AU498132B2 - 5 - nitro - pyrimidine derivatives - Google Patents

5 - nitro - pyrimidine derivatives

Info

Publication number
AU498132B2
AU498132B2 AU81055/75A AU8105575A AU498132B2 AU 498132 B2 AU498132 B2 AU 498132B2 AU 81055/75 A AU81055/75 A AU 81055/75A AU 8105575 A AU8105575 A AU 8105575A AU 498132 B2 AU498132 B2 AU 498132B2
Authority
AU
Australia
Prior art keywords
nitro
pyrimidine derivatives
pyrimidine
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU81055/75A
Other languages
English (en)
Other versions
AU8105575A (en
Inventor
H Fischer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of AU8105575A publication Critical patent/AU8105575A/en
Application granted granted Critical
Publication of AU498132B2 publication Critical patent/AU498132B2/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
    • C07D239/545—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/553—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms with halogen atoms or nitro radicals directly attached to ring carbon atoms, e.g. fluorouracil
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/56—One oxygen atom and one sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/58—Two sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU81055/75A 1974-05-10 1975-05-12 5 - nitro - pyrimidine derivatives Expired AU498132B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CHCH6426/74 1974-05-10
CH642674A CH595061A5 (US06265458-20010724-C00056.png) 1974-05-10 1974-05-10

Publications (2)

Publication Number Publication Date
AU8105575A AU8105575A (en) 1976-11-18
AU498132B2 true AU498132B2 (en) 1979-02-15

Family

ID=4309440

Family Applications (1)

Application Number Title Priority Date Filing Date
AU81055/75A Expired AU498132B2 (en) 1974-05-10 1975-05-12 5 - nitro - pyrimidine derivatives

Country Status (14)

Country Link
US (1) US4014677A (US06265458-20010724-C00056.png)
JP (1) JPS50155624A (US06265458-20010724-C00056.png)
AT (1) AT344750B (US06265458-20010724-C00056.png)
AU (1) AU498132B2 (US06265458-20010724-C00056.png)
BE (1) BE828869A (US06265458-20010724-C00056.png)
CA (1) CA1042890A (US06265458-20010724-C00056.png)
CH (1) CH595061A5 (US06265458-20010724-C00056.png)
DE (1) DE2520381A1 (US06265458-20010724-C00056.png)
ES (1) ES437518A1 (US06265458-20010724-C00056.png)
FR (1) FR2270249B1 (US06265458-20010724-C00056.png)
GB (1) GB1501935A (US06265458-20010724-C00056.png)
IL (1) IL47256A (US06265458-20010724-C00056.png)
NL (1) NL7505503A (US06265458-20010724-C00056.png)
ZA (1) ZA752999B (US06265458-20010724-C00056.png)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU634751B2 (en) * 1989-02-22 1993-03-04 Hoechst Aktiengesellschaft Substituted pyrimidine derivatives, a process for the preparation thereof, and the use thereof as a tool

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL57416A (en) * 1978-05-30 1983-03-31 Smith Kline French Lab Nitro compounds,processes for preparing them and compositions containing them
US4405624A (en) * 1978-05-30 1983-09-20 Smith Kline & French Laboratories Limited Nitro-substituted dihydropyrroles and tetrahydropyridines, compositions, compounds, and medicinal use
US4560402A (en) * 1979-08-15 1985-12-24 Ciba Geigy Corporation 2,4-Diamo-5-(alkylsulfinyl) or alkylsulphonyl)-6-halopyrimidines
US4402730A (en) * 1980-01-25 1983-09-06 Sandoz Ltd. Pyrimidine derivatives and their use as herbicides
US4505910A (en) * 1983-06-30 1985-03-19 American Home Products Corporation Amino-pyrimidine derivatives, compositions and use
PH21918A (en) * 1983-07-25 1988-04-08 Ciba Geigy Ag N-(2-nitrophenyl)-5-aminopyrimidine derivatives,the preparation and use thereof
DE19917785A1 (de) * 1999-04-20 2000-10-26 Bayer Ag 2,4-Diamino-pyrimidin-Derivate
CN1894220B (zh) * 2003-12-19 2012-06-06 纳幕尔杜邦公司 除草的嘧啶
TWI355894B (en) * 2003-12-19 2012-01-11 Du Pont Herbicidal pyrimidines
GB0512844D0 (en) * 2005-06-23 2005-08-03 Novartis Ag Organic compounds
MX2008012995A (es) * 2006-04-10 2008-10-17 Du Pont Mezclas herbicidas.
GB0725218D0 (en) * 2007-12-24 2008-02-06 Syngenta Ltd Chemical compounds
PT2364314E (pt) * 2008-12-09 2014-06-09 Gilead Sciences Inc Moduladores de recetores toll-like
EP2229813A1 (de) * 2009-03-21 2010-09-22 Bayer CropScience AG Pyrimidin-4-ylpropandinitril-derivate, Verfahren zu deren Herstellung sowie deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3126271A (en) * 1964-03-24 Method of controlling weeds
US3118754A (en) * 1961-10-10 1964-01-21 Pfizer & Co C Process for stimulating plant growth
US3461461A (en) * 1965-11-01 1969-08-12 Upjohn Co 6-amino-4-(substituted amino)-1,2-dihydro-1-hydroxy-2-iminopyrimidines
US3806333A (en) * 1969-04-02 1974-04-23 Monsanto Chemicals Herbicidal composition and method employing pyridine derivatives
US3926997A (en) * 1971-05-17 1975-12-16 Ciba Geigy Corp 2-Alkylthio-4,6-bis(substituted amino)-5-nitropyrimidines
CH558137A (de) * 1971-05-17 1975-01-31 Ciba Geigy Ag Mittel zur beeinflussung des pflanzenwachstums.
CH574206A5 (US06265458-20010724-C00056.png) * 1972-11-16 1976-04-15 Ciba Geigy Ag

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU634751B2 (en) * 1989-02-22 1993-03-04 Hoechst Aktiengesellschaft Substituted pyrimidine derivatives, a process for the preparation thereof, and the use thereof as a tool

Also Published As

Publication number Publication date
AT344750B (de) 1978-08-10
BE828869A (fr) 1975-11-10
IL47256A0 (en) 1975-07-28
JPS50155624A (US06265458-20010724-C00056.png) 1975-12-16
CH595061A5 (US06265458-20010724-C00056.png) 1978-01-31
ATA355675A (de) 1977-12-15
IL47256A (en) 1979-01-31
GB1501935A (en) 1978-02-22
FR2270249A1 (US06265458-20010724-C00056.png) 1975-12-05
DE2520381A1 (de) 1975-11-20
US4014677A (en) 1977-03-29
AU8105575A (en) 1976-11-18
ZA752999B (en) 1976-04-28
NL7505503A (nl) 1975-11-12
FR2270249B1 (US06265458-20010724-C00056.png) 1978-09-01
ES437518A1 (es) 1977-01-01
CA1042890A (en) 1978-11-21

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