AU547922B2 - Benzazole derivatives with antiparasitic action - Google Patents

Benzazole derivatives with antiparasitic action

Info

Publication number
AU547922B2
AU547922B2 AU70910/81A AU7091081A AU547922B2 AU 547922 B2 AU547922 B2 AU 547922B2 AU 70910/81 A AU70910/81 A AU 70910/81A AU 7091081 A AU7091081 A AU 7091081A AU 547922 B2 AU547922 B2 AU 547922B2
Authority
AU
Australia
Prior art keywords
benzazole derivatives
antiparasitic action
antiparasitic
action
benzazole
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU70910/81A
Other languages
English (en)
Other versions
AU7091081A (en
Inventor
Jean Jacques Gallay
Ernst Schweizer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of AU7091081A publication Critical patent/AU7091081A/en
Application granted granted Critical
Publication of AU547922B2 publication Critical patent/AU547922B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56—Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/08—Radicals containing only hydrogen and carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/10—Radicals substituted by halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU70910/81A 1980-05-22 1981-05-21 Benzazole derivatives with antiparasitic action Ceased AU547922B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH4016/80 1980-05-22
CH401680 1980-05-22

Publications (2)

Publication Number Publication Date
AU7091081A AU7091081A (en) 1981-11-26
AU547922B2 true AU547922B2 (en) 1985-11-14

Family

ID=4268232

Family Applications (1)

Application Number Title Priority Date Filing Date
AU70910/81A Ceased AU547922B2 (en) 1980-05-22 1981-05-21 Benzazole derivatives with antiparasitic action

Country Status (28)

Country Link
US (1) US4511567A (OSRAM)
EP (1) EP0041046B1 (OSRAM)
JP (1) JPS5718670A (OSRAM)
KR (1) KR850000555B1 (OSRAM)
AU (1) AU547922B2 (OSRAM)
CY (1) CY1339A (OSRAM)
DD (1) DD159073A5 (OSRAM)
DE (1) DE3176402D1 (OSRAM)
DK (1) DK164786C (OSRAM)
ES (3) ES8300724A1 (OSRAM)
FI (1) FI75564C (OSRAM)
GB (1) GB2076399B (OSRAM)
GR (1) GR75253B (OSRAM)
HK (1) HK74686A (OSRAM)
HU (1) HU186770B (OSRAM)
IE (1) IE52426B1 (OSRAM)
IL (1) IL62928A (OSRAM)
IN (1) IN153293B (OSRAM)
KE (1) KE3645A (OSRAM)
MA (1) MA19290A1 (OSRAM)
MW (1) MW2181A1 (OSRAM)
MY (1) MY8700141A (OSRAM)
OA (1) OA06816A (OSRAM)
PH (1) PH16754A (OSRAM)
PT (1) PT73066B (OSRAM)
ZA (1) ZA8103409D (OSRAM)
ZM (1) ZM4481A1 (OSRAM)
ZW (1) ZW11981A1 (OSRAM)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8423697D0 (en) * 1984-09-19 1984-10-24 Ciba Geigy Ag Benzazole derivatives
US5246927A (en) * 1988-08-17 1993-09-21 Ciba-Geigy Corporation Benzazole derivatives, processes for their preparation containing such compounds and the use thereof
WO1992012144A1 (en) * 1990-12-28 1992-07-23 Teijin Limited Condensed benzoxa ring compound, production thereof, and pharmaceutical composition containing the same
WO1997047610A1 (en) * 1996-06-07 1997-12-18 Novartis Ag Benzazole derivatives
US6177572B1 (en) * 1997-08-20 2001-01-23 Sepracor, Inc. Solid and liquid-phase synthesis of benzoxazoles and benzothiazoles and their use
EP3235815A1 (de) * 2016-04-19 2017-10-25 Philipps-Universität Marburg Wirkstoffe gegen parasitäre helminthen

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1087561A (en) * 1963-02-16 1967-10-18 Fisons Pest Control Ltd Fluorinated benzimidazoles and compositions containing them
IE31812B1 (en) * 1967-02-03 1973-01-10 Merck & Co Inc Benzimidazole derivatives
US3646049A (en) * 1970-03-05 1972-02-29 Merck & Co Inc Acylaminobenzimidazole derivatives
US3714180A (en) * 1970-08-12 1973-01-30 Squibb & Sons Inc Sulfonyl benzimidazoles
BE792402A (fr) * 1971-12-07 1973-06-07 Ciba Geigy Composes heterocycliques azotes et medicaments anthelminthiqueset antimicrobiens qui en contiennent

Also Published As

Publication number Publication date
ES513169A0 (es) 1984-07-01
KR850000555B1 (ko) 1985-04-26
GB2076399B (en) 1983-11-02
GB2076399A (en) 1981-12-02
IN153293B (OSRAM) 1984-06-30
PT73066A (en) 1981-06-01
DK164786C (da) 1993-01-04
ZW11981A1 (en) 1981-12-16
MA19290A1 (fr) 1982-04-01
IE52426B1 (en) 1987-10-28
FI75564B (fi) 1988-03-31
IL62928A0 (en) 1981-07-31
GR75253B (OSRAM) 1984-07-13
MY8700141A (en) 1987-12-31
AU7091081A (en) 1981-11-26
CY1339A (en) 1987-01-16
IE811127L (en) 1981-11-22
ES513170A0 (es) 1983-09-01
OA06816A (fr) 1982-12-31
ES8406452A1 (es) 1984-07-01
ZA8103409D (en) 1982-06-30
DK224381A (da) 1981-11-23
DD159073A5 (de) 1983-02-16
FI811531L (fi) 1981-11-23
EP0041046A1 (de) 1981-12-02
PH16754A (en) 1984-02-15
JPH0357099B2 (OSRAM) 1991-08-30
MW2181A1 (en) 1982-10-13
IL62928A (en) 1985-03-31
ES502355A0 (es) 1982-11-01
US4511567A (en) 1985-04-16
HU186770B (en) 1985-09-30
ZM4481A1 (en) 1982-01-21
EP0041046B1 (de) 1987-09-02
HK74686A (en) 1986-10-10
FI75564C (fi) 1988-07-11
DE3176402D1 (en) 1987-10-08
JPS5718670A (en) 1982-01-30
DK164786B (da) 1992-08-17
KE3645A (en) 1986-07-11
ES8300724A1 (es) 1982-11-01
PT73066B (en) 1983-02-08
KR830006231A (ko) 1983-09-20
ES8308316A1 (es) 1983-09-01

Similar Documents

Publication Publication Date Title
AU542623B2 (en) 1-hydroxyethyl-azole derivatives
AU557689B2 (en) 1-sulfo-2-oxoazetidine derivatives
AU544723B2 (en) Imidazolylpropanol derivatives
AU7199081A (en) l
AU7551681A (en) 3-aryl-5-isothiazole derivatives
AU540898B2 (en) 17-disubstituted-androst-4-en-3-one derivatives
AU534878B2 (en) Amino-saccharide derivatives
AU544527B2 (en) Bis-carboxamide derivatives
AU554360B2 (en) S-triazinyl-aminofluorescein derivatives
AU545357B2 (en) Triazolo-benzodiazepine derivatives
AU7420281A (en) 2-substituted thio-penem derivatives
AU551238B2 (en) 1-hydroxy-2 -fluorocholecalciferol derivatives
AU538505B2 (en) Phenoxy-aminopropanol derivatives
AU541724B2 (en) 2-amino 4-pyrimidone derivatives
AU7091081A (en) Benzazole derivatives with antiparasitic action
AU7576681A (en) Isonicotinanilide derivatives
AU540239B2 (en) 2-guanidinothiazole derivatives
AU539443B2 (en) Phenoxybutyltriazole derivatives
AU6898281A (en) Biphenylyl-azolylethane derivatives
AU7596281A (en) Sydnonimined derivatives
AU7494381A (en) Fluorinated-1-azolyl-butane derivatives
AU7486481A (en) N-oxyamide derivatives
AU526941B2 (en) Pyrazole-substituted oximino-cyano-acetamide derivatives
AU6826781A (en) Steroid-spiro-oxathiazolidine derivatives
AU7776681A (en) Bisaminomethyl-anthraquinone derivatives