AU5130596A - New sulfone ester analogues of iso-clozapine and related structures: atypical neuroleptics - Google Patents

New sulfone ester analogues of iso-clozapine and related structures: atypical neuroleptics

Info

Publication number
AU5130596A
AU5130596A AU51305/96A AU5130596A AU5130596A AU 5130596 A AU5130596 A AU 5130596A AU 51305/96 A AU51305/96 A AU 51305/96A AU 5130596 A AU5130596 A AU 5130596A AU 5130596 A AU5130596 A AU 5130596A
Authority
AU
Australia
Prior art keywords
clozapine
iso
related structures
sulfone ester
atypical neuroleptics
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU51305/96A
Inventor
Peter De Boer
Yi Liao
Hakan Wikstrom
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of AU5130596A publication Critical patent/AU5130596A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D281/14—[b, e]-condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/38—[b, e]- or [b, f]-condensed with six-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D267/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D267/02—Seven-membered rings
    • C07D267/08—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D267/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D267/16—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D267/18—[b, e]-condensed
AU51305/96A 1995-03-19 1996-03-19 New sulfone ester analogues of iso-clozapine and related structures: atypical neuroleptics Abandoned AU5130596A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE9500998 1995-03-19
SE9500998A SE9500998D0 (en) 1995-03-19 1995-03-19 New sulfone ester analogues of iso-clozapine and related structures: atypical neuroleptics
PCT/SE1996/000344 WO1996029316A1 (en) 1995-03-19 1996-03-19 NEW SULFONE ESTER ANALOGUES OF iso-CLOZAPINE AND RELATED STRUCTURES: ATYPICAL NEUROLEPTICS

Publications (1)

Publication Number Publication Date
AU5130596A true AU5130596A (en) 1996-10-08

Family

ID=20397615

Family Applications (1)

Application Number Title Priority Date Filing Date
AU51305/96A Abandoned AU5130596A (en) 1995-03-19 1996-03-19 New sulfone ester analogues of iso-clozapine and related structures: atypical neuroleptics

Country Status (3)

Country Link
AU (1) AU5130596A (en)
SE (1) SE9500998D0 (en)
WO (1) WO1996029316A1 (en)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9615767D0 (en) * 1996-07-26 1996-09-04 Smithkline Beecham Plc Novel treatment
CN1247556C (en) * 1999-07-09 2006-03-29 宇部兴产株式会社 Process for producing dibenzothiazepine derivatives
US7141563B2 (en) 2000-11-03 2006-11-28 Wyeth Process for the preparation of 1, 2, 3, 4, 8, 9, 10, 10a-octahydro-7bH-cyclopenta[b] [1, 4]diazepino[6, 7, 1-hi] indole derivatives
ES2230382T3 (en) * 2000-11-03 2005-05-01 Wyeth CYCLOPENTAL (B) (1,4) DIAZPINO (6,7,1-HI) INDOLES AS 5HT2C ANTAGONISTS.
AR031202A1 (en) 2000-11-03 2003-09-10 Wyeth Corp CYCLOPENTA (B) (1,4) DIAZEPINO (6,7,1-HI) INDOLES AND DERIVATIVES
AR031199A1 (en) 2000-11-03 2003-09-10 Wyeth Corp CICLOHEPTA / B // 1,4 / DIACEPINO / 6,7,1-HI / INDOLES AND DERIVATIVES
AR031200A1 (en) 2000-11-03 2003-09-10 Wyeth Corp CYCLOCATE [B] [1,4] DIAZEPINO [6,7,1-HI] INDOLES AND DERIVATIVES
AR031195A1 (en) 2000-11-03 2003-09-10 Wyeth Corp PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 1,2,3,4,8,9,10,10A-OCTAHIDRO-7BH-CICLOPENTA (B) (1,4) DIAZEPINO (6,7,1) DIAZEPINO (6,7, 1-HI) INDOL
AR031196A1 (en) 2000-11-03 2003-09-10 Wyeth Corp PROCEDURE FOR THE PREPARATION OF CYCLOPENTA (B) (1,4) -DIAZEPINO (6,7,1-HI) INDOLES AND DERIVATIVES
TWI312781B (en) 2002-04-25 2009-08-01 [1,4]diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents
TW200307540A (en) 2002-04-25 2003-12-16 Wyeth Corp [1, 4]Diazocino[7, 8, 1-hi] indole derivatives as antipsychotic and antiobesity agents
TW200307682A (en) 2002-04-25 2003-12-16 Wyeth Corp 1,2,3,4,7,8-Hexahydro-6H-[1,4]diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents
WO2004087124A1 (en) * 2003-03-29 2004-10-14 Mitsubishi Pharma Corporation Compounds having serotonin 5-ht17 receptor antagonist activity and muscarinic m4 receptor agonist activity and their use in the treatment of psychotic disorders
ES2324713T3 (en) 2003-12-22 2009-08-13 Acadia Pharmaceuticals Inc. DIARIL ANALOGS (A, D) AMINO-SUBSTITUTED CYCLHEPTENE AS MUSCARINIC AGONISTS AND METHODS OF TREATMENT OF NEUROPSYCHIATRIC DISORDERS.
CN1913900B (en) * 2003-12-22 2010-11-24 阿卡蒂亚药品公司 Amino bustituted diaryl[a,d]cycloheptene analogs as muscarinic agonists and methods of treatment of neuropsychiatric disorders
GT200500317A (en) 2004-11-05 2006-10-27 PROCESS TO PREPARE QUINOLINE COMPOUNDS AND PRODUCTS OBTAINED FROM THEM
WO2007004234A1 (en) * 2005-07-04 2007-01-11 Usv Limited A PROCESS FOR THE PREPARATION OF 2-[2-(4-DIBENZO[b,f] [L,4] THIAZEPIN-11-yl-1- PIPERAZINYL)ETHOXY] ETHANOL FUMARATE
AR054849A1 (en) 2005-07-26 2007-07-18 Wyeth Corp DIAZEPINOQUINOLINAS, SYNTHESIS OF THE SAME, AND INTERMEDIARIES TO OBTAIN THEM
WO2007053618A1 (en) * 2005-10-31 2007-05-10 Acadia Pharmaceuticals Inc. Prodrugs of muscarinic agonists and methods of treatment of neuropsychiatric disorders

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH422793A (en) * 1961-07-20 1966-10-31 Wander Ag Dr A Process for the preparation of 11-basic substituted dibenzo (b, f) (1,4) thiazepines
IL29571A (en) * 1967-03-13 1972-04-27 Wander Ag Dr A 11-substituted dibenzo(b,f)-1,4-oxazepines,dibenzo(b,f)-1,4-thiazepines and dibenzo(b,e)-1,4-diazepines and their preparation
DK72693D0 (en) * 1993-06-18 1993-06-18 Lundbeck & Co As H COMPOUNDS

Also Published As

Publication number Publication date
WO1996029316A1 (en) 1996-09-26
SE9500998D0 (en) 1995-03-19

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