AU5634386A - Process for preparing (z)-1-phenyl-1-diethylaminocarbonyl-2- aminomethylcyclopropane hydrochloride - Google Patents

Process for preparing (z)-1-phenyl-1-diethylaminocarbonyl-2- aminomethylcyclopropane hydrochloride

Info

Publication number
AU5634386A
AU5634386A AU56343/86A AU5634386A AU5634386A AU 5634386 A AU5634386 A AU 5634386A AU 56343/86 A AU56343/86 A AU 56343/86A AU 5634386 A AU5634386 A AU 5634386A AU 5634386 A AU5634386 A AU 5634386A
Authority
AU
Australia
Prior art keywords
diethylaminocarbonyl
phenyl
preparing
aminomethylcyclopropane hydrochloride
aminomethylcyclopropane
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU56343/86A
Other versions
AU587613B2 (en
Inventor
Bernard Bonnaud
Henri Cousse
Gilbert Mouzin
Jean-Francois Patoiseau
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pierre Fabre Medicament SA
Original Assignee
Pierre Fabre Medicament SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9318686&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU5634386(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pierre Fabre Medicament SA filed Critical Pierre Fabre Medicament SA
Publication of AU5634386A publication Critical patent/AU5634386A/en
Application granted granted Critical
Publication of AU587613B2 publication Critical patent/AU587613B2/en
Anticipated expiration legal-status Critical
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/24—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/12—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups
AU56343/86A 1985-04-25 1986-04-17 Process for preparing (z)-1-phenyl-1-diethylaminocarbonyl-2- aminomethylcyclopropane hydrochloride Expired AU587613B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8506335A FR2581059B1 (en) 1985-04-25 1985-04-25 PROCESS FOR THE PREPARATION OF PHENYL-1 HYDROCHLORIDE DIETHYL AMINO CARBONYL-1 AMINOMETHYL-2 CYCLOPROPANE (Z)
FR8506335 1985-04-25

Publications (2)

Publication Number Publication Date
AU5634386A true AU5634386A (en) 1986-10-30
AU587613B2 AU587613B2 (en) 1989-08-24

Family

ID=9318686

Family Applications (1)

Application Number Title Priority Date Filing Date
AU56343/86A Expired AU587613B2 (en) 1985-04-25 1986-04-17 Process for preparing (z)-1-phenyl-1-diethylaminocarbonyl-2- aminomethylcyclopropane hydrochloride

Country Status (23)

Country Link
EP (1) EP0200638B1 (en)
JP (1) JPS61251650A (en)
KR (1) KR940006764B1 (en)
AR (1) AR240695A1 (en)
AT (1) ATE42273T1 (en)
AU (1) AU587613B2 (en)
CA (1) CA1266486A (en)
DE (1) DE3662877D1 (en)
DK (1) DK170888B1 (en)
ES (1) ES8704449A1 (en)
FI (1) FI87196C (en)
FR (1) FR2581059B1 (en)
GE (1) GEP19970789B (en)
GR (1) GR860980B (en)
HU (1) HU195182B (en)
IE (1) IE59015B1 (en)
MX (1) MX162896B (en)
NO (1) NO165143C (en)
OA (1) OA08241A (en)
PT (1) PT82461B (en)
SU (1) SU1443797A3 (en)
YU (1) YU44915B (en)
ZA (1) ZA862929B (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7592485B2 (en) 2004-06-24 2009-09-22 Sumitomo Chemical Company, Limited Process for producing (Z)-1-phenyl-1-diethylaminocarbonyl-2-aminomethylcyclopropane hydrochloride
CN104058992A (en) * 2014-06-13 2014-09-24 上海现代制药股份有限公司 Crystal form of levomilnacipran hydrochloride

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2640972B1 (en) * 1988-12-28 1991-04-19 Pf Medicament
US5621142A (en) * 1994-02-22 1997-04-15 Asahi Kasei Kogyo Kabushiki Kaisha Aminoalkylcyclopropane derivatives
FR2752732B1 (en) * 1996-08-28 1998-11-20 Pf Medicament EXTENDED RELEASE GALENIC FORM OF MILNACIPRAN
JP4828863B2 (en) * 2005-01-28 2011-11-30 住友化学株式会社 Process for producing (Z) -1-phenyl-1- (N, N-diethylaminocarbonyl) -2-phthalimidomethylcyclopropane
US8309128B2 (en) 2005-06-10 2012-11-13 Pierre Fabre Medicament Stabilized milnacipran formulation
KR100772244B1 (en) * 2005-07-20 2007-11-01 안국약품 주식회사 Method for the preparation of milnacipran hydrogen chloride salt
SG160362A1 (en) * 2006-04-17 2010-04-29 Sumitomo Chemical Co Cyclic carboxylic acid
JP5338035B2 (en) * 2006-04-17 2013-11-13 住友化学株式会社 Process for producing polycyclic lactams
EP2114868A2 (en) * 2007-02-28 2009-11-11 Ranbaxy Laboratories Limited Novel polymorphic forms of milnacipran hydrochloride
FR2941454B1 (en) 2009-01-29 2011-04-01 Pf Medicament PROCESS FOR THE SYNTHESIS OF (1S, 2R) -MILNACIPRAN
US20100274050A1 (en) * 2009-04-23 2010-10-28 Glenmark Generics Limited Solid milnacipran and process for the preparation of the same
US20140045936A1 (en) 2011-04-21 2014-02-13 Wake Forest University Health Sciences Cyclopropyl derivatives and methods of use
CN103242289B (en) * 2012-02-03 2015-01-07 暨明医药科技（苏州）有限公司 Preparation method of N,N-diallyl-(1R,2R)-2-aminomethyl-1-(2-thienyl)cyclopropanecarboxamide hydrochloride
WO2014009767A1 (en) 2012-07-07 2014-01-16 Micro Labs Limited An improved process for the preparation of 1-aryl 2-aminomethyl cyclopropane carboxyamide (z) derivatives, their isomers and salts
EP2906518A4 (en) 2012-10-09 2016-07-27 California Inst Of Techn In vivo and in vitro olefin cyclopropanation catalyzed by heme enzymes
FR2998892B1 (en) * 2012-12-04 2015-01-02 Pf Medicament AMINOCYCLOBUTANE DERIVATIVES, PROCESS FOR PREPARING THEM AND THEIR USE AS MEDICAMENTS
CN103613513B (en) * 2013-12-09 2016-01-20 上海现代制药股份有限公司 Milnacipran hydrochloride intermediate and its preparation method and application
US9399762B2 (en) 2014-02-18 2016-07-26 California Institute Of Technology Methods and systems for sulfimidation or sulfoximidation of organic molecules
WO2016071303A1 (en) 2014-11-04 2016-05-12 Quimica Sintetica, S.A. Process for the preparation of (1s,2r)-milnacipran

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2508035A1 (en) * 1981-06-23 1982-12-24 Fabre Sa Pierre ARYL-1-AMINOMETHYL-2 CYCLOPROPANES CARBOXAMIDE (Z) DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICAMENTS USEFUL IN THE TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7592485B2 (en) 2004-06-24 2009-09-22 Sumitomo Chemical Company, Limited Process for producing (Z)-1-phenyl-1-diethylaminocarbonyl-2-aminomethylcyclopropane hydrochloride
CN104058992A (en) * 2014-06-13 2014-09-24 上海现代制药股份有限公司 Crystal form of levomilnacipran hydrochloride

Also Published As

Publication number Publication date
ZA862929B (en) 1986-12-30
KR860008126A (en) 1986-11-12
DK191286D0 (en) 1986-04-24
HU195182B (en) 1988-04-28
NO165143C (en) 1991-01-09
FR2581059A1 (en) 1986-10-31
FR2581059B1 (en) 1988-04-22
FI87196C (en) 1992-12-10
NO165143B (en) 1990-09-24
GEP19970789B (en) 1997-01-28
SU1443797A3 (en) 1988-12-07
DK170888B1 (en) 1996-03-04
AR240695A1 (en) 1990-09-28
ATE42273T1 (en) 1989-05-15
ES8704449A1 (en) 1987-04-01
PT82461B (en) 1988-10-14
AU587613B2 (en) 1989-08-24
CA1266486A (en) 1990-03-06
ES554321A0 (en) 1987-04-01
JPS61251650A (en) 1986-11-08
EP0200638A1 (en) 1986-11-05
IE59015B1 (en) 1993-12-15
PT82461A (en) 1986-05-01
NO861573L (en) 1986-10-27
IE861057L (en) 1986-10-25
HUT40618A (en) 1987-01-28
GR860980B (en) 1986-08-25
JPH0567136B2 (en) 1993-09-24
OA08241A (en) 1987-10-30
MX162896B (en) 1991-07-08
EP0200638B1 (en) 1989-04-19
DK191286A (en) 1986-10-26
FI87196B (en) 1992-08-31
FI861755A0 (en) 1986-04-25
YU65586A (en) 1987-12-31
DE3662877D1 (en) 1989-05-24
KR940006764B1 (en) 1994-07-27
FI861755A (en) 1986-10-26
YU44915B (en) 1991-04-30

Similar Documents

Publication Publication Date Title
EP0215379A3 (en) Process for preparing polyvinylpyrrolidone
AU587613B2 (en) Process for preparing (z)-1-phenyl-1-diethylaminocarbonyl-2- aminomethylcyclopropane hydrochloride
AU586469B2 (en) Process for preparing unsaturated flouroelastomers
HUT42441A (en) Process for preparing indolyl- and indazolyl-carboxamide derivatives
EP0199997A3 (en) Process for preparing diaryl-pentaerythritol
PT82445A (en) Process for preparing novel glycopeptide derivatives
HUT42500A (en) New process for preparing sphyngosine derivatives
AU591537B2 (en) Process for preparing l-rhamnose
PT83293B (en) Process for preparing dihidropyridine-2-hydroxyamines useful asmedicaments
PT83154A (en) Process for preparing quinolizinesulphonamides
ZA863454B (en) Process for preparing benzothiazolesulphenamides
HUT42766A (en) Process for preparing n-sulfamyl-3-(2-guanidino-thiazolyl-4-methyl-thio)-propionamidine
AU588017B2 (en) Process for preparing 4,4-dialkyl-2-axetidinones
AU583451B2 (en) Process for making alumina
PT81988A (en) Process for preparing novel alkylamino-furanone derivatives
HUT40445A (en) Process for preparing 2-bromo-alpha-ergochristine
HUT43022A (en) Process for preparing monochloro-pinacolone
PT84031A (en) Process for preparing 1-carbacephalosporin antibiotics
HUT42432A (en) Process for preparing substituted phenyl-carbamide derivatives
HUT43039A (en) Process for preparing 4-hydroxy-2-oxo-pyrrolidin-1-yl-acetamide
HUT42769A (en) Process for preparing pyridazodiazepines
PT82643A (en) Process for preparing substituted hexanydro arylquinolizines
HUT42438A (en) Process for preparing novel 4-alkoxy-2-oxo-pyrrolidin-1-yl-acetic acid-alkylesters
HUT42066A (en) Process for preparing 4-phenyl-propyl-indole derivatives
AU1210488A (en) Method for preparing aminohydrocarbyl-substituted ketoximosilanes