AU476694B2 - Process forthe manufacture of benzyl-pyrimidines - Google Patents

Process forthe manufacture of benzyl-pyrimidines

Info

Publication number
AU476694B2
AU476694B2 AU62755/73A AU6275573A AU476694B2 AU 476694 B2 AU476694 B2 AU 476694B2 AU 62755/73 A AU62755/73 A AU 62755/73A AU 6275573 A AU6275573 A AU 6275573A AU 476694 B2 AU476694 B2 AU 476694B2
Authority
AU
Australia
Prior art keywords
pyrimidines
benzyl
process forthe
forthe manufacture
manufacture
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU62755/73A
Other versions
AU6275573A (en
Inventor
MARCHAND; PERRY ROSEN and PIUS ANTON WEHRLI PERCY
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of AU6275573A publication Critical patent/AU6275573A/en
Application granted granted Critical
Publication of AU476694B2 publication Critical patent/AU476694B2/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/64—Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU62755/73A 1972-12-21 1973-11-21 Process forthe manufacture of benzyl-pyrimidines Expired AU476694B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31750072A 1972-12-21 1972-12-21
USUS317500 1972-12-21

Publications (2)

Publication Number Publication Date
AU6275573A AU6275573A (en) 1975-05-22
AU476694B2 true AU476694B2 (en) 1976-09-30

Family

ID=23233931

Family Applications (1)

Application Number Title Priority Date Filing Date
AU62755/73A Expired AU476694B2 (en) 1972-12-21 1973-11-21 Process forthe manufacture of benzyl-pyrimidines

Country Status (15)

Country Link
JP (1) JPS4988886A (en)
AT (1) AT339315B (en)
AU (1) AU476694B2 (en)
BE (1) BE808870A (en)
CA (1) CA986937A (en)
CH (1) CH592065A5 (en)
DE (1) DE2363533A1 (en)
DK (1) DK135531B (en)
FR (1) FR2211463B1 (en)
GB (1) GB1411170A (en)
HU (1) HU169082B (en)
IL (1) IL43658A (en)
NL (1) NL7317484A (en)
PH (1) PH12708A (en)
ZA (1) ZA738760B (en)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL122146C (en) * 1960-09-02
US3485840A (en) * 1964-11-12 1969-12-23 Hoffmann La Roche 2,4-diamino - 5 - (2',4',5'-substituted benzyl) pyrimidines,intermediates and processes
GB1407971A (en) * 1971-04-16 1975-10-01 Wellcome Found 2,4-diamino -4-3,4,5-triethoxybenzyl pyrimidine and methods of preparation therefor
BE792096A (en) * 1971-12-01 1973-05-30 Hoffmann La Roche NEW BENZYLPYRIMIDINES
BE795023A (en) * 1972-02-07 1973-08-06 Hoffmann La Roche NEW BENZYLPYRIMIDINES

Also Published As

Publication number Publication date
DK135531C (en) 1977-10-10
CA986937A (en) 1976-04-06
FR2211463A1 (en) 1974-07-19
AT339315B (en) 1977-10-10
CH592065A5 (en) 1977-10-14
NL7317484A (en) 1974-06-25
HU169082B (en) 1976-09-28
FR2211463B1 (en) 1979-05-11
IL43658A0 (en) 1974-03-14
PH12708A (en) 1979-07-20
ATA1070773A (en) 1977-02-15
JPS4988886A (en) 1974-08-24
BE808870A (en) 1974-06-20
DK135531B (en) 1977-05-16
AU6275573A (en) 1975-05-22
ZA738760B (en) 1974-08-28
IL43658A (en) 1976-12-31
DE2363533A1 (en) 1974-06-27
GB1411170A (en) 1975-10-29

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