AU5892490A - Thienodiazepine derivatives - Google Patents
Thienodiazepine derivativesInfo
- Publication number
- AU5892490A AU5892490A AU58924/90A AU5892490A AU5892490A AU 5892490 A AU5892490 A AU 5892490A AU 58924/90 A AU58924/90 A AU 58924/90A AU 5892490 A AU5892490 A AU 5892490A AU 5892490 A AU5892490 A AU 5892490A
- Authority
- AU
- Australia
- Prior art keywords
- thienodiazepine
- derivatives
- thienodiazepine derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/49—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reaction with carbon monoxide
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE3922944 | 1989-07-12 | ||
DE3922944 | 1989-07-12 | ||
DE4011345 | 1990-04-07 | ||
DE4011345 | 1990-04-07 |
Publications (2)
Publication Number | Publication Date |
---|---|
AU5892490A true AU5892490A (en) | 1991-01-17 |
AU636155B2 AU636155B2 (en) | 1993-04-22 |
Family
ID=25882911
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU58924/90A Expired - Fee Related AU636155B2 (en) | 1989-07-12 | 1990-07-12 | Thienodiazepine derivatives |
Country Status (14)
Country | Link |
---|---|
EP (1) | EP0407955A1 (en) |
JP (1) | JPH03215489A (en) |
KR (1) | KR910002863A (en) |
AU (1) | AU636155B2 (en) |
CA (1) | CA2020806A1 (en) |
FI (1) | FI903509A0 (en) |
HU (1) | HUT59144A (en) |
IE (1) | IE902526A1 (en) |
IL (1) | IL95045A0 (en) |
NO (1) | NO903088L (en) |
NZ (1) | NZ234476A (en) |
PL (1) | PL286019A1 (en) |
PT (1) | PT94673A (en) |
YU (1) | YU133090A (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU621413B2 (en) * | 1988-10-31 | 1992-03-12 | Eisai Co. Ltd. | 1,4-diazepine derivative and its pharmaceutical use |
Families Citing this family (32)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE4027470A1 (en) * | 1990-08-30 | 1992-03-05 | Boehringer Ingelheim Kg | NEW HETRAZEPINOIDE AMIDE |
DE4101146A1 (en) * | 1991-01-16 | 1992-07-23 | Boehringer Ingelheim Kg | NEW DIAZEPINE SUBSTITUTED IN 6-POSITION, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS A MEDICAMENT |
DE4107521A1 (en) * | 1991-03-08 | 1992-09-10 | Boehringer Ingelheim Kg | NEW ACYLAMINOSUBSTITUTED HETRAZEPINE |
DE69717160T2 (en) * | 1996-09-13 | 2003-05-08 | Mitsubishi Pharma Corp | THIENOTRIAZOLODIAZEPINE COMPOUNDS AND THEIR MEDICAL APPLICATIONS |
US5939432A (en) | 1997-10-29 | 1999-08-17 | Medco Research, Inc. | Thiophenes useful for modulating the adenosine receptor |
US6323214B1 (en) | 1997-10-29 | 2001-11-27 | Medco Research, Inc | Allosteric adenosine receptor modulators |
US6727258B2 (en) | 1997-10-29 | 2004-04-27 | King Pharmaceutical Research & Development, Inc. | Allosteric adenosine receptor modulators |
US6184226B1 (en) | 1998-08-28 | 2001-02-06 | Scios Inc. | Quinazoline derivatives as inhibitors of P-38 α |
JP5008796B2 (en) * | 2001-01-19 | 2012-08-22 | ダイト株式会社 | Method for producing aromatic carboxylic acid |
JP5159305B2 (en) * | 2005-05-30 | 2013-03-06 | 田辺三菱製薬株式会社 | Thienotriazolodiazepine compounds and their use as pharmaceuticals |
ES2534521T3 (en) | 2010-05-14 | 2015-04-23 | Dana-Farber Cancer Institute, Inc. | Compositions and their use in the treatment of neoplasia, inflammatory diseases and other diseases |
EP2571875A4 (en) | 2010-05-14 | 2013-10-30 | Dana Farber Cancer Inst Inc | Male contraceptive compositions and methods of use |
AU2011252799B2 (en) | 2010-05-14 | 2015-05-14 | Cold Spring Harbor Laboratory | Compositions and methods for treating leukemia |
AR084070A1 (en) | 2010-12-02 | 2013-04-17 | Constellation Pharmaceuticals Inc | BROMODOMINIUM INHIBITORS AND USES OF THE SAME |
WO2012075456A1 (en) | 2010-12-02 | 2012-06-07 | Constellation Pharmaceuticals | Bromodomain inhibitors and uses thereof |
WO2012151512A2 (en) | 2011-05-04 | 2012-11-08 | Constellation Pharmaceuticals, Inc. | Bromodomain inhibitors and uses thereof |
EP2721031B1 (en) | 2011-06-17 | 2016-01-20 | Constellation Pharmaceuticals, Inc. | Bromodomain inhibitors and uses thereof |
TWI602820B (en) | 2012-06-06 | 2017-10-21 | 星宿藥物公司 | Bromodomain inhibitors and uses thereof |
EP2864336B1 (en) | 2012-06-06 | 2016-11-23 | Constellation Pharmaceuticals, Inc. | Benzo[b]isoxazoloazepine bromodomain inhibitors and uses thereof |
KR20160034379A (en) | 2013-07-25 | 2016-03-29 | 다나-파버 캔서 인스티튜트 인크. | Inhibitors of transcription factors and uses thereof |
CN105849110B (en) | 2013-11-08 | 2019-08-02 | 达纳-法伯癌症研究所有限公司 | Use the combination treatment for cancer of bromine structural domain and additional terminals (BET) protein inhibitor |
US10793571B2 (en) | 2014-01-31 | 2020-10-06 | Dana-Farber Cancer Institute, Inc. | Uses of diazepane derivatives |
CA2936865A1 (en) | 2014-01-31 | 2015-08-06 | Dana-Farber Cancer Institute, Inc. | Diaminopyrimidine benzenesulfone derivatives and uses thereof |
MX2016011160A (en) | 2014-02-28 | 2017-04-27 | Tensha Therapeutics Inc | Treatment of conditions associated with hyperinsulinaemia. |
CA2952830C (en) | 2014-06-20 | 2022-11-01 | Constellation Pharmaceuticals, Inc. | Crystalline forms of 2-((4s)-6-(4-chlorophenyl)-1-methyl-4h-benzo[c]isoxazolo[4,5-e]azepin-4-yl)acetamide |
WO2016022970A1 (en) | 2014-08-08 | 2016-02-11 | Dana-Farber Cancer Institute, Inc. | Dihydropteridinone derivatives and uses thereof |
CN106715437A (en) | 2014-08-08 | 2017-05-24 | 达纳-法伯癌症研究所股份有限公司 | Diazepane derivatives and uses thereof |
EP3212654B1 (en) | 2014-10-27 | 2020-04-08 | Tensha Therapeutics, Inc. | Bromodomain inhibitors |
US10702527B2 (en) | 2015-06-12 | 2020-07-07 | Dana-Farber Cancer Institute, Inc. | Combination therapy of transcription inhibitors and kinase inhibitors |
CN108472300A (en) | 2015-09-11 | 2018-08-31 | 达纳-法伯癌症研究所股份有限公司 | Cyano thiophene and triazol diazacyclo heptantriene and application thereof |
JP2018526424A (en) | 2015-09-11 | 2018-09-13 | ダナ−ファーバー キャンサー インスティテュート, インコーポレイテッド | Acetamidhienotriazolodiazepines and their use |
SG10201913450PA (en) | 2015-11-25 | 2020-03-30 | Dana Farber Cancer Inst Inc | Bivalent bromodomain inhibitors and uses thereof |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2712951A1 (en) * | 1977-03-24 | 1978-10-05 | Bosch Gmbh Robert | BIMETAL WITH AN ELECTRIC HEATING ELEMENT |
DE3701344A1 (en) * | 1986-01-21 | 1987-07-23 | Boehringer Ingelheim Kg | Novel thieno-1,4-diazepines |
DE3778559D1 (en) * | 1986-01-21 | 1992-06-04 | Boehringer Ingelheim Kg | THIENO-1,4-DIAZEPINE. |
DE3610848A1 (en) * | 1986-04-01 | 1987-10-15 | Boehringer Ingelheim Kg | NEW 1,4-DIAZEPINE |
DE3724031A1 (en) * | 1986-07-22 | 1988-01-28 | Boehringer Ingelheim Kg | Novel hetrazepines and process for their preparation |
DE3624779C2 (en) * | 1986-07-22 | 1996-03-07 | Boehringer Ingelheim Kg | Process for the preparation of thieno-triazolo-1,4-diazepino-2-carboxylic acid amides |
-
1990
- 1990-07-10 EP EP90113130A patent/EP0407955A1/en not_active Withdrawn
- 1990-07-10 YU YU133090A patent/YU133090A/en unknown
- 1990-07-10 CA CA002020806A patent/CA2020806A1/en not_active Abandoned
- 1990-07-11 PL PL28601990A patent/PL286019A1/en unknown
- 1990-07-11 IE IE252690A patent/IE902526A1/en unknown
- 1990-07-11 NO NO90903088A patent/NO903088L/en unknown
- 1990-07-11 JP JP2183872A patent/JPH03215489A/en active Pending
- 1990-07-11 FI FI903509A patent/FI903509A0/en not_active IP Right Cessation
- 1990-07-11 KR KR1019900010441A patent/KR910002863A/en not_active Application Discontinuation
- 1990-07-11 IL IL95045A patent/IL95045A0/en unknown
- 1990-07-11 HU HU904169A patent/HUT59144A/en unknown
- 1990-07-12 NZ NZ234476A patent/NZ234476A/en unknown
- 1990-07-12 PT PT94673A patent/PT94673A/en not_active Application Discontinuation
- 1990-07-12 AU AU58924/90A patent/AU636155B2/en not_active Expired - Fee Related
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU621413B2 (en) * | 1988-10-31 | 1992-03-12 | Eisai Co. Ltd. | 1,4-diazepine derivative and its pharmaceutical use |
Also Published As
Publication number | Publication date |
---|---|
HUT59144A (en) | 1992-04-28 |
KR910002863A (en) | 1991-02-26 |
EP0407955A1 (en) | 1991-01-16 |
CA2020806A1 (en) | 1991-01-13 |
NZ234476A (en) | 1992-08-26 |
IE902526A1 (en) | 1991-02-13 |
NO903088L (en) | 1991-01-14 |
PT94673A (en) | 1991-03-20 |
NO903088D0 (en) | 1990-07-11 |
IL95045A0 (en) | 1991-06-10 |
AU636155B2 (en) | 1993-04-22 |
YU133090A (en) | 1993-10-20 |
JPH03215489A (en) | 1991-09-20 |
PL286019A1 (en) | 1991-10-21 |
HU904169D0 (en) | 1990-12-28 |
FI903509A0 (en) | 1990-07-11 |
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