)

Families Citing this family (163)

* Cited by examiner, † Cited by third party
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