AU4119289A - 2-amino-pyrimidine derivatives - Google Patents

2-amino-pyrimidine derivatives

Info

Publication number
AU4119289A
AU4119289A AU41192/89A AU4119289A AU4119289A AU 4119289 A AU4119289 A AU 4119289A AU 41192/89 A AU41192/89 A AU 41192/89A AU 4119289 A AU4119289 A AU 4119289A AU 4119289 A AU4119289 A AU 4119289A
Authority
AU
Australia
Prior art keywords
alkyl
denotes
alkenyl
cycloalkyl
halogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU41192/89A
Other versions
AU626913B2 (en
Inventor
Adolf Hubele
Helmut Zondler
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of AU4119289A publication Critical patent/AU4119289A/en
Application granted granted Critical
Publication of AU626913B2 publication Critical patent/AU626913B2/en
Assigned to NOVARTIS AG reassignment NOVARTIS AG Alteration of Name(s) in Register under S187 Assignors: CIBA-GEIGY AG
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

Compounds of the formula <IMAGE> in which: R1 denotes phenyl or phenyl which is monosubstituted to trisubstituted by R4; R2 denotes hydrogen, C1-C5-alkyl, C1-C5-alkyl substituted by the radicals OR5 or SR5, C3-C6-cycloalkyl, C3-C6-cycloalkyl monosubstituted to trisubstituted by C1-C4-alkyl or halogen, C2-C5-alkenyl, C2-C5-alkynyl or the formyl radical; R3 denotes hydrogen, C1-C4-alkyl, C1-C4-alkyl which is substituted by halogen, cyano or the radicals OR5 or SR5, C3-C6-cycloalkyl or C3-C6-cycloalkyl which is monosubstituted to trisubstituted by C1-C4-alkyl or halogen; R4 denotes halogen, C1-C3-alkyl, C1-C2-haloalkyl, C1-C3-alkoxy or C1-C3-haloalkoxy; R5 denotes hydrogen, C1-C5-alkyl, C3-C5-alkenyl, C3-C5-alkynyl or the radical (CH2)n-X-C1-C3-alkyl; R7 denotes the group -NH2, <IMAGE> or <IMAGE>; R8 denotes hydrogen, C1-C3-alkyl or C1-C3-haloalkyl; R9 denotes hydrogen, C1-C8-alkyl, C1-C3-alkyl substituted by hydroxyl, OR12, SR12 or N(R12)2, C3-C6-cycloalkyl, cyclopropyl substituted by SR12, C3-C10-alkenyl, C1-C3-haloalkyl, phenyl, phenyl which is monosubstituted to trisubstituted by halogen, C1-C3-alkyl, C1-C3-alkoxy, C1-C3-haloalkoxy, C1-C2-haloalkyl, hydroxyl, nitro, cyano, amino or dimethylamino, 1- or 2-naphthyl, 1-, 2- or 3-pyridyl, <IMAGE> or <IMAGE>; R8 and R9, together with the carbon atom in the radical R7, form a saturated or unsaturated ring consisting of 4 to 7 carbon atoms; R10 denotes CH(R8)R9, phenyl, C3-C5-alkenyl, C3-C5-alkynyl or cyanoalkyl having 2 or 3 carbon atoms in the alkyl radical; R11 denotes hydrogen, C1-C5-alkyl, C3-C5-alkenyl, C3-C5-alkynyl or cyanoalkyl having 2 or 3 carbon atoms in the alkyl radical; R12 denotes CH3 or C2H5; X denotes oxygen or sulphur; Z denotes O, S, NH or NCH3; and n denotes 1 to 3; including their acid addition salts and metal salt complexes, have useful microbicidal properties. The novel active compounds can be employed in plant protection for preventing the attack of crop plants by phytopathogenic microorganisms or by harmful insects and for controlling these pests.
AU41192/89A 1988-09-09 1989-09-08 2-amino-pyrimidine derivatives Ceased AU626913B2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH3371/88 1988-09-09
CH337188 1988-09-09
CH2579/89 1989-07-11
CH257989 1989-07-11

Publications (2)

Publication Number Publication Date
AU4119289A true AU4119289A (en) 1990-03-15
AU626913B2 AU626913B2 (en) 1992-08-13

Family

ID=25690828

Family Applications (1)

Application Number Title Priority Date Filing Date
AU41192/89A Ceased AU626913B2 (en) 1988-09-09 1989-09-08 2-amino-pyrimidine derivatives

Country Status (15)

Country Link
EP (1) EP0358609B1 (en)
JP (1) JP2832544B2 (en)
AT (1) ATE140699T1 (en)
AU (1) AU626913B2 (en)
BR (1) BR8904485A (en)
DE (1) DE58909704D1 (en)
DK (1) DK170336B1 (en)
ES (1) ES2090045T3 (en)
FI (1) FI98914C (en)
GR (1) GR3020621T3 (en)
HU (1) HU207998B (en)
IE (1) IE72462B1 (en)
IL (1) IL91556A (en)
NZ (1) NZ230592A (en)
PT (1) PT91648B (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU619762B2 (en) * 1987-09-28 1992-02-06 Syngenta Participations Ag Pesticides
AU632319B2 (en) * 1989-03-22 1992-12-24 Novartis Ag Pest control compositions

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0859628A (en) * 1994-08-26 1996-03-05 Sumitomo Chem Co Ltd Production of pyrimidine derivative

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL38815A0 (en) * 1971-03-05 1972-04-27 Ciba Geigy Ag Iodoethynyl compounds,their manufacture and their use
JPS55151570A (en) * 1979-05-15 1980-11-26 Takeda Chem Ind Ltd Pyrimidine derivatives, their preparation and antimicrobial for agriculture
DE3441935A1 (en) * 1984-11-16 1986-05-28 Bayer Ag, 5090 Leverkusen METHOD FOR PRODUCING 2,4-DIHYDROXYPYRIMIDINES
JPH0784445B2 (en) * 1986-12-03 1995-09-13 クミアイ化学工業株式会社 Pyrimidine derivatives and agricultural and horticultural fungicides
US4929726A (en) * 1988-02-09 1990-05-29 Georgia State University Foundation, Inc. Novel diazines and their method of preparation
EP0388838B1 (en) * 1989-03-22 1996-01-10 Ciba-Geigy Ag Parasiticide
DE4017460A1 (en) * 1989-10-10 1991-04-18 Bayer Ag New substd. sulphonyl-amidino hydrazone(s) - are defoliants, desiccants and weed killers

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU619762B2 (en) * 1987-09-28 1992-02-06 Syngenta Participations Ag Pesticides
AU632319B2 (en) * 1989-03-22 1992-12-24 Novartis Ag Pest control compositions

Also Published As

Publication number Publication date
EP0358609A2 (en) 1990-03-14
ES2090045T3 (en) 1996-10-16
IL91556A0 (en) 1990-04-29
DK170336B1 (en) 1995-08-07
IL91556A (en) 1994-01-25
FI98914B (en) 1997-05-30
FI894212A0 (en) 1989-09-06
EP0358609A3 (en) 1990-10-10
GR3020621T3 (en) 1996-10-31
JPH02115174A (en) 1990-04-27
IE72462B1 (en) 1997-04-09
BR8904485A (en) 1990-04-24
DK444189D0 (en) 1989-09-08
IE892881L (en) 1990-03-09
HU207998B (en) 1993-07-28
PT91648A (en) 1990-03-30
DE58909704D1 (en) 1996-08-29
EP0358609B1 (en) 1996-07-24
FI98914C (en) 1997-09-10
JP2832544B2 (en) 1998-12-09
PT91648B (en) 1995-05-31
AU626913B2 (en) 1992-08-13
DK444189A (en) 1990-03-10
FI894212A (en) 1990-03-10
ATE140699T1 (en) 1996-08-15
NZ230592A (en) 1992-02-25
HUT51604A (en) 1990-05-28

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